JP2009541404A5 - - Google Patents
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- JP2009541404A5 JP2009541404A5 JP2009517024A JP2009517024A JP2009541404A5 JP 2009541404 A5 JP2009541404 A5 JP 2009541404A5 JP 2009517024 A JP2009517024 A JP 2009517024A JP 2009517024 A JP2009517024 A JP 2009517024A JP 2009541404 A5 JP2009541404 A5 JP 2009541404A5
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- JP
- Japan
- Prior art keywords
- alkyl
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- disorder
- membered
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06116592 | 2006-07-04 | ||
| PCT/EP2007/005851 WO2008003452A1 (en) | 2006-07-04 | 2007-07-02 | Pyrazolealkanamide substituted thiophenes as ampa potentiators |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2009541404A JP2009541404A (ja) | 2009-11-26 |
| JP2009541404A5 true JP2009541404A5 (enExample) | 2013-04-11 |
Family
ID=37226676
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009517024A Ceased JP2009541404A (ja) | 2006-07-04 | 2007-07-02 | Ａｍｐａ増強剤としてのピラゾールアルカンアミド置換チオフェン |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US7820707B2 (enExample) |
| EP (1) | EP2041124B1 (enExample) |
| JP (1) | JP2009541404A (enExample) |
| KR (1) | KR20090027672A (enExample) |
| CN (1) | CN101484448B (enExample) |
| AR (1) | AR061792A1 (enExample) |
| AU (1) | AU2007271469B2 (enExample) |
| CA (1) | CA2655680A1 (enExample) |
| IL (1) | IL196302A0 (enExample) |
| MX (1) | MX2008016494A (enExample) |
| NZ (1) | NZ573325A (enExample) |
| PE (1) | PE20080378A1 (enExample) |
| TW (1) | TW200817385A (enExample) |
| WO (1) | WO2008003452A1 (enExample) |
| ZA (1) | ZA200810165B (enExample) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2269990A4 (en) * | 2008-03-25 | 2012-04-18 | Takeda Pharmaceutical | Heterocyclic compound |
| TW201012803A (en) * | 2008-06-06 | 2010-04-01 | Organon Nv | Heterocyclic derivatives |
| WO2011036889A1 (ja) * | 2009-09-25 | 2011-03-31 | 武田薬品工業株式会社 | 複素環化合物 |
| WO2011036885A1 (ja) * | 2009-09-25 | 2011-03-31 | 武田薬品工業株式会社 | 複素環化合物 |
| PT2603494T (pt) | 2010-08-10 | 2017-02-03 | Syngenta Participations Ag | Processo para a preparação de 3-haloalquilopirazóis |
| JO3225B1 (ar) * | 2012-11-27 | 2018-03-08 | Lilly Co Eli | 6-((s)-1-{1-[5-(2-هيدروكسي-إيثوكسي)-بيريدين-2-يل]-1h-بيرازول-3-يل}إيثيل)-3h-1 ، 3-بنزو ثيازول-2- أون باعتباره مضاد مستقبل ampa يعتمد على tarp- جاما 8 |
| EP3030568B1 (en) | 2013-08-08 | 2018-09-19 | Galapagos NV | Thieno[2,3-c]pyrans as cftr modulators |
| CN103772282B (zh) * | 2014-02-26 | 2015-09-23 | 上海毕得医药科技有限公司 | 一种3-叔丁基-1h-吡唑-4-甲醛的制备方法 |
| TW201609719A (zh) * | 2014-05-28 | 2016-03-16 | 美國禮來大藥廠 | 作為ＴＡＲＰ－γ８依賴性ＡＭＰＡ受體拮抗劑之６－經取代－３Ｈ－１，３－苯并噻唑－２－酮化合物 |
| CN107286114B (zh) * | 2016-04-13 | 2020-08-18 | 中国人民解放军军事医学科学院毒物药物研究所 | Ampa受体增效剂的脑靶向前药及其医药用途 |
| GB201702221D0 (en) * | 2017-02-10 | 2017-03-29 | Univ Of Sussex | Compounds |
| GB201803340D0 (en) | 2018-03-01 | 2018-04-18 | Univ Of Sussex | Compounds |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2311131A1 (en) * | 1997-11-21 | 1999-06-03 | Nps Pharmaceuticals, Inc. | Metabotropic glutamate receptor antagonists for treating central nervous system diseases |
| ES2249272T3 (es) * | 1999-06-02 | 2006-04-01 | Nps Pharmaceuticals, Inc. | Antagonistas de receptores de glutamato metabotropicos y su uso para el tratamiento de enfermedades del sistema nervioso central. |
| US6414013B1 (en) * | 2000-06-19 | 2002-07-02 | Pharmacia & Upjohn S.P.A. | Thiophene compounds, process for preparing the same, and pharmaceutical compositions containing the same background of the invention |
| US20040171603A1 (en) | 2001-05-18 | 2004-09-02 | Janos Pato | Novel therapeutic targets for the treatment of mycobacterial infections and compounds useful therefor |
| US7345036B2 (en) * | 2001-06-14 | 2008-03-18 | N.V. Organon | (Pyrido/thieno)—[f]—oxazepine-5-one derivatives |
| US20050085531A1 (en) | 2003-10-03 | 2005-04-21 | Hodge Carl N. | Thiophene-based compounds exhibiting ATP-utilizing enzyme inhibitory activity, and compositions, and uses thereof |
| CA2541458C (en) | 2003-10-08 | 2011-09-20 | Eli Lilly And Company | Pyrrole and pyrazole derivatives as potentiators of glutamate receptors |
| ATE552251T1 (de) | 2004-01-09 | 2012-04-15 | Lilly Co Eli | Thiophen- und furanverbindungen |
| JP2008517061A (ja) | 2004-10-20 | 2008-05-22 | コンパス ファーマシューティカルズ リミティド ライアビリティ カンパニー | 抗腫瘍剤としての化合物及びそれらの使用 |
-
2007
- 2007-06-14 TW TW096121620A patent/TW200817385A/zh unknown
- 2007-06-29 US US11/771,198 patent/US7820707B2/en active Active
- 2007-07-02 EP EP07801415.6A patent/EP2041124B1/en active Active
- 2007-07-02 CA CA002655680A patent/CA2655680A1/en not_active Abandoned
- 2007-07-02 WO PCT/EP2007/005851 patent/WO2008003452A1/en not_active Ceased
- 2007-07-02 KR KR1020087031534A patent/KR20090027672A/ko not_active Withdrawn
- 2007-07-02 MX MX2008016494A patent/MX2008016494A/es active IP Right Grant
- 2007-07-02 AR ARP070102955A patent/AR061792A1/es unknown
- 2007-07-02 JP JP2009517024A patent/JP2009541404A/ja not_active Ceased
- 2007-07-02 AU AU2007271469A patent/AU2007271469B2/en not_active Ceased
- 2007-07-02 NZ NZ573325A patent/NZ573325A/en unknown
- 2007-07-02 CN CN2007800248081A patent/CN101484448B/zh not_active Expired - Fee Related
- 2007-07-03 PE PE2007000848A patent/PE20080378A1/es not_active Application Discontinuation
-
2008
- 2008-11-28 ZA ZA200810165A patent/ZA200810165B/xx unknown
- 2008-12-31 IL IL196302A patent/IL196302A0/en unknown
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