JP2009541404A5 - - Google Patents
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- Publication number
- JP2009541404A5 JP2009541404A5 JP2009517024A JP2009517024A JP2009541404A5 JP 2009541404 A5 JP2009541404 A5 JP 2009541404A5 JP 2009517024 A JP2009517024 A JP 2009517024A JP 2009517024 A JP2009517024 A JP 2009517024A JP 2009541404 A5 JP2009541404 A5 JP 2009541404A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
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- optionally substituted
- disorder
- membered
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06116592 | 2006-07-04 | ||
| PCT/EP2007/005851 WO2008003452A1 (en) | 2006-07-04 | 2007-07-02 | Pyrazolealkanamide substituted thiophenes as ampa potentiators |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2009541404A JP2009541404A (ja) | 2009-11-26 |
| JP2009541404A5 true JP2009541404A5 (cg-RX-API-DMAC7.html) | 2013-04-11 |
Family
ID=37226676
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009517024A Ceased JP2009541404A (ja) | 2006-07-04 | 2007-07-02 | Ａｍｐａ増強剤としてのピラゾールアルカンアミド置換チオフェン |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US7820707B2 (cg-RX-API-DMAC7.html) |
| EP (1) | EP2041124B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP2009541404A (cg-RX-API-DMAC7.html) |
| KR (1) | KR20090027672A (cg-RX-API-DMAC7.html) |
| CN (1) | CN101484448B (cg-RX-API-DMAC7.html) |
| AR (1) | AR061792A1 (cg-RX-API-DMAC7.html) |
| AU (1) | AU2007271469B2 (cg-RX-API-DMAC7.html) |
| CA (1) | CA2655680A1 (cg-RX-API-DMAC7.html) |
| IL (1) | IL196302A0 (cg-RX-API-DMAC7.html) |
| MX (1) | MX2008016494A (cg-RX-API-DMAC7.html) |
| NZ (1) | NZ573325A (cg-RX-API-DMAC7.html) |
| PE (1) | PE20080378A1 (cg-RX-API-DMAC7.html) |
| TW (1) | TW200817385A (cg-RX-API-DMAC7.html) |
| WO (1) | WO2008003452A1 (cg-RX-API-DMAC7.html) |
| ZA (1) | ZA200810165B (cg-RX-API-DMAC7.html) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20110118236A1 (en) * | 2008-03-25 | 2011-05-19 | Michiyo Mochizuki | Heterocyclic compound |
| TW201012803A (en) * | 2008-06-06 | 2010-04-01 | Organon Nv | Heterocyclic derivatives |
| WO2011036889A1 (ja) * | 2009-09-25 | 2011-03-31 | 武田薬品工業株式会社 | 複素環化合物 |
| WO2011036885A1 (ja) * | 2009-09-25 | 2011-03-31 | 武田薬品工業株式会社 | 複素環化合物 |
| JP5869570B2 (ja) | 2010-08-10 | 2016-02-24 | シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト | ３−ハロアルキルピラゾールの調製方法 |
| JO3225B1 (ar) * | 2012-11-27 | 2018-03-08 | Lilly Co Eli | 6-((s)-1-{1-[5-(2-هيدروكسي-إيثوكسي)-بيريدين-2-يل]-1h-بيرازول-3-يل}إيثيل)-3h-1 ، 3-بنزو ثيازول-2- أون باعتباره مضاد مستقبل ampa يعتمد على tarp- جاما 8 |
| SG11201600891UA (en) | 2013-08-08 | 2016-03-30 | Galapagos Nv | Thieno[2,3-c]pyrans as cftr modulators |
| CN103772282B (zh) * | 2014-02-26 | 2015-09-23 | 上海毕得医药科技有限公司 | 一种3-叔丁基-1h-吡唑-4-甲醛的制备方法 |
| TW201609719A (zh) * | 2014-05-28 | 2016-03-16 | 美國禮來大藥廠 | 作為ＴＡＲＰ－γ８依賴性ＡＭＰＡ受體拮抗劑之６－經取代－３Ｈ－１，３－苯并噻唑－２－酮化合物 |
| CN107286114B (zh) * | 2016-04-13 | 2020-08-18 | 中国人民解放军军事医学科学院毒物药物研究所 | Ampa受体增效剂的脑靶向前药及其医药用途 |
| GB201702221D0 (en) * | 2017-02-10 | 2017-03-29 | Univ Of Sussex | Compounds |
| GB201803340D0 (en) | 2018-03-01 | 2018-04-18 | Univ Of Sussex | Compounds |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MXPA00004940A (es) * | 1997-11-21 | 2002-10-17 | Nps Pharma Inc | Antagonistas de receptor de glutamato metabotropico para tratar enfermedades del sistema nervioso central. |
| HK1048635A1 (zh) * | 1999-06-02 | 2003-04-11 | Nps药物有限公司 | 代谢移变的谷氨酸盐受体拮抗剂和它们治疗中枢神经系统疾病的用途 |
| US6414013B1 (en) * | 2000-06-19 | 2002-07-02 | Pharmacia & Upjohn S.P.A. | Thiophene compounds, process for preparing the same, and pharmaceutical compositions containing the same background of the invention |
| US20040171603A1 (en) * | 2001-05-18 | 2004-09-02 | Janos Pato | Novel therapeutic targets for the treatment of mycobacterial infections and compounds useful therefor |
| US7345036B2 (en) * | 2001-06-14 | 2008-03-18 | N.V. Organon | (Pyrido/thieno)—[f]—oxazepine-5-one derivatives |
| US20050085531A1 (en) | 2003-10-03 | 2005-04-21 | Hodge Carl N. | Thiophene-based compounds exhibiting ATP-utilizing enzyme inhibitory activity, and compositions, and uses thereof |
| DE602004021011D1 (de) | 2003-10-08 | 2009-06-18 | Lilly Co Eli | Pyrrol- und pyrazolderivate als potentiatoren von glutamatrezeptoren |
| ATE552251T1 (de) | 2004-01-09 | 2012-04-15 | Lilly Co Eli | Thiophen- und furanverbindungen |
| JP2008517061A (ja) | 2004-10-20 | 2008-05-22 | コンパス ファーマシューティカルズ リミティド ライアビリティ カンパニー | 抗腫瘍剤としての化合物及びそれらの使用 |
-
2007
- 2007-06-14 TW TW096121620A patent/TW200817385A/zh unknown
- 2007-06-29 US US11/771,198 patent/US7820707B2/en active Active
- 2007-07-02 AR ARP070102955A patent/AR061792A1/es unknown
- 2007-07-02 CN CN2007800248081A patent/CN101484448B/zh not_active Expired - Fee Related
- 2007-07-02 EP EP07801415.6A patent/EP2041124B1/en active Active
- 2007-07-02 NZ NZ573325A patent/NZ573325A/en unknown
- 2007-07-02 AU AU2007271469A patent/AU2007271469B2/en not_active Ceased
- 2007-07-02 KR KR1020087031534A patent/KR20090027672A/ko not_active Withdrawn
- 2007-07-02 MX MX2008016494A patent/MX2008016494A/es active IP Right Grant
- 2007-07-02 JP JP2009517024A patent/JP2009541404A/ja not_active Ceased
- 2007-07-02 CA CA002655680A patent/CA2655680A1/en not_active Abandoned
- 2007-07-02 WO PCT/EP2007/005851 patent/WO2008003452A1/en not_active Ceased
- 2007-07-03 PE PE2007000848A patent/PE20080378A1/es not_active Application Discontinuation
-
2008
- 2008-11-28 ZA ZA200810165A patent/ZA200810165B/xx unknown
- 2008-12-31 IL IL196302A patent/IL196302A0/en unknown
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