JP2008511541A - 胃腸障害処置用プロスタグランジン誘導体 - Google Patents
胃腸障害処置用プロスタグランジン誘導体 Download PDFInfo
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- JP2008511541A JP2008511541A JP2007511111A JP2007511111A JP2008511541A JP 2008511541 A JP2008511541 A JP 2008511541A JP 2007511111 A JP2007511111 A JP 2007511111A JP 2007511111 A JP2007511111 A JP 2007511111A JP 2008511541 A JP2008511541 A JP 2008511541A
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- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/94—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems condensed with rings other than six-membered or with ring systems containing such rings
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/557—Eicosanoids, e.g. leukotrienes or prostaglandins
- A61K31/558—Eicosanoids, e.g. leukotrienes or prostaglandins having heterocyclic rings containing oxygen as the only ring hetero atom, e.g. thromboxanes
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- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A—HUMAN NECESSITIES
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
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- Bioinformatics & Cheminformatics (AREA)
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- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pyrane Compounds (AREA)
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| US60652104P | 2004-09-02 | 2004-09-02 | |
| US66631705P | 2005-03-30 | 2005-03-30 | |
| US66659305P | 2005-03-31 | 2005-03-31 | |
| PCT/JP2005/016464 WO2006025599A1 (en) | 2004-09-02 | 2005-09-01 | Prostaglandin derivatives for treating gastrointestinal disorder |
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| JP2012232180A Division JP2013049688A (ja) | 2004-09-02 | 2012-10-19 | 胃腸障害処置用プロスタグランジン誘導体 |
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| JP2008511541A true JP2008511541A (ja) | 2008-04-17 |
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| JP2012232180A Withdrawn JP2013049688A (ja) | 2004-09-02 | 2012-10-19 | 胃腸障害処置用プロスタグランジン誘導体 |
| JP2015102184A Expired - Lifetime JP6408426B2 (ja) | 2004-09-02 | 2015-05-19 | 胃腸障害処置用プロスタグランジン誘導体 |
| JP2018102339A Withdrawn JP2018150354A (ja) | 2004-09-02 | 2018-05-29 | 胃腸障害処置用プロスタグランジン誘導体 |
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| JP2012232180A Withdrawn JP2013049688A (ja) | 2004-09-02 | 2012-10-19 | 胃腸障害処置用プロスタグランジン誘導体 |
| JP2015102184A Expired - Lifetime JP6408426B2 (ja) | 2004-09-02 | 2015-05-19 | 胃腸障害処置用プロスタグランジン誘導体 |
| JP2018102339A Withdrawn JP2018150354A (ja) | 2004-09-02 | 2018-05-29 | 胃腸障害処置用プロスタグランジン誘導体 |
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| TW (1) | TWI387454B (cg-RX-API-DMAC7.html) |
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| PT1562604E (pt) * | 2002-10-23 | 2012-04-09 | Sucampo Ag | Compostos de prostaglandina para o tratamento de obesidade |
| EP1641462B1 (en) * | 2003-07-03 | 2010-11-24 | Sucampo AG | Enteric coated composition comprising prostaglandin analogs as chloride channel opener |
| EP1984027B1 (en) | 2006-01-24 | 2015-12-30 | R-Tech Ueno, Ltd. | Pharmaceutical composition comprising a bi-cyclic compound and method for stabilizing the bi-cyclic compound |
| US20090030072A1 (en) * | 2007-07-03 | 2009-01-29 | Sucampo Ag | Pharmaceutical combination of opioid and prostaglandin compound |
| CA2870252A1 (en) * | 2012-04-23 | 2013-10-31 | Sucampo Ag | Method for treating irritable bowel syndrome with diarrhea |
| AU2014213251B2 (en) * | 2013-02-04 | 2017-07-20 | Taisho Pharmaceutical Co., Ltd. | Prophylactic or therapeutic drug for constipation |
| WO2014159679A1 (en) | 2013-03-12 | 2014-10-02 | The United States Of America, As Represented By The Secretary, Department Of Health & Human Services | Methods for using lubiprostone to absorb fluid from the subretinal space |
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| WO2002089812A1 (en) * | 2001-05-02 | 2002-11-14 | Sucampo Ag | Composition for treating drug-induced constipation with 15-keto-prostaglandins |
| WO2003041716A1 (en) * | 2001-11-14 | 2003-05-22 | Sucampo Ag | Dosage unit comprising a prostaglandin analog for treating constipation |
| JP2004508327A (ja) * | 2000-09-05 | 2004-03-18 | スカンポ・アクチェンゲゼルシャフト | 下剤組成物 |
| WO2004060377A1 (en) * | 2002-12-27 | 2004-07-22 | Sucampo Ag | Derivatives of prostaglandins for treating abdominal discomfort |
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| US5166174A (en) | 1987-01-28 | 1992-11-24 | K.K. Ueno Seiyaku Oyo Kenkyujo | Prostaglandins E and anti-ulcers containing same |
| US5380709A (en) | 1987-01-28 | 1995-01-10 | K.K. Ueno Seiyaku Oyo Kenkyujo | Prostaglandins E and anti ulcers containing same |
| US5225439A (en) | 1987-01-28 | 1993-07-06 | K.K. Ueno Seiyaku Oyo Kenkyujo | Prostaglandins E and anti ulcers containing same |
| US5317032A (en) * | 1987-10-02 | 1994-05-31 | Kabushiki Kaisha Ueno Seiyaku Oyo Kenkyujo | Prostaglandin cathartic |
| JP4332316B2 (ja) | 1999-10-15 | 2009-09-16 | スキャンポ・アーゲー | 二環式化合物組成物およびその安定化方法 |
| PT1389116E (pt) | 2001-05-18 | 2008-04-11 | Sucampo Ag | Composição de indução catártica |
| BR0212233A (pt) * | 2001-08-31 | 2004-10-05 | Sucampo Ag | Abridor de canal de cloreto |
| US7732487B2 (en) | 2001-11-19 | 2010-06-08 | Sucampo Ag | Method for treating a disease or condition responsive to opening of C1C-2 channel |
| EP1641462B1 (en) | 2003-07-03 | 2010-11-24 | Sucampo AG | Enteric coated composition comprising prostaglandin analogs as chloride channel opener |
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2005
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- 2005-09-01 KR KR1020077004900A patent/KR20070048221A/ko not_active Ceased
- 2005-09-01 AU AU2005278323A patent/AU2005278323B2/en not_active Expired
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- 2005-09-01 KR KR1020137034994A patent/KR20140019006A/ko not_active Ceased
- 2005-09-01 BR BRPI0514891-0A patent/BRPI0514891A/pt not_active Application Discontinuation
- 2005-09-01 KR KR1020167036382A patent/KR20170003712A/ko not_active Ceased
- 2005-09-01 CA CA002577284A patent/CA2577284A1/en not_active Withdrawn
- 2005-09-01 CN CN2012103704021A patent/CN102885821A/zh active Pending
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- 2005-09-01 ES ES05782157.1T patent/ES2603381T3/es not_active Expired - Lifetime
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- 2005-09-01 MX MX2007002602A patent/MX2007002602A/es active IP Right Grant
- 2005-09-01 JP JP2007511111A patent/JP2008511541A/ja not_active Withdrawn
- 2005-09-01 US US11/216,012 patent/US8748481B2/en not_active Expired - Lifetime
- 2005-09-01 EP EP05782157.1A patent/EP1791545B1/en not_active Expired - Lifetime
- 2005-09-02 AR ARP050103687A patent/AR050626A1/es not_active Application Discontinuation
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2007
- 2007-02-14 IL IL181332A patent/IL181332A/en not_active IP Right Cessation
- 2007-03-30 NO NO20071704A patent/NO340989B1/no not_active IP Right Cessation
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2012
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2014
- 2014-04-30 US US14/265,801 patent/US20140315994A1/en not_active Abandoned
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2015
- 2015-05-19 JP JP2015102184A patent/JP6408426B2/ja not_active Expired - Lifetime
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2018
- 2018-05-29 JP JP2018102339A patent/JP2018150354A/ja not_active Withdrawn
Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2004508327A (ja) * | 2000-09-05 | 2004-03-18 | スカンポ・アクチェンゲゼルシャフト | 下剤組成物 |
| WO2002089812A1 (en) * | 2001-05-02 | 2002-11-14 | Sucampo Ag | Composition for treating drug-induced constipation with 15-keto-prostaglandins |
| WO2003041716A1 (en) * | 2001-11-14 | 2003-05-22 | Sucampo Ag | Dosage unit comprising a prostaglandin analog for treating constipation |
| WO2004060377A1 (en) * | 2002-12-27 | 2004-07-22 | Sucampo Ag | Derivatives of prostaglandins for treating abdominal discomfort |
Non-Patent Citations (1)
| Title |
|---|
| JPN6011057700; ＳＯＲＢＥＲＡ，Ｌ． ｅｔ ａｌ: 'Ｌｕｂｉｐｒｏｓｔｏｎｅ： Ｔｒｅａｔｍｅｎｔ ｏｆ ｃｏｎｓｔｉｐａｔｉｏｎ ｔｒｅａｔｍｅｎｔ ｏｆ ｉｒｒｉｔａｂｌｅ ｂｏｗｅｌ ｓｙｎｄｒｏｍｅ ｔｒｅａｔｍｅｎｔ ｏｆ ｐｏｓｔｏｐｅｒａ' Ｄｒｕｇｓ ｏｆ ｔｈｅ Ｆｕｔｕｒｅ Ｖｏｌ．２９， Ｎｏ．４, 200404, ｐｐ．３３６-３４１ * |
Also Published As
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| CN102885821A (zh) | 2013-01-23 |
| ES2603381T3 (es) | 2017-02-27 |
| US8748481B2 (en) | 2014-06-10 |
| TWI387454B (zh) | 2013-03-01 |
| AR050626A1 (es) | 2006-11-08 |
| IL181332A0 (en) | 2007-07-04 |
| NZ553434A (en) | 2010-01-29 |
| NO340989B1 (no) | 2017-07-31 |
| JP6408426B2 (ja) | 2018-10-17 |
| KR20070048221A (ko) | 2007-05-08 |
| US20060063830A1 (en) | 2006-03-23 |
| AU2005278323A1 (en) | 2006-03-09 |
| BRPI0514891A (pt) | 2008-06-24 |
| KR20170003712A (ko) | 2017-01-09 |
| KR20180033310A (ko) | 2018-04-02 |
| EP1791545B1 (en) | 2016-08-31 |
| WO2006025599A1 (en) | 2006-03-09 |
| MX2007002602A (es) | 2007-04-25 |
| JP2018150354A (ja) | 2018-09-27 |
| JP2015166377A (ja) | 2015-09-24 |
| AU2005278323B2 (en) | 2011-03-17 |
| NO20071704L (no) | 2007-05-31 |
| EP1791545A1 (en) | 2007-06-06 |
| JP2013049688A (ja) | 2013-03-14 |
| US20140315994A1 (en) | 2014-10-23 |
| CA2577284A1 (en) | 2006-03-09 |
| IL181332A (en) | 2015-09-24 |
| KR20140019006A (ko) | 2014-02-13 |
| TW200612901A (en) | 2006-05-01 |
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