JP2009539846A - Ｎ−［５−［［［５−（１，１−ジメチルエチル）−２−オキサゾリル］メチル］チオ］−２−チアゾリル］−４−ピペリジンカルボキサミドの結晶形 - Google Patents

Ｎ−［５−［［［５−（１，１−ジメチルエチル）−２−オキサゾリル］メチル］チオ］−２−チアゾリル］−４−ピペリジンカルボキサミドの結晶形 Download PDF

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JP2009539846A
JP2009539846A JP2009514368A JP2009514368A JP2009539846A JP 2009539846 A JP2009539846 A JP 2009539846A JP 2009514368 A JP2009514368 A JP 2009514368A JP 2009514368 A JP2009514368 A JP 2009514368A JP 2009539846 A JP2009539846 A JP 2009539846A
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compound
powder
ray diffraction
diffraction pattern
temperature
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ゼット．ゴウゴウタス ジャクク
エフ．マルレイ マリ
ディー．ディマルコ ジョフン
キム ソオジン
クイアオ ハイ‐ユン
ナライン ミスラ ラジェ
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ブリストル−ミエルス スクイッブ カンパニー
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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  • Physical Education & Sports Medicine (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Communicable Diseases (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
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  • Molecular Biology (AREA)
  • Urology & Nephrology (AREA)
  • Biotechnology (AREA)
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  • Hospice & Palliative Care (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Obesity (AREA)
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JP2009514368A 2006-06-06 2007-06-06 Ｎ−［５−［［［５−（１，１−ジメチルエチル）−２−オキサゾリル］メチル］チオ］−２−チアゾリル］−４−ピペリジンカルボキサミドの結晶形 Pending JP2009539846A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US81148206P 2006-06-06 2006-06-06
PCT/US2007/013384 WO2007146039A2 (en) 2006-06-06 2007-06-06 Crystalline forms of n-[5-[[[5-(1,1-dimethylethyl)-2-oxazolyl]methyl] thio]-2-thiazolyl]-4-piperidinecarboxamide

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JP2009539846A true JP2009539846A (ja) 2009-11-19
JP2009539846A5 JP2009539846A5 (enExample) 2010-07-29

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Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008036954A1 (en) * 2006-09-21 2008-03-27 Sunesis Pharmaceuticals, Inc. Use of n- [5- [ [ [5- (1, 1-dimethylethyl) -2-oxazoyl] methyl] thio] -2-thiazolyl] -4-piperidinecarboxamide
KR101643280B1 (ko) * 2014-09-02 2016-07-28 한국원자력의학원 항암 효과, 방사선 병용치료 효과 및 당뇨병 치료 효과를 갖는 피페리딘카복사마이드 유도체 및 이의 의학적 용도

Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2002507196A (ja) * 1997-05-29 2002-03-05 レオ・ファーマシューティカル・プロダクツ・リミテッド・アクティーゼルスカブ（レーベンス・ケミスケ・ファブリック・プロデュクチオンスアクティーゼルスカブ） 細胞増殖抑制剤としてのシアノグアニジン
JP2002518399A (ja) * 1998-06-15 2002-06-25 サノフィ−サンテラボ 多形クロピドグレル硫酸水素塩フォーム
US6515004B1 (en) * 1999-12-15 2003-02-04 Bristol-Myers Squibb Company N-[5-[[[5-alkyl-2-oxazolyl]methyl]thio]-2-thiazolyl]-carboxamide inhibitors of cyclin dependent kinases
JP2003506433A (ja) * 1999-08-10 2003-02-18 ロンザ ア−ゲ− ジシアネートカルコンおよびその製造方法
JP2004509857A (ja) * 2000-07-26 2004-04-02 ブリストル−マイヤーズ　スクイブ　カンパニー サイクリン依存性キナーゼのｎ−［５−［［［５−アルキル−２−オキサゾリル］メチル］チオ］−２−チアゾリル］カルボキサミドインヒビター
JP2004269547A (ja) * 1997-02-27 2004-09-30 Pfizer Inc キノキサリンジオン類の製造方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6262096B1 (en) * 1997-11-12 2001-07-17 Bristol-Myers Squibb Company Aminothiazole inhibitors of cyclin dependent kinases
US6414156B2 (en) * 1998-10-21 2002-07-02 Bristol-Myers Squibb Company Process for preparing azacycloalkanoylaminothiazoles
US6534531B2 (en) * 2000-04-27 2003-03-18 Bristol-Myers Squibb Company Methods for preventing and treating alopecia induced by chemotherapy or radiotherapy

Patent Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2004269547A (ja) * 1997-02-27 2004-09-30 Pfizer Inc キノキサリンジオン類の製造方法
JP2002507196A (ja) * 1997-05-29 2002-03-05 レオ・ファーマシューティカル・プロダクツ・リミテッド・アクティーゼルスカブ（レーベンス・ケミスケ・ファブリック・プロデュクチオンスアクティーゼルスカブ） 細胞増殖抑制剤としてのシアノグアニジン
JP2002518399A (ja) * 1998-06-15 2002-06-25 サノフィ−サンテラボ 多形クロピドグレル硫酸水素塩フォーム
JP2003506433A (ja) * 1999-08-10 2003-02-18 ロンザ ア−ゲ− ジシアネートカルコンおよびその製造方法
US6515004B1 (en) * 1999-12-15 2003-02-04 Bristol-Myers Squibb Company N-[5-[[[5-alkyl-2-oxazolyl]methyl]thio]-2-thiazolyl]-carboxamide inhibitors of cyclin dependent kinases
JP2004509857A (ja) * 2000-07-26 2004-04-02 ブリストル−マイヤーズ　スクイブ　カンパニー サイクリン依存性キナーゼのｎ−［５−［［［５−アルキル−２−オキサゾリル］メチル］チオ］−２−チアゾリル］カルボキサミドインヒビター

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WO2007146039A3 (en) 2008-07-17
WO2007146039A2 (en) 2007-12-21

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