JP2009514935A - 新規化合物 - Google Patents

新規化合物 Download PDF

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Publication number
JP2009514935A
JP2009514935A JP2008539486A JP2008539486A JP2009514935A JP 2009514935 A JP2009514935 A JP 2009514935A JP 2008539486 A JP2008539486 A JP 2008539486A JP 2008539486 A JP2008539486 A JP 2008539486A JP 2009514935 A JP2009514935 A JP 2009514935A
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JP
Japan
Prior art keywords
methyl
phenyl
halogen
chloro
alkyl
Prior art date
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Withdrawn
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JP2008539486A
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English (en)
Japanese (ja)
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JP2009514935A5 (enExample
Inventor
ティモシー・ルーカー
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AstraZeneca AB
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AstraZeneca AB
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Filing date
Publication date
Priority claimed from GB0522619A external-priority patent/GB0522619D0/en
Priority claimed from GB0607353A external-priority patent/GB0607353D0/en
Application filed by AstraZeneca AB filed Critical AstraZeneca AB
Publication of JP2009514935A publication Critical patent/JP2009514935A/ja
Publication of JP2009514935A5 publication Critical patent/JP2009514935A5/ja
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/26—Sulfur atoms
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    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Ophthalmology & Optometry (AREA)
  • Obesity (AREA)
  • Psychiatry (AREA)
  • Biochemistry (AREA)
  • Hospice & Palliative Care (AREA)
  • Emergency Medicine (AREA)
  • Gastroenterology & Hepatology (AREA)
JP2008539486A 2005-11-05 2006-11-01 新規化合物 Withdrawn JP2009514935A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0522619A GB0522619D0 (en) 2005-11-05 2005-11-05 Novel compounds
GB0607353A GB0607353D0 (en) 2006-04-12 2006-04-12 Novel Compounds
PCT/GB2006/004075 WO2007052023A2 (en) 2005-11-05 2006-11-01 Novel compounds

Publications (2)

Publication Number Publication Date
JP2009514935A true JP2009514935A (ja) 2009-04-09
JP2009514935A5 JP2009514935A5 (enExample) 2009-10-22

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Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008539486A Withdrawn JP2009514935A (ja) 2005-11-05 2006-11-01 新規化合物

Country Status (4)

Country Link
US (1) US20080255150A1 (enExample)
EP (1) EP1948630A2 (enExample)
JP (1) JP2009514935A (enExample)
WO (1) WO2007052023A2 (enExample)

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2020500178A (ja) * 2016-11-16 2020-01-09 ルンドベック ラ ホーヤ リサーチ センター，インク． Ｍａｇｌ阻害剤
JP2020504707A (ja) * 2016-11-16 2020-02-13 ルンドベック ラ ホーヤ リサーチ センター，インク． Ｍａｇｌ阻害剤
US11332453B2 (en) 2018-05-15 2022-05-17 H. Lundbeck A/S MAGL inhibitors
US11530189B2 (en) 2012-01-06 2022-12-20 H. Lundbecka/S Carbamate compounds and methods of making and using same
US12378219B2 (en) 2022-05-04 2025-08-05 H. Lundbeck A/S Crystalline forms of a MAGL inhibitor

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0301010D0 (sv) * 2003-04-07 2003-04-07 Astrazeneca Ab Novel compounds
SE0301009D0 (sv) * 2003-04-07 2003-04-07 Astrazeneca Ab Novel compounds
SA04250253B1 (ar) 2003-08-21 2009-11-10 استرازينيكا ايه بي احماض فينوكسي اسيتيك مستبدلة باعتبارها مركبات صيدلانية لعلاج الامراض التنفسية مثل الربو ومرض الانسداد الرئوي المزمن
GB0415320D0 (en) * 2004-07-08 2004-08-11 Astrazeneca Ab Novel compounds
GB0418830D0 (en) * 2004-08-24 2004-09-22 Astrazeneca Ab Novel compounds
GB0422057D0 (en) * 2004-10-05 2004-11-03 Astrazeneca Ab Novel compounds
ATE517085T1 (de) 2004-11-23 2011-08-15 Astrazeneca Ab Zur behandlung von atemwegserkrankungen geeignete phenoxyessigsäurederivate
US8148572B2 (en) 2005-10-06 2012-04-03 Astrazeneca Ab Compounds
TW200745003A (en) 2005-10-06 2007-12-16 Astrazeneca Ab Novel compounds
ES2380683T3 (es) * 2005-12-15 2012-05-17 Astrazeneca Ab Difenil-éteres, -amidas, -sulfuros y - metanos sustituidos para el tratamiento de la enfermedad respiratoria
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