JP2008531559A - スピロ−複素環式クロマン、チオクロマン及びジヒドロキノリン - Google Patents
スピロ−複素環式クロマン、チオクロマン及びジヒドロキノリン Download PDFInfo
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/10—Spiro-condensed systems
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
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Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Immunology (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
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- Physical Education & Sports Medicine (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Rheumatology (AREA)
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- Vascular Medicine (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US65671105P | 2005-02-25 | 2005-02-25 | |
| US65674805P | 2005-02-25 | 2005-02-25 | |
| PCT/US2005/044713 WO2006093548A1 (en) | 2005-02-25 | 2005-12-09 | Spiro-heterocyclic chromans, thiochromans and dihydroquinolines |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2008531559A true JP2008531559A (ja) | 2008-08-14 |
| JP2008531559A5 JP2008531559A5 (enExample) | 2009-01-15 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007557016A Withdrawn JP2008531559A (ja) | 2005-02-25 | 2005-12-09 | スピロ−複素環式クロマン、チオクロマン及びジヒドロキノリン |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20080207588A1 (enExample) |
| EP (1) | EP1856079A4 (enExample) |
| JP (1) | JP2008531559A (enExample) |
| AU (1) | AU2005328328A1 (enExample) |
| BR (1) | BRPI0520097A2 (enExample) |
| CA (1) | CA2600004A1 (enExample) |
| MX (1) | MX2007010328A (enExample) |
| WO (1) | WO2006093548A1 (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2589363A1 (en) | 2004-12-13 | 2006-06-22 | Eli Lilly And Company | Spiro derivatives as lipoxygenase inhibitors |
| CA2924141C (en) | 2013-08-22 | 2022-06-07 | The General Hospital Corporation | 5-amino 4-cyano substituted oxazole and thiazole derivatives as inhibitors of human 12/15-lipoxygenase |
| BR122019007990B1 (pt) | 2013-11-18 | 2021-05-04 | Forma Therapeutics, Inc | Composto, e, composição farmacêutica |
| RU2720237C2 (ru) | 2013-11-18 | 2020-04-28 | Форма Терапеутикс, Инк. | Композиции, содержащие бензопиперазин, в качестве ингибиторов бромодоменов вет |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
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| CA1261835A (en) | 1984-08-20 | 1989-09-26 | Masaaki Toda | (fused) benz(thio)amides |
| GB8626344D0 (en) | 1986-11-04 | 1986-12-03 | Zyma Sa | Bicyclic compounds |
| US5059609A (en) | 1987-10-19 | 1991-10-22 | Pfizer Inc. | Substituted tetralins, chromans and related compounds in the treatment of asthma, arthritis and related diseases |
| US4950684A (en) | 1988-05-20 | 1990-08-21 | G. D. Searle & Co. | 2,2-di-substituted benzopyran leukotriene-D4 antagonists |
| US5015661A (en) | 1988-08-09 | 1991-05-14 | Hoffmann-La Roche Inc. | Chromanes and their pharmaceutical compositions and methods |
| US5250547A (en) * | 1991-08-29 | 1993-10-05 | Syntex (U.S.A.) Inc. | Benzopyran derivatives |
| EP0543417A1 (en) | 1991-11-22 | 1993-05-26 | Lipogenics, Incorporated | Tocotrienols and tocotrienol-like compounds and methods for their use |
| FR2695387B1 (fr) | 1992-09-09 | 1994-10-21 | Adir | Nouveaux composés benzopyraniques, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent. |
| US5686389A (en) * | 1994-04-13 | 1997-11-11 | City Of Hope | Growth inhibition of Erwinia amylovora |
| CN1160399A (zh) | 1994-10-13 | 1997-09-24 | 美国辉瑞有限公司 | 苯并吡喃和苯并稠合化合物、其制备方法和它们作为白三烯b4(ltb4)拮抗剂的用途 |
| MX9702734A (es) | 1994-10-13 | 1997-06-28 | Pfizer | Benzopirano y compuestos benzocondensados, su preparacion y su uso como antagonistas de leucotrieno b4 (ltb4). |
| US5925673A (en) | 1994-12-23 | 1999-07-20 | Alcon Laboratories, Inc. | Benzofurans and benzopyrans as cytoprotective agents |
| TW472051B (en) * | 1997-05-23 | 2002-01-11 | Chugai Pharmaceutical Co Ltd | 2,3-dihydrobenzofuran derivatives |
| CA2589363A1 (en) * | 2004-12-13 | 2006-06-22 | Eli Lilly And Company | Spiro derivatives as lipoxygenase inhibitors |
| AU2005328327A1 (en) * | 2005-02-25 | 2006-09-08 | Galileo Pharmaceuticals, Inc. | Novel lipoxygenase inhibitors |
-
2005
- 2005-12-09 CA CA002600004A patent/CA2600004A1/en not_active Abandoned
- 2005-12-09 EP EP05853595A patent/EP1856079A4/en not_active Withdrawn
- 2005-12-09 WO PCT/US2005/044713 patent/WO2006093548A1/en not_active Ceased
- 2005-12-09 BR BRPI0520097-0A patent/BRPI0520097A2/pt not_active IP Right Cessation
- 2005-12-09 AU AU2005328328A patent/AU2005328328A1/en not_active Abandoned
- 2005-12-09 JP JP2007557016A patent/JP2008531559A/ja not_active Withdrawn
- 2005-12-09 US US11/814,878 patent/US20080207588A1/en not_active Abandoned
- 2005-12-09 MX MX2007010328A patent/MX2007010328A/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| WO2006093548A1 (en) | 2006-09-08 |
| EP1856079A4 (en) | 2008-12-31 |
| AU2005328328A1 (en) | 2006-09-08 |
| CA2600004A1 (en) | 2006-09-08 |
| MX2007010328A (es) | 2008-03-13 |
| BRPI0520097A2 (pt) | 2009-08-25 |
| US20080207588A1 (en) | 2008-08-28 |
| EP1856079A1 (en) | 2007-11-21 |
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