JP2009529541A5 - - Google Patents

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Publication number
JP2009529541A5
JP2009529541A5 JP2008558554A JP2008558554A JP2009529541A5 JP 2009529541 A5 JP2009529541 A5 JP 2009529541A5 JP 2008558554 A JP2008558554 A JP 2008558554A JP 2008558554 A JP2008558554 A JP 2008558554A JP 2009529541 A5 JP2009529541 A5 JP 2009529541A5
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JP
Japan
Prior art keywords
group
treatment
prevention
pharmaceutical formulation
pharmaceutical preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2008558554A
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English (en)
Japanese (ja)
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JP2009529541A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2007/063699 external-priority patent/WO2007104053A2/en
Publication of JP2009529541A publication Critical patent/JP2009529541A/ja
Publication of JP2009529541A5 publication Critical patent/JP2009529541A5/ja
Pending legal-status Critical Current

Links

JP2008558554A 2006-03-09 2007-03-09 代謝性障害治療のための８−ヘテロアリ−ルプリンのｍｎｋ２阻害剤 Pending JP2009529541A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US78080006P 2006-03-09 2006-03-09
PCT/US2007/063699 WO2007104053A2 (en) 2006-03-09 2007-03-09 8-heteroarylpurine mnk2 inhibitors for treating metabolic disorders

Publications (2)

Publication Number Publication Date
JP2009529541A JP2009529541A (ja) 2009-08-20
JP2009529541A5 true JP2009529541A5 (OSRAM) 2010-04-30

Family

ID=38371082

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008558554A Pending JP2009529541A (ja) 2006-03-09 2007-03-09 代謝性障害治療のための８−ヘテロアリ−ルプリンのｍｎｋ２阻害剤

Country Status (12)

Country Link
US (2) US7951803B2 (OSRAM)
EP (1) EP1991547A2 (OSRAM)
JP (1) JP2009529541A (OSRAM)
KR (1) KR20080107466A (OSRAM)
CN (1) CN101454325A (OSRAM)
AU (1) AU2007222982A1 (OSRAM)
BR (1) BRPI0709007A2 (OSRAM)
CA (1) CA2646429A1 (OSRAM)
EA (1) EA014907B1 (OSRAM)
MX (1) MX2008011525A (OSRAM)
WO (1) WO2007104053A2 (OSRAM)
ZA (1) ZA200807715B (OSRAM)

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US20130065883A1 (en) 2010-02-18 2013-03-14 Centro Nacional de Investigaceiones Oncologicas (CNIO) Triazolo [4, 5- B] Pyridin Derivatives
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US9133123B2 (en) 2010-04-23 2015-09-15 Cytokinetics, Inc. Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use
EP2582709B1 (de) 2010-06-18 2018-01-24 Sanofi Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen
US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
TW201215387A (en) 2010-07-05 2012-04-16 Sanofi Aventis Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament
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US8871758B2 (en) 2011-03-08 2014-10-28 Sanofi Tetrasubstituted oxathiazine derivatives, method for producing them, their use as medicine and drug containing said derivatives and the use thereof
EP2683704B1 (de) 2011-03-08 2014-12-17 Sanofi Verzweigte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
EP2683705B1 (de) 2011-03-08 2015-04-22 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
US8710050B2 (en) 2011-03-08 2014-04-29 Sanofi Di and tri- substituted oxathiazine derivatives, method for the production, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
EP2567959B1 (en) 2011-09-12 2014-04-16 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
EP2760862B1 (en) 2011-09-27 2015-10-21 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
GB201205669D0 (en) 2012-03-30 2012-05-16 Agency Science Tech & Res Bicyclic heterocyclic derivatives as mnk2 and mnk2 modulators and uses thereof
US10280168B2 (en) 2012-03-30 2019-05-07 Agency For Science, Technology And Research Bicyclic heteroaryl derivatives as MNK1 and MNK2 modulators and uses thereof
ES2635262T3 (es) 2012-11-09 2017-10-03 Evotec International Gmbh Quinazolinas sustituidas con sulfoximina para composiciones farmacéuticas
US20150051208A1 (en) 2013-08-14 2015-02-19 Boehringer Ingelheim International Gmbh Pyridinones
JP6457523B2 (ja) 2013-12-04 2019-01-23 エヴォテック・インターナショナル・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＥｖｏｔｅｃ Ｉｎｔｅｒｎａｔｉｏｎａｌ ＧｍｂＨ 医薬組成物のためのスルホキシイミン置換キナゾリン
WO2015091156A1 (en) 2013-12-17 2015-06-25 Boehringer Ingelheim International Gmbh Sulfoximine substituted pyrrolotriazines for pharmaceutical compositions
AU2015257917C1 (en) 2014-05-07 2019-03-14 Evotec International Gmbh Sulfoximine substituted quinazolines for pharmaceutical compositions
CN105001096B (zh) * 2015-07-21 2017-07-21 沈阳化工研究院有限公司 一种制备4‑氨基‑n‑烷基苄胺的方法
CN106008506B (zh) * 2016-06-27 2018-02-13 山东大学 取代嘌呤类衍生物及其制备方法与应用
CN120284862A (zh) 2018-12-07 2025-07-11 纽罗克里生物科学有限公司 用于治疗先天性肾上腺皮质增生症的crf1受体拮抗剂、其药物制剂和固体形式
US12383536B2 (en) 2019-09-27 2025-08-12 Neurocrine Biosciences, Inc. CRF receptor antagonists and methods of use
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