JP2010504913A - 炎症及び免疫関連使用のための縮合環化合物 - Google Patents

炎症及び免疫関連使用のための縮合環化合物 Download PDF

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JP2010504913A
JP2010504913A JP2009529277A JP2009529277A JP2010504913A JP 2010504913 A JP2010504913 A JP 2010504913A JP 2009529277 A JP2009529277 A JP 2009529277A JP 2009529277 A JP2009529277 A JP 2009529277A JP 2010504913 A JP2010504913 A JP 2010504913A
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JP2010504913A5 (enExample
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フウ ボ,ニャ
チェ,クィンリン
チェン,ショウジュン
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シンタ ファーマシューティカルズ コーポレーション
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    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
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  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
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  • Gastroenterology & Hepatology (AREA)
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  • Endocrinology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Emergency Medicine (AREA)
  • Pain & Pain Management (AREA)
JP2009529277A 2006-09-26 2007-09-26 炎症及び免疫関連使用のための縮合環化合物 Ceased JP2010504913A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US84732506P 2006-09-26 2006-09-26
US11/861,278 US8779154B2 (en) 2006-09-26 2007-09-25 Fused ring compounds for inflammation and immune-related uses
PCT/US2007/020864 WO2008039520A2 (en) 2006-09-26 2007-09-26 Fused ring compounds for inflammation and immune-related uses

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JP2010504913A true JP2010504913A (ja) 2010-02-18
JP2010504913A5 JP2010504913A5 (enExample) 2011-08-18

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US (1) US8779154B2 (enExample)
EP (1) EP2086983A4 (enExample)
JP (1) JP2010504913A (enExample)
AU (1) AU2007300450B2 (enExample)
CA (1) CA2664301A1 (enExample)
WO (1) WO2008039520A2 (enExample)

Cited By (3)

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JP2011509261A (ja) * 2008-01-07 2011-03-24 シンタ ファーマシューティカルズ コーポレーション 炎症および免疫関連用途向けの化合物
JP2011517457A (ja) * 2008-03-31 2011-06-09 ジェネンテック, インコーポレイテッド ベンゾピランおよびベンゾキセピンpi3k阻害剤化合物および使用方法
JP2016510752A (ja) * 2013-03-06 2016-04-11 ヤンセン ファーマシューティカ エヌ.ベー. ヒスタミンh4受容体のベンゾイミダゾール−2−イルピリミジンモジュレータ

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JP2009524683A (ja) 2006-01-25 2009-07-02 シンタ ファーマシューティカルズ コーポレーション 炎症および免疫関連用途のためのビニル−フェニル誘導体
WO2007087441A2 (en) * 2006-01-25 2007-08-02 Synta Pharmaceuticals Corp. Substituted aromatic compounds for inflammation and immune-related uses
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BRPI0710083A2 (pt) 2006-03-31 2011-08-02 Janssen Pharmaceutica Nv entidade quìmica benzoimidazol-2-il pirimidina e pirazina, composição farmacêutica e uso destas
US9371311B2 (en) 2008-06-30 2016-06-21 Janssen Pharmaceutica Nv Benzoimidazol-2-yl pyrimidine derivatives
US8288379B2 (en) * 2009-04-22 2012-10-16 Boehringer Ingelheim International Gmbh Thia-triaza-cyclopentazulenes
PE20121025A1 (es) 2009-09-28 2012-08-06 Hoffmann La Roche Compuestos de benzoxazepina como inhibidores de la p13k
NZ599090A (en) * 2009-09-28 2014-02-28 Hoffmann La Roche Benzoxepin pi3k inhibitor compounds and methods of use
US8993612B2 (en) 2009-10-08 2015-03-31 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel and methods for treatment of non-small cell lung cancer
US8377970B2 (en) 2009-10-08 2013-02-19 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel
EP2592071B1 (en) * 2009-10-29 2019-09-18 Bristol-Myers Squibb Company Tricyclic heterocyclic compounds
AU2010321832B2 (en) 2009-11-20 2014-08-14 Amgen Inc. Anti-Orai1 antigen binding proteins and uses thereof
CA2825966A1 (en) 2011-03-21 2012-09-27 F. Hoffmann-La Roche Ag Benzoxazepin compounds selective for pi3k p110 delta and methods of use
WO2013113863A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
WO2013113773A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
EA201400858A1 (ru) 2012-02-03 2015-01-30 Басф Се Фунгицидные пиримидиновые соединения
WO2013113791A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
WO2013113716A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
WO2013113776A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
US9462809B2 (en) 2012-03-13 2016-10-11 Basf Se Fungicidal pyrimidine compounds
WO2013135672A1 (en) 2012-03-13 2013-09-19 Basf Se Fungicidal pyrimidine compounds
EP2738172A1 (en) 2012-11-28 2014-06-04 Almirall, S.A. New bicyclic compounds as crac channel modulators
WO2014118099A1 (en) 2013-01-30 2014-08-07 Basf Se Fungicidal naphthoquinones and derivatives
EP2848615A1 (en) 2013-07-03 2015-03-18 Almirall, S.A. New pyrazole derivatives as CRAC channel modulators
JP7029445B2 (ja) 2016-09-02 2022-03-03 ブリストル-マイヤーズ スクイブ カンパニー 置換された三環式ヘテロ環化合物
WO2018206820A1 (en) 2017-05-12 2018-11-15 Mavalon Therapeutics Limited Substituted heterocyclic compounds as allosteric modulators of group ii metabotropic glutamate receptors
WO2019032632A1 (en) 2017-08-09 2019-02-14 Bristol-Myers Squibb Company ALKYLPHENYL COMPOUNDS
WO2019032631A1 (en) 2017-08-09 2019-02-14 Bristol-Myers Squibb Company Oxime ether compounds
JP2022508468A (ja) 2018-09-14 2022-01-19 ルヒゼン ファーマスティカルズ アクツィエンゲゼルシャフト Crac阻害剤およびコルチコステロイドを含む組成物ならびにそれらの使用方法
JP7744350B2 (ja) 2020-01-13 2025-09-25 バージ アナリティクス,インコーポレイテッド 置換ピラゾロ-ピリミジンおよびその使用
CN114621070B (zh) * 2022-04-02 2024-03-19 上海陶术生物科技有限公司 3,4-二氢萘-1(2h)-酮衍生物的合成方法
WO2025082467A1 (zh) * 2023-10-19 2025-04-24 成都先导药物开发股份有限公司 一种免疫调节剂

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