JP2010501541A5 - - Google Patents
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- Publication number
- JP2010501541A5 JP2010501541A5 JP2009525123A JP2009525123A JP2010501541A5 JP 2010501541 A5 JP2010501541 A5 JP 2010501541A5 JP 2009525123 A JP2009525123 A JP 2009525123A JP 2009525123 A JP2009525123 A JP 2009525123A JP 2010501541 A5 JP2010501541 A5 JP 2010501541A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- substituted
- phenyl
- pyridin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 0 CC(*)(CNC)CNI Chemical compound CC(*)(CNC)CNI 0.000 description 2
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN1336MU2006 | 2006-08-24 | ||
| PCT/IB2007/002405 WO2008023248A2 (en) | 2006-08-24 | 2007-08-22 | Novel macrolides and ketolides having antimicrobial activity |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010501541A JP2010501541A (ja) | 2010-01-21 |
| JP2010501541A5 true JP2010501541A5 (cg-RX-API-DMAC7.html) | 2010-10-14 |
Family
ID=39107171
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009525123A Pending JP2010501541A (ja) | 2006-08-24 | 2007-08-22 | 抗菌活性を有する新規マクロライド及びケトライド |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US8097594B2 (cg-RX-API-DMAC7.html) |
| EP (1) | EP2056844A4 (cg-RX-API-DMAC7.html) |
| JP (1) | JP2010501541A (cg-RX-API-DMAC7.html) |
| KR (1) | KR20090042971A (cg-RX-API-DMAC7.html) |
| CN (1) | CN101541331A (cg-RX-API-DMAC7.html) |
| CA (1) | CA2661538A1 (cg-RX-API-DMAC7.html) |
| WO (1) | WO2008023248A2 (cg-RX-API-DMAC7.html) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2748599T3 (es) | 2007-08-27 | 2020-03-17 | Dart Neuroscience Cayman Ltd | Compuestos terapéuticos de isoxazol |
| CN101910159B (zh) * | 2007-12-26 | 2013-06-19 | 卫材R&D管理有限公司 | 杂环取代吡啶衍生物的制备方法 |
| EP2435460B1 (en) * | 2009-05-27 | 2015-01-07 | Wockhardt Limited | Ketolide compounds having antimicrobial activity |
| CN103384676B (zh) * | 2010-12-09 | 2016-02-03 | 沃克哈特有限公司 | 酮内酯化合物 |
| CN103619849B (zh) * | 2011-03-01 | 2016-05-25 | 沃克哈特有限公司 | 酮内酯中间体的制备方法 |
| WO2012127351A1 (en) * | 2011-03-22 | 2012-09-27 | Wockhardt Limited | Process for preparation of ketolide compounds |
| WO2012129564A2 (en) | 2011-03-24 | 2012-09-27 | H. Lee Moffitt Cancer Center And Research Institute, Inc. | Proteasome chymotrypsin-like inhibition using pi-1833 analogs |
| CN102260225B (zh) * | 2011-06-02 | 2013-08-21 | 蒋杰 | 用于抑制肿瘤转移和肿瘤血管生长的苯基哌嗪类衍生物 |
| JP2017531663A (ja) * | 2014-10-08 | 2017-10-26 | プレジデント アンド フェローズ オブ ハーバード カレッジ | 14員ケトライドならびにそれらの調製および使用の方法 |
| JP6887022B2 (ja) * | 2017-03-16 | 2021-06-16 | ウォックハート リミテッド | ケトライド化合物を製造するための方法 |
| ES2948122A1 (es) * | 2022-02-10 | 2023-08-31 | Fundacion Instituto De Investig Sanitaria Aragon | Compuestos para el tratamiento y/o prevención de una infección o enfermedad causada por Helicobacter o Campylobacter |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2473525A1 (fr) | 1980-01-11 | 1981-07-17 | Roussel Uclaf | Nouvelles oximes derivees de l'erythromycine, leur procede de preparation et leur application comme medicaments |
| US4331803A (en) | 1980-06-04 | 1982-05-25 | Taisho Pharmaceutical Co., Ltd. | Novel erythromycin compounds |
| YU43006B (en) | 1981-03-06 | 1989-02-28 | Pliva Pharm & Chem Works | Process for preparing n-methyl-11-aza-10-deoxo-10-dihydro erythromycin and derivatives thereof |
| FR2719587B1 (fr) | 1994-05-03 | 1996-07-12 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
| DK1291351T3 (da) | 1996-09-04 | 2005-10-24 | Abbott Lab | 6-O-substituerede ketolider med antibakteriel aktivitet |
| KR100502031B1 (ko) * | 2000-08-22 | 2005-07-25 | 바실리어 파마슈티카 아게 | 항균 활성을 갖는 신규한 매크롤라이드 |
| GB0031312D0 (en) | 2000-12-21 | 2001-02-07 | Glaxo Group Ltd | Macrolides |
| CN1492874A (zh) | 2000-12-21 | 2004-04-28 | 大环内酯 | |
| CN1533388A (zh) | 2001-07-19 | 2004-09-29 | CVҽҩ����˾ | 取代的哌嗪化合物及其作为脂肪酸氧化抑制剂的应用 |
| GB0127349D0 (en) | 2001-11-14 | 2002-01-02 | Glaxo Group Ltd | Macrolides |
| US6995143B2 (en) | 2002-02-28 | 2006-02-07 | Basilea Pharmaceutica Ag | Macrolides with antibacterial activity |
| US6727229B2 (en) | 2002-08-19 | 2004-04-27 | Enanta Pharmaceuticals, Inc. | 11,12-substituted lactone ketolide derivatives having antibacterial activity |
| HRP20090302T1 (hr) * | 2005-02-09 | 2009-07-31 | Basilea Pharmaceutica Ag | Novi makrolidi |
-
2007
- 2007-08-22 CN CNA2007800373931A patent/CN101541331A/zh active Pending
- 2007-08-22 EP EP07804796A patent/EP2056844A4/en not_active Withdrawn
- 2007-08-22 WO PCT/IB2007/002405 patent/WO2008023248A2/en not_active Ceased
- 2007-08-22 CA CA002661538A patent/CA2661538A1/en not_active Abandoned
- 2007-08-22 KR KR1020097005432A patent/KR20090042971A/ko not_active Ceased
- 2007-08-22 JP JP2009525123A patent/JP2010501541A/ja active Pending
-
2009
- 2009-02-24 US US12/379,539 patent/US8097594B2/en not_active Expired - Fee Related
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