JP2009526776A5 - - Google Patents

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Publication number
JP2009526776A5
JP2009526776A5 JP2008553787A JP2008553787A JP2009526776A5 JP 2009526776 A5 JP2009526776 A5 JP 2009526776A5 JP 2008553787 A JP2008553787 A JP 2008553787A JP 2008553787 A JP2008553787 A JP 2008553787A JP 2009526776 A5 JP2009526776 A5 JP 2009526776A5
Authority
JP
Japan
Prior art keywords
alkyl
group
alkoxy
cycloalkyl
pain
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
JP2008553787A
Other languages
English (en)
Japanese (ja)
Other versions
JP2009526776A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2007/051396 external-priority patent/WO2007093600A1/en
Publication of JP2009526776A publication Critical patent/JP2009526776A/ja
Publication of JP2009526776A5 publication Critical patent/JP2009526776A5/ja
Abandoned legal-status Critical Current

Links

JP2008553787A 2006-02-14 2007-02-13 新規なジアザビシクロアルカン誘導体及びその医療上の使用 Abandoned JP2009526776A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DKPA200600210 2006-02-14
US77332506P 2006-02-15 2006-02-15
PCT/EP2007/051396 WO2007093600A1 (en) 2006-02-14 2007-02-13 Novel diazabicycloalkane derivatives and their medical use

Publications (2)

Publication Number Publication Date
JP2009526776A JP2009526776A (ja) 2009-07-23
JP2009526776A5 true JP2009526776A5 (OSRAM) 2010-04-02

Family

ID=38137474

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008553787A Abandoned JP2009526776A (ja) 2006-02-14 2007-02-13 新規なジアザビシクロアルカン誘導体及びその医療上の使用

Country Status (6)

Country Link
US (1) US20090075983A1 (OSRAM)
EP (1) EP1987033B1 (OSRAM)
JP (1) JP2009526776A (OSRAM)
AU (1) AU2007216531A1 (OSRAM)
CA (1) CA2641767A1 (OSRAM)
WO (1) WO2007093600A1 (OSRAM)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101878204A (zh) * 2007-11-30 2010-11-03 神经研究公司 新颖的羧酸4-苯基偶氮-苯基酯衍生物及其作为单胺神经递质再摄取抑制剂的用途
US20110118268A1 (en) 2008-03-11 2011-05-19 Dan Peters Novel 1,4-diaza-bicyclo[3.2.1]octane derivatives useful as nicotinic acetylcholine receptor modulators
FR2931823B1 (fr) 2008-06-02 2012-08-17 Sanofi Aventis Sel de fumarate du 1,4-diazabicyclo°3.2.2!nonane-carboxylate de 4-bromophenyle, ses formes cristallines, leur preparation et leur utilisation en therapeutique
FR2931677B1 (fr) * 2008-06-02 2010-08-20 Sanofi Aventis Association d'un agoniste partiel des recepteurs nicotiniques et d'un inhibiteur d'acetylcholinesterase, composition la contenant et son utilisation dans le traitement des troubles cognitifs
AR072297A1 (es) 2008-06-27 2010-08-18 Novartis Ag Derivados de indol-2-il-piridin-3-ilo, composicion farmaceutica que los comprende y su uso en medicamentos para el tratamiento de enfermedades mediadas por la sintasa aldosterona.
JO3250B1 (ar) 2009-09-22 2018-09-16 Novartis Ag إستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7
US8759535B2 (en) 2010-02-18 2014-06-24 High Point Pharmaceuticals, Llc Substituted fused imidazole derivatives, pharmaceutical compositions, and methods of use thereof
DK2536285T3 (en) 2010-02-18 2018-07-16 Vtv Therapeutics Llc Substituted fused imidazole derivatives, pharmaceutical compositions and methods for their use
WO2016089648A1 (en) 2014-12-01 2016-06-09 Vtv Therapeutics Llc Bach 1 inhibitors in combination with nrf2 activators and pharmaceutical compositions thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1147112E (pt) * 1999-01-29 2004-03-31 Abbott Lab Derivados diazabiciclicos como liganos nicotinicos do receptor de acetilcolina
FR2791678B1 (fr) * 1999-03-30 2001-05-04 Synthelabo Derives de 1,4-diazabicyclo [3.2.2] nonane-4-carboxylates et -carboxamides, leur preparation et leur application en therapeutique
US20020086871A1 (en) * 2000-12-29 2002-07-04 O'neill Brian Thomas Pharmaceutical composition for the treatment of CNS and other disorders
DE60216830T2 (de) * 2001-02-06 2007-06-14 Pfizer Products Inc., Groton Pharmazeutische Zusammensetzungen zur Behandlung von Störungen des ZNS oder anderen Erkrankungen
JP2005505506A (ja) * 2001-06-12 2005-02-24 イーラン ファーマスーティカルズ、インコーポレイテッド アルツハイマー病の治療に有用な大環状分子
EP1863819B1 (en) * 2005-02-16 2011-01-12 NeuroSearch A/S Diazabicyclic aryl derivatives and their use as chinolinergic ligands at the nicotinic acetylcholine receptors

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