JP2010512366A - Ｍｃｈ拮抗活性を有する新規ピリダジン誘導体及びこれらの化合物を含む薬物 - Google Patents

Ｍｃｈ拮抗活性を有する新規ピリダジン誘導体及びこれらの化合物を含む薬物 Download PDF

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JP2010512366A
JP2010512366A JP2009540731A JP2009540731A JP2010512366A JP 2010512366 A JP2010512366 A JP 2010512366A JP 2009540731 A JP2009540731 A JP 2009540731A JP 2009540731 A JP2009540731 A JP 2009540731A JP 2010512366 A JP2010512366 A JP 2010512366A
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alkyl
group
amino
cycloalkyl
substituted
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JP2010512366A5 (enExample
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リンツ トルシュテン レーマン
ディルク シュテンカンプ
ゲラルト ユールゲン ロート
シュテファン ゲオルク ミューラー
ヨルグ クライ
アルミン ヘッケル
クラウス ルドルフ
マルクス シンドラー
ラルフ ロッツ
パトリック ティールマン
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ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
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JP2009540731A 2006-12-11 2007-12-10 Ｍｃｈ拮抗活性を有する新規ピリダジン誘導体及びこれらの化合物を含む薬物 Pending JP2010512366A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06125763 2006-12-11
PCT/EP2007/063575 WO2008071646A1 (en) 2006-12-11 2007-12-10 New pyridazine derivatives with mch antagonistic activity and medicaments comprising these compounds

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JP2010512366A true JP2010512366A (ja) 2010-04-22
JP2010512366A5 JP2010512366A5 (enExample) 2011-02-03

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JP2009540731A Pending JP2010512366A (ja) 2006-12-11 2007-12-10 Ｍｃｈ拮抗活性を有する新規ピリダジン誘導体及びこれらの化合物を含む薬物

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US (1) US20100197908A1 (enExample)
EP (1) EP2102171A1 (enExample)
JP (1) JP2010512366A (enExample)
AR (1) AR064293A1 (enExample)
CA (1) CA2671984A1 (enExample)
CL (1) CL2007003580A1 (enExample)
TW (1) TW200831485A (enExample)
WO (1) WO2008071646A1 (enExample)

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Publication number Priority date Publication date Assignee Title
JP2011502983A (ja) * 2007-11-01 2011-01-27 アキュセラ インコーポレイテッド 眼の疾患及び障害治療用のアミン誘導体化合物
JP2013525376A (ja) * 2010-04-23 2013-06-20 サイトキネティクス・インコーポレーテッド 特定のアミノピリダジン、その組成物、及びこれらの使用方法
US9730886B2 (en) 2010-04-23 2017-08-15 Cytokinetics, Inc. Amino-pyrimidine skeletal muscle modulators
JPWO2022009911A1 (enExample) * 2020-07-08 2022-01-13

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US9133123B2 (en) 2010-04-23 2015-09-15 Cytokinetics, Inc. Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use
EP2650284A1 (en) * 2012-04-10 2013-10-16 Merz Pharma GmbH & Co. KGaA Heterocyclic derivatives as metabotropic glutamate receptor modulators
CN104971286A (zh) * 2015-05-25 2015-10-14 广东工业大学 一种治疗肩腰腿不适症的中药组合物
BR112018077281A2 (pt) * 2016-07-01 2019-04-02 Boulos & Cooper Pharmaceuticals Pty Ltd novos antibióticos
DK3494120T3 (da) 2016-08-05 2021-05-31 Boehringer Ingelheim Int Oxadiazolopyridinderivater til anvendelse som ghrelin-o-acyl-transferase-(goat)-inhibitorer
BR112021004635A2 (pt) 2018-10-29 2021-05-25 Boehringer Ingelheim International Gmbh derivados de piridinil sulfonamida, composições farmacêuticas e usos das mesmas
CN112955214B (zh) 2018-10-29 2024-05-07 勃林格殷格翰国际有限公司 吡啶基磺酰胺衍生物、药物组合物及其用途
US11465982B2 (en) 2019-07-22 2022-10-11 Boehringer Ingelheim International Gmbh Pyridazines
US11485727B2 (en) * 2019-07-22 2022-11-01 Boehringer Ingelheim International Gmbh N-methyl, n-(6-(methoxy)pyridazin-3-yl) amine derivatives as autotaxin (ATX) modulators
DK4003978T3 (da) * 2019-07-22 2024-07-22 Boehringer Ingelheim Int N-methyl, n-(6-(methoxy)pyridazin-3-yl) aminderivater som autotaxin (atx) modulatorer til behandlingen af inflammatoriske luftvejs- eller fibrotiske sygdomme

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WO2004039780A1 (de) * 2002-10-31 2004-05-13 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue alkin-verbindungen mit mch-antagonistischer wirkung und diese verbindungen enthaltende arzneimittel
WO2005103029A1 (de) * 2004-04-14 2005-11-03 Boehringer Ingelheim International Gmbh Neue alkin-verbindungen mit mch-antagonistischer wirkung und diese verbindungen enthaltende arzneimittel
WO2005103032A2 (de) * 2004-04-14 2005-11-03 Boehringer Ingelheim International Gmbh Neue alkin-verbindungen mit mch-antagonistischer wirkung und diese verbindungen enthaltende arzneimittel

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AU2001252596A1 (en) 2000-04-28 2001-11-12 Takeda Chemical Industries Ltd. Melanin concentrating hormone antagonists
JP2005519895A (ja) 2002-01-18 2005-07-07 ファルマシア・コーポレーション Ｐ３８阻害剤としての置換ピリダジノン
AP1822A (en) 2002-02-14 2008-01-30 Pharmacia Corp Substituted pyridinones as modulators of P38 MAP kinase.
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