JP2010513434A5 - - Google Patents
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- Publication number
- JP2010513434A5 JP2010513434A5 JP2009542194A JP2009542194A JP2010513434A5 JP 2010513434 A5 JP2010513434 A5 JP 2010513434A5 JP 2009542194 A JP2009542194 A JP 2009542194A JP 2009542194 A JP2009542194 A JP 2009542194A JP 2010513434 A5 JP2010513434 A5 JP 2010513434A5
- Authority
- JP
- Japan
- Prior art keywords
- oxy
- azoniabicyclo
- octane
- alkyl
- phenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 CC1(C)C(CC2)*[N+]2(*)CC1 Chemical compound CC1(C)C(CC2)*[N+]2(*)CC1 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US87063806P | 2006-12-19 | 2006-12-19 | |
| PCT/GB2007/004817 WO2008075005A1 (en) | 2006-12-19 | 2007-12-17 | Quinuclidinol derivatives as muscarinic receptor antagonists |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2010513434A JP2010513434A (ja) | 2010-04-30 |
| JP2010513434A5 true JP2010513434A5 (enExample) | 2010-06-17 |
| JP4604129B2 JP4604129B2 (ja) | 2010-12-22 |
Family
ID=39166793
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009542194A Expired - Fee Related JP4604129B2 (ja) | 2006-12-19 | 2007-12-17 | ムスカリン受容体アンタゴニストとしてのキヌクリジノール誘導体 |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US20100113510A1 (enExample) |
| EP (1) | EP2121137B1 (enExample) |
| JP (1) | JP4604129B2 (enExample) |
| KR (1) | KR20090094460A (enExample) |
| CN (1) | CN101610813A (enExample) |
| AR (1) | AR064414A1 (enExample) |
| AT (1) | ATE555111T1 (enExample) |
| AU (1) | AU2007336054A1 (enExample) |
| BR (1) | BRPI0721039A2 (enExample) |
| CA (1) | CA2672446A1 (enExample) |
| CL (1) | CL2007003690A1 (enExample) |
| CO (1) | CO6180439A2 (enExample) |
| EC (1) | ECSP099394A (enExample) |
| ES (1) | ES2385681T3 (enExample) |
| IL (1) | IL199015A0 (enExample) |
| MX (1) | MX2009006018A (enExample) |
| NO (1) | NO20092689L (enExample) |
| PE (1) | PE20081837A1 (enExample) |
| RU (1) | RU2009120229A (enExample) |
| TW (1) | TW200831507A (enExample) |
| UY (1) | UY30803A1 (enExample) |
| WO (1) | WO2008075005A1 (enExample) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW200825084A (en) | 2006-11-14 | 2008-06-16 | Astrazeneca Ab | New compounds 521 |
| NZ589091A (en) | 2008-05-13 | 2011-07-29 | Astrazeneca Ab | Quinuclidine derivatives as muscarinic m3 receptor antagonists |
| GB0808707D0 (en) * | 2008-05-13 | 2008-06-18 | Argenta Discovery Ltd | New compounds 275 |
| GB0811100D0 (en) * | 2008-06-17 | 2008-07-23 | Astrazeneca Ab | New combination |
| GB0811099D0 (en) * | 2008-06-17 | 2008-07-23 | Astrazeneca Ab | New combination 376 |
| WO2009153536A1 (en) * | 2008-06-17 | 2009-12-23 | Argenta Discovery Limited | 1-aza-bicyclo [2.2.2] octane derivatives useful as muscarinic receptor antagonists |
| WO2010008341A1 (en) * | 2008-07-16 | 2010-01-21 | Astrazeneca Ab | A combination of (a) glucocorticoid receptor modulator and (b) a muscarinic antagonist |
| EP2206712A1 (en) * | 2008-12-23 | 2010-07-14 | CHIESI FARMACEUTICI S.p.A. | "Alkaloid aminoester derivatives and medicinal composition thereof" |
| TW201036957A (en) | 2009-02-20 | 2010-10-16 | Astrazeneca Ab | Novel salt 628 |
| WO2010144043A1 (en) * | 2009-06-12 | 2010-12-16 | Astrazeneca Ab | A novel 4-methylbenzenesulphonate salt and a process for preparing a pharmaceutical composition comprising the salt |
| JP2013500962A (ja) | 2009-07-31 | 2013-01-10 | カディラ ヘルスケア リミティド | グルココルチコイド受容体のモジュレーターとしての新規化合物 |
| WO2011073662A1 (en) | 2009-12-17 | 2011-06-23 | Astrazeneca Ab | Combination of a benzoxazinone and a further agent for treating respiratory diseases |
| ES2545812T3 (es) * | 2010-06-22 | 2015-09-16 | Chiesi Farmaceutici S.P.A. | Derivados aminoéster de alcaloides y composición medicinal de estos |
| CN102947299B (zh) * | 2010-06-22 | 2015-07-15 | 奇斯药制品公司 | 生物碱氨基酯衍生物及其药物组合物 |
| WO2013098145A1 (en) | 2011-12-30 | 2013-07-04 | Chiesi Farmaceutici S.P.A. | Quinuclidine esters of 1-azaheterocyclylacetic acid as antimuscarinic agents, process for their preparation and medicinal compositions thereof |
| CN105431432B (zh) * | 2013-07-13 | 2018-01-09 | 北京硕佰医药科技有限责任公司 | 奎宁类化合物、其光学异构体及其制备方法和医药用途 |
Family Cites Families (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8334494D0 (en) | 1983-12-24 | 1984-02-01 | Tanabe Seiyaku Co | Carbostyril derivatives |
| GB8923590D0 (en) * | 1989-10-19 | 1989-12-06 | Pfizer Ltd | Antimuscarinic bronchodilators |
| GR1001529B (el) | 1990-09-07 | 1994-03-31 | Elmuquimica Farm Sl | Μέ?οδος για την λήψη νέων 21-εστέρων της 16-17-ακετάλης της πρ να-1,4-διενο-3,20-διόνης. |
| GB9624482D0 (en) | 1995-12-18 | 1997-01-15 | Zeneca Phaema S A | Chemical compounds |
| WO1997030035A1 (en) | 1996-02-13 | 1997-08-21 | Zeneca Limited | Quinazoline derivatives as vegf inhibitors |
| ES2169355T3 (es) | 1996-03-05 | 2002-07-01 | Astrazeneca Ab | Derivados de 4-anilinoquinazolina. |
| GB9718972D0 (en) | 1996-09-25 | 1997-11-12 | Zeneca Ltd | Chemical compounds |
| GB9714249D0 (en) | 1997-07-08 | 1997-09-10 | Angiogene Pharm Ltd | Vascular damaging agents |
| GB9900334D0 (en) | 1999-01-07 | 1999-02-24 | Angiogene Pharm Ltd | Tricylic vascular damaging agents |
| GB9900752D0 (en) | 1999-01-15 | 1999-03-03 | Angiogene Pharm Ltd | Benzimidazole vascular damaging agents |
| IL152682A0 (en) | 2000-05-31 | 2003-06-24 | Astrazeneca Ab | Indole derivatives with vascular damaging activity |
| GB0015876D0 (en) | 2000-06-28 | 2000-08-23 | Novartis Ag | Organic compounds |
| HUP0301742A3 (en) | 2000-07-07 | 2005-08-29 | Angiogene Pharm Ltd | Colchinol derivatives as angiogenesis inhibitors, process for producing them, pharmaceutical compositions containing them and their use |
| BR0112224A (pt) | 2000-07-07 | 2003-06-10 | Angiogene Pharm Ltd | Composto, composição farmacêutica, uso de um composto ou de um sal, solvato ou pró-droga farmaceuticamente aceitável do mesmo, e, processo para preparar um composto |
| WO2002076933A1 (en) | 2001-03-22 | 2002-10-03 | Glaxo Group Limited | Formailide derivatives as beta2-adrenoreceptor agonists |
| WO2002088167A1 (en) | 2001-04-30 | 2002-11-07 | Glaxo Group Limited | Anti-inflammatory 17.beta.-carbothioate ester derivatives of androstane with a cyclic ester group in position 17.alpha |
| US20030229058A1 (en) | 2001-11-13 | 2003-12-11 | Moran Edmund J. | Aryl aniline beta2 adrenergic receptor agonists |
| TWI249515B (en) | 2001-11-13 | 2006-02-21 | Theravance Inc | Aryl aniline beta2 adrenergic receptor agonists |
| ES2302938T3 (es) | 2002-10-11 | 2008-08-01 | Pfizer Inc. | Derivados de indol como agonistas beta-2. |
| US7056916B2 (en) | 2002-11-15 | 2006-06-06 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Medicaments for the treatment of chronic obstructive pulmonary disease |
| CN100445281C (zh) * | 2003-05-02 | 2008-12-24 | 诺瓦提斯公司 | 与毒蕈碱性m3受体结合的奎宁环衍生物 |
| AR044134A1 (es) * | 2003-05-02 | 2005-08-24 | Novartis Ag | Derivados de quinuclidina, metodo de preparacion y composiciones farmaceuticas. |
| AU2004285592B2 (en) | 2003-11-03 | 2010-02-18 | Norton Healthcare, Ltd. | Soft steroid compositions for use in dry powder inhalers |
| CA2584413A1 (en) | 2004-10-29 | 2006-05-04 | Astrazeneca Ab | Novel sulphonamide derivatives as glucocorticoid receptor modulators for the treatment of inflammatory diseases |
| GB0424284D0 (en) * | 2004-11-02 | 2004-12-01 | Novartis Ag | Organic compounds |
| TW200722418A (en) * | 2005-04-20 | 2007-06-16 | Astrazeneca Ab | Novel compounds |
-
2007
- 2007-12-17 WO PCT/GB2007/004817 patent/WO2008075005A1/en not_active Ceased
- 2007-12-17 KR KR1020097014992A patent/KR20090094460A/ko not_active Withdrawn
- 2007-12-17 CN CNA2007800514963A patent/CN101610813A/zh active Pending
- 2007-12-17 US US12/518,185 patent/US20100113510A1/en not_active Abandoned
- 2007-12-17 AU AU2007336054A patent/AU2007336054A1/en not_active Abandoned
- 2007-12-17 BR BRPI0721039-6A patent/BRPI0721039A2/pt not_active IP Right Cessation
- 2007-12-17 AT AT07848557T patent/ATE555111T1/de active
- 2007-12-17 JP JP2009542194A patent/JP4604129B2/ja not_active Expired - Fee Related
- 2007-12-17 EP EP07848557A patent/EP2121137B1/en active Active
- 2007-12-17 MX MX2009006018A patent/MX2009006018A/es not_active Application Discontinuation
- 2007-12-17 ES ES07848557T patent/ES2385681T3/es active Active
- 2007-12-17 CA CA002672446A patent/CA2672446A1/en not_active Abandoned
- 2007-12-17 RU RU2009120229/15A patent/RU2009120229A/ru not_active Application Discontinuation
- 2007-12-18 AR ARP070105689A patent/AR064414A1/es unknown
- 2007-12-18 UY UY30803A patent/UY30803A1/es unknown
- 2007-12-18 CL CL200703690A patent/CL2007003690A1/es unknown
- 2007-12-18 TW TW096148391A patent/TW200831507A/zh unknown
-
2008
- 2008-01-02 PE PE2008000007A patent/PE20081837A1/es not_active Application Discontinuation
-
2009
- 2009-05-27 IL IL199015A patent/IL199015A0/en unknown
- 2009-05-28 CO CO09054972A patent/CO6180439A2/es not_active Application Discontinuation
- 2009-06-08 EC EC2009009394A patent/ECSP099394A/es unknown
- 2009-07-15 NO NO20092689A patent/NO20092689L/no not_active Application Discontinuation
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