JP2010524947A5 - - Google Patents
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- Publication number
- JP2010524947A5 JP2010524947A5 JP2010504113A JP2010504113A JP2010524947A5 JP 2010524947 A5 JP2010524947 A5 JP 2010524947A5 JP 2010504113 A JP2010504113 A JP 2010504113A JP 2010504113 A JP2010504113 A JP 2010504113A JP 2010524947 A5 JP2010524947 A5 JP 2010524947A5
- Authority
- JP
- Japan
- Prior art keywords
- aryl
- cycloalkyl
- alkyl
- heterocyclic
- fused
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 *C(N(*)Cc1cc(CN(*)*)c(*C(*)=N2)c2c1)=* Chemical compound *C(N(*)Cc1cc(CN(*)*)c(*C(*)=N2)c2c1)=* 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US91298007P | 2007-04-20 | 2007-04-20 | |
| US60/912,980 | 2007-04-20 | ||
| PCT/US2008/005084 WO2008130669A1 (en) | 2007-04-20 | 2008-04-21 | Benzimidazoles and pharmaceutical compositions thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2010524947A JP2010524947A (ja) | 2010-07-22 |
| JP2010524947A5 true JP2010524947A5 (OSRAM) | 2011-06-16 |
| JP5400032B2 JP5400032B2 (ja) | 2014-01-29 |
Family
ID=39875833
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010504113A Expired - Fee Related JP5400032B2 (ja) | 2007-04-20 | 2008-04-21 | ベンズイミダゾール及びその医薬組成物 |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US8232410B2 (OSRAM) |
| EP (1) | EP2154966B1 (OSRAM) |
| JP (1) | JP5400032B2 (OSRAM) |
| CN (1) | CN101677553A (OSRAM) |
| AU (1) | AU2008242488B2 (OSRAM) |
| BR (1) | BRPI0810244A2 (OSRAM) |
| CA (1) | CA2684594C (OSRAM) |
| DK (1) | DK2154966T3 (OSRAM) |
| EA (1) | EA016726B1 (OSRAM) |
| ES (1) | ES2434693T3 (OSRAM) |
| HR (1) | HRP20131103T1 (OSRAM) |
| IN (1) | IN2009KN03959A (OSRAM) |
| MX (1) | MX2009011281A (OSRAM) |
| PL (1) | PL2154966T3 (OSRAM) |
| PT (1) | PT2154966E (OSRAM) |
| SI (1) | SI2154966T1 (OSRAM) |
| WO (1) | WO2008130669A1 (OSRAM) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8232310B2 (en) | 2006-12-29 | 2012-07-31 | Georgetown University | Targeting of EWS-FLI1 as anti-tumor therapy |
| US8039502B2 (en) | 2007-07-24 | 2011-10-18 | The Ohio State University Research Foundation | Anti-infective agents against intracellular pathogens |
| US20120108823A1 (en) | 2009-04-22 | 2012-05-03 | The Ohio State University Research Foundation | Anti-francisella agents |
| ES2548913T3 (es) | 2009-09-11 | 2015-10-21 | Probiodrug Ag | Derivados heterocíclicos como inhibidores de glutaminil ciclasa |
| WO2013116823A1 (en) * | 2012-02-02 | 2013-08-08 | The Research Foundation Of State University Of New York | Benzimidazoles and uses thereof |
| WO2013142326A1 (en) * | 2012-03-23 | 2013-09-26 | The Research Foundation Of State University Of New York | 5-carbonylamino-/(sulfonamido-) substituted benz imidazoles and use thereof treatment of tuberculosis |
| WO2013155341A1 (en) * | 2012-04-12 | 2013-10-17 | Georgetown University | Methods and compositions for treating ewings sarcoma family of tumors |
| CN103333170B (zh) * | 2013-06-14 | 2016-08-10 | 清华大学 | 苯并咪唑类化合物及其用途 |
| CA2927148A1 (en) | 2013-10-24 | 2015-04-30 | Georgetown University | Methods and compositions for treating cancer |
| CN106061951A (zh) * | 2013-11-22 | 2016-10-26 | 纽约州立大学研究基金会 | 苯并咪唑及其在结核病治疗中的用途 |
| WO2015138611A2 (en) | 2014-03-11 | 2015-09-17 | Colorado State University Research Foundation | Methods for improved in vitro-in vivo efficacy determination |
| KR102582563B1 (ko) * | 2014-06-20 | 2023-09-25 | 재단법인 한국파스퇴르연구소 | 항감염 화합물 |
| MX388564B (es) | 2014-10-09 | 2025-03-20 | Oncternal Therapeutics Inc | Compuestos de indolinona y usos de los mismos. |
| JP6864379B2 (ja) | 2016-03-31 | 2021-04-28 | オンターナル セラピューティック インコーポレイテッドOncternal Therapeutics, Inc. | インドール類似体及びその使用 |
| KR102282794B1 (ko) | 2016-07-29 | 2021-07-27 | 온크터널 테라퓨틱스, 인코포레이티드. | 인돌리논 화합물의 용도 |
| CN111303092B (zh) * | 2020-04-07 | 2021-05-25 | 山东昌邑灶户盐化有限公司 | 2,4-二硝基-6-氯苯胺衍生物、合成方法及其应用 |
| WO2023283425A1 (en) | 2021-07-09 | 2023-01-12 | Plexium, Inc. | Aryl compounds and pharmaceutical compositions that modulate ikzf2 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS61170732A (ja) * | 1985-01-25 | 1986-08-01 | Fuji Photo Film Co Ltd | ハロゲン化銀写真感光材料 |
| US7405235B2 (en) * | 2001-05-04 | 2008-07-29 | Paratek Pharmaceuticals, Inc. | Transcription factor modulating compounds and methods of use thereof |
| CN101065363B (zh) * | 2004-09-30 | 2012-05-02 | 詹森药业有限公司 | 可用作选择性雄激素受体调节剂(sarms)的新苯并咪唑衍生物 |
| CN101438288A (zh) * | 2006-03-15 | 2009-05-20 | Csir公司 | 谷氨酰胺合成酶的磷酰基转移酶活性的调节 |
-
2008
- 2008-04-21 JP JP2010504113A patent/JP5400032B2/ja not_active Expired - Fee Related
- 2008-04-21 IN IN3959KON2009 patent/IN2009KN03959A/en unknown
- 2008-04-21 HR HRP20131103AT patent/HRP20131103T1/hr unknown
- 2008-04-21 CN CN200880021064A patent/CN101677553A/zh active Pending
- 2008-04-21 MX MX2009011281A patent/MX2009011281A/es active IP Right Grant
- 2008-04-21 EP EP08799882.9A patent/EP2154966B1/en not_active Not-in-force
- 2008-04-21 EA EA200901423A patent/EA016726B1/ru not_active IP Right Cessation
- 2008-04-21 US US12/596,347 patent/US8232410B2/en not_active Expired - Fee Related
- 2008-04-21 AU AU2008242488A patent/AU2008242488B2/en not_active Ceased
- 2008-04-21 PT PT87998829T patent/PT2154966E/pt unknown
- 2008-04-21 WO PCT/US2008/005084 patent/WO2008130669A1/en not_active Ceased
- 2008-04-21 CA CA2684594A patent/CA2684594C/en active Active
- 2008-04-21 PL PL08799882T patent/PL2154966T3/pl unknown
- 2008-04-21 SI SI200831097T patent/SI2154966T1/sl unknown
- 2008-04-21 DK DK08799882.9T patent/DK2154966T3/da active
- 2008-04-21 BR BRPI0810244-9A patent/BRPI0810244A2/pt not_active Application Discontinuation
- 2008-04-21 ES ES08799882T patent/ES2434693T3/es active Active
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