JP2009545549A5 - - Google Patents

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Publication number
JP2009545549A5
JP2009545549A5 JP2009522200A JP2009522200A JP2009545549A5 JP 2009545549 A5 JP2009545549 A5 JP 2009545549A5 JP 2009522200 A JP2009522200 A JP 2009522200A JP 2009522200 A JP2009522200 A JP 2009522200A JP 2009545549 A5 JP2009545549 A5 JP 2009545549A5
Authority
JP
Japan
Prior art keywords
butyrate
amino
carbamoyl
compound
trimethylammonium
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2009522200A
Other languages
English (en)
Japanese (ja)
Other versions
JP2009545549A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2007/057030 external-priority patent/WO2008015081A1/en
Publication of JP2009545549A publication Critical patent/JP2009545549A/ja
Publication of JP2009545549A5 publication Critical patent/JP2009545549A5/ja
Withdrawn legal-status Critical Current

Links

JP2009522200A 2006-08-02 2007-07-10 Cpt阻害剤としての4−トリメチルアンモニウム−3−アミノブチレートおよび4−トリメチルフォスフォニウム−3−アミノブチレート誘導体 Withdrawn JP2009545549A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06118338 2006-08-02
PCT/EP2007/057030 WO2008015081A1 (en) 2006-08-02 2007-07-10 Derivatives of 4-trimethylammonium-3-aminobutyrate and 4-trimethylphosphonium-3-aminobutyrate as cpt-inhibitors

Publications (2)

Publication Number Publication Date
JP2009545549A JP2009545549A (ja) 2009-12-24
JP2009545549A5 true JP2009545549A5 (enExample) 2010-09-02

Family

ID=37395789

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009522200A Withdrawn JP2009545549A (ja) 2006-08-02 2007-07-10 Cpt阻害剤としての4−トリメチルアンモニウム−3−アミノブチレートおよび4−トリメチルフォスフォニウム−3−アミノブチレート誘導体

Country Status (15)

Country Link
US (1) US20090312286A1 (enExample)
EP (1) EP2046734A1 (enExample)
JP (1) JP2009545549A (enExample)
KR (1) KR20090034969A (enExample)
CN (1) CN101511780A (enExample)
AR (1) AR062217A1 (enExample)
AU (1) AU2007280604A1 (enExample)
BR (1) BRPI0715084A2 (enExample)
CA (1) CA2658797A1 (enExample)
EA (1) EA200970170A1 (enExample)
IL (1) IL196594A0 (enExample)
MX (1) MX2009001104A (enExample)
SG (1) SG174032A1 (enExample)
TW (1) TW200815326A (enExample)
WO (1) WO2008015081A1 (enExample)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8410150B2 (en) 2007-03-09 2013-04-02 University Health Network Inhibitors of carnitine palmitoyltransferase and treating cancer
US8680282B2 (en) 2007-08-01 2014-03-25 University Health Network Cyclic inhibitors of carnitine palmitoyltransferase and treating cancer
EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
MX2010008196A (es) * 2008-04-29 2010-08-11 Hoffmann La Roche Derivados de acido 4-dimetilaminobutirico.
WO2009132979A1 (en) * 2008-04-29 2009-11-05 F. Hoffmann-La Roche Ag 4-trimethylammonio-butyrates as cpt2 inhibitors
US8957032B2 (en) * 2008-05-06 2015-02-17 Alba Therapeutics Corporation Inhibition of gliadin peptides
KR20110044209A (ko) * 2008-06-24 2011-04-28 다라 바이오싸이언시즈, 아이엔씨. 효소 억제제 및 그의 용도
EP2582709B1 (de) 2010-06-18 2018-01-24 Sanofi Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen
EP2567959B1 (en) 2011-09-12 2014-04-16 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0127098B1 (en) 1983-05-25 1989-02-08 Takeda Chemical Industries, Ltd. Derivatives of beta-amino-gamma-trimethylammonio-butyrate, their production and use
HUT65327A (en) 1992-06-11 1994-05-02 Sandoz Ag Process for producing phosphinyloxy-propyl-ammonium inner sact derwatives ang pharmateutical preparations containing them
IT1299266B1 (it) 1998-05-15 2000-02-29 Sigma Tau Ind Farmaceuti Inibitori reversibili della carnitina palmitoil trasferasi

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