JP2010513434A5 - - Google Patents

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Publication number
JP2010513434A5
JP2010513434A5 JP2009542194A JP2009542194A JP2010513434A5 JP 2010513434 A5 JP2010513434 A5 JP 2010513434A5 JP 2009542194 A JP2009542194 A JP 2009542194A JP 2009542194 A JP2009542194 A JP 2009542194A JP 2010513434 A5 JP2010513434 A5 JP 2010513434A5
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JP
Japan
Prior art keywords
oxy
azoniabicyclo
octane
alkyl
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2009542194A
Other languages
English (en)
Japanese (ja)
Other versions
JP2010513434A (ja
JP4604129B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/GB2007/004817 external-priority patent/WO2008075005A1/en
Publication of JP2010513434A publication Critical patent/JP2010513434A/ja
Publication of JP2010513434A5 publication Critical patent/JP2010513434A5/ja
Application granted granted Critical
Publication of JP4604129B2 publication Critical patent/JP4604129B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2009542194A 2006-12-19 2007-12-17 ムスカリン受容体アンタゴニストとしてのキヌクリジノール誘導体 Expired - Fee Related JP4604129B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US87063806P 2006-12-19 2006-12-19
PCT/GB2007/004817 WO2008075005A1 (en) 2006-12-19 2007-12-17 Quinuclidinol derivatives as muscarinic receptor antagonists

Publications (3)

Publication Number Publication Date
JP2010513434A JP2010513434A (ja) 2010-04-30
JP2010513434A5 true JP2010513434A5 (enExample) 2010-06-17
JP4604129B2 JP4604129B2 (ja) 2010-12-22

Family

ID=39166793

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009542194A Expired - Fee Related JP4604129B2 (ja) 2006-12-19 2007-12-17 ムスカリン受容体アンタゴニストとしてのキヌクリジノール誘導体

Country Status (22)

Country Link
US (1) US20100113510A1 (enExample)
EP (1) EP2121137B1 (enExample)
JP (1) JP4604129B2 (enExample)
KR (1) KR20090094460A (enExample)
CN (1) CN101610813A (enExample)
AR (1) AR064414A1 (enExample)
AT (1) ATE555111T1 (enExample)
AU (1) AU2007336054A1 (enExample)
BR (1) BRPI0721039A2 (enExample)
CA (1) CA2672446A1 (enExample)
CL (1) CL2007003690A1 (enExample)
CO (1) CO6180439A2 (enExample)
EC (1) ECSP099394A (enExample)
ES (1) ES2385681T3 (enExample)
IL (1) IL199015A0 (enExample)
MX (1) MX2009006018A (enExample)
NO (1) NO20092689L (enExample)
PE (1) PE20081837A1 (enExample)
RU (1) RU2009120229A (enExample)
TW (1) TW200831507A (enExample)
UY (1) UY30803A1 (enExample)
WO (1) WO2008075005A1 (enExample)

Families Citing this family (16)

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Publication number Priority date Publication date Assignee Title
TW200825084A (en) 2006-11-14 2008-06-16 Astrazeneca Ab New compounds 521
GB0808707D0 (en) * 2008-05-13 2008-06-18 Argenta Discovery Ltd New compounds 275
WO2009138707A1 (en) 2008-05-13 2009-11-19 Astrazeneca Ab Quinuclidine derivatives as muscarinic m3 receptor antagonists
GB0811099D0 (en) * 2008-06-17 2008-07-23 Astrazeneca Ab New combination 376
GB0811100D0 (en) * 2008-06-17 2008-07-23 Astrazeneca Ab New combination
WO2009153536A1 (en) * 2008-06-17 2009-12-23 Argenta Discovery Limited 1-aza-bicyclo [2.2.2] octane derivatives useful as muscarinic receptor antagonists
WO2010008341A1 (en) * 2008-07-16 2010-01-21 Astrazeneca Ab A combination of (a) glucocorticoid receptor modulator and (b) a muscarinic antagonist
EP2206712A1 (en) 2008-12-23 2010-07-14 CHIESI FARMACEUTICI S.p.A. "Alkaloid aminoester derivatives and medicinal composition thereof"
TW201036957A (en) 2009-02-20 2010-10-16 Astrazeneca Ab Novel salt 628
WO2010144043A1 (en) * 2009-06-12 2010-12-16 Astrazeneca Ab A novel 4-methylbenzenesulphonate salt and a process for preparing a pharmaceutical composition comprising the salt
JP2013500962A (ja) 2009-07-31 2013-01-10 カディラ ヘルスケア リミティド グルココルチコイド受容体のモジュレーターとしての新規化合物
WO2011073662A1 (en) 2009-12-17 2011-06-23 Astrazeneca Ab Combination of a benzoxazinone and a further agent for treating respiratory diseases
KR20130087406A (ko) * 2010-06-22 2013-08-06 키에시 파르마슈티시 엣스. 피. 에이. 알칼로이드 아미노에스테르 유도체 및 이의 의약 조성물
RU2569846C2 (ru) * 2010-06-22 2015-11-27 КЬЕЗИ ФАРМАЧЕУТИЧИ С.п.А. Алкалоидные производные сложных аминоэфиров и включающие их лекарственные композиции
RU2628082C2 (ru) * 2011-12-30 2017-08-14 КЬЕЗИ ФАРМАЧЕУТИЧИ С.п.А. Хинуклидиновые эфиры 1-азагетероциклилуксусной кислоты в качестве антимускариновых средств, способ их получения и их лекарственные композиции
KR101823451B1 (ko) * 2013-07-13 2018-01-30 베이징 에프에스웰컴 테크놀로지 디벨롭먼트 컴퍼니 리미티드 퀴논계 화합물, 이의 광학 이성질체 및 이의 제조 방법과 의약 용도

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GB9624482D0 (en) 1995-12-18 1997-01-15 Zeneca Phaema S A Chemical compounds
JP4471404B2 (ja) 1996-02-13 2010-06-02 アストラゼネカ ユーケイ リミテッド Vegfインヒビターとしてのキナゾリン誘導体
ATE211134T1 (de) 1996-03-05 2002-01-15 4-anilinochinazolin derivate
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CA2410562A1 (en) 2000-07-07 2002-01-31 Angiogene Pharmaceuticals Limited Colchinol derivatives as angiogenesis inhibitors
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AR044134A1 (es) * 2003-05-02 2005-08-24 Novartis Ag Derivados de quinuclidina, metodo de preparacion y composiciones farmaceuticas.
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GB0424284D0 (en) * 2004-11-02 2004-12-01 Novartis Ag Organic compounds
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