JP2009503089A5 - - Google Patents

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Publication number
JP2009503089A5
JP2009503089A5 JP2008525104A JP2008525104A JP2009503089A5 JP 2009503089 A5 JP2009503089 A5 JP 2009503089A5 JP 2008525104 A JP2008525104 A JP 2008525104A JP 2008525104 A JP2008525104 A JP 2008525104A JP 2009503089 A5 JP2009503089 A5 JP 2009503089A5
Authority
JP
Japan
Prior art keywords
alkyl
substituted
aryl
heterocycle
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2008525104A
Other languages
English (en)
Japanese (ja)
Other versions
JP2009503089A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2006/029877 external-priority patent/WO2007019130A2/en
Publication of JP2009503089A publication Critical patent/JP2009503089A/ja
Publication of JP2009503089A5 publication Critical patent/JP2009503089A5/ja
Pending legal-status Critical Current

Links

JP2008525104A 2005-08-04 2006-07-28 Hivインテグラーゼ阻害薬 Pending JP2009503089A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US70534205P 2005-08-04 2005-08-04
PCT/US2006/029877 WO2007019130A2 (en) 2005-08-04 2006-07-28 Hiv integrase inhibitors

Publications (2)

Publication Number Publication Date
JP2009503089A JP2009503089A (ja) 2009-01-29
JP2009503089A5 true JP2009503089A5 (https=) 2009-09-03

Family

ID=37727857

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008525104A Pending JP2009503089A (ja) 2005-08-04 2006-07-28 Hivインテグラーゼ阻害薬

Country Status (4)

Country Link
US (1) US20080234231A1 (https=)
EP (1) EP1909578A4 (https=)
JP (1) JP2009503089A (https=)
WO (1) WO2007019130A2 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8283366B2 (en) 2010-01-22 2012-10-09 Ambrilia Biopharma, Inc. Derivatives of pyridoxine for inhibiting HIV integrase
US11116737B1 (en) 2020-04-10 2021-09-14 University Of Georgia Research Foundation, Inc. Methods of using probenecid for treatment of coronavirus infections

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6225318B1 (en) * 1996-10-17 2001-05-01 Pfizer Inc 4-aminoquinazolone derivatives
CA2425440C (en) * 2000-10-12 2010-04-13 Merck & Co., Inc. Aza- and polyaza-naphthalenyl carboxamides useful as hiv integrase inhibitors
US6919351B2 (en) * 2000-10-12 2005-07-19 Merck & Co., Inc. Aza-and polyaza-naphthalenyl-carboxamides useful as HIV integrase inhibitors
EP1467970B1 (en) * 2002-01-17 2007-08-22 Merck & Co., Inc. Hydroxynaphthyridinone carboxamides useful as hiv integrase inhibitors
EP1541558B1 (en) * 2002-08-13 2008-08-13 Shionogi & Co., Ltd. Heterocyclic compounds having hiv integrase inhibitory activity
US20040157804A1 (en) * 2002-10-16 2004-08-12 Gilead Sciences, Inc. Pre-organized tricyclic integrase inhibitor compounds
TW200505902A (en) * 2003-03-20 2005-02-16 Schering Corp Cannabinoid receptor ligands
US20070185007A1 (en) * 2003-09-19 2007-08-09 Haolun Jin Aza-quinolinol phosphonate integrase inhibitor compounds
CA2555176A1 (en) * 2004-02-11 2005-08-25 Smithkline Beecham Corporation Hiv integrase inhibitors

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