KR20070048221A - 위장 장애 치료를 위한 프로스타글란딘 유도체 - Google Patents

위장 장애 치료를 위한 프로스타글란딘 유도체 Download PDF

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Publication number
KR20070048221A
KR20070048221A KR1020077004900A KR20077004900A KR20070048221A KR 20070048221 A KR20070048221 A KR 20070048221A KR 1020077004900 A KR1020077004900 A KR 1020077004900A KR 20077004900 A KR20077004900 A KR 20077004900A KR 20070048221 A KR20070048221 A KR 20070048221A
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KR
South Korea
Prior art keywords
halogen
alkyl
composition
aryl
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
KR1020077004900A
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English (en)
Korean (ko)
Inventor
류지 우에노
Original Assignee
수캄포 아게
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35229739&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR20070048221(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 수캄포 아게 filed Critical 수캄포 아게
Publication of KR20070048221A publication Critical patent/KR20070048221A/ko
Ceased legal-status Critical Current

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/94Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems condensed with rings other than six-membered or with ring systems containing such rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/557Eicosanoids, e.g. leukotrienes or prostaglandins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/557Eicosanoids, e.g. leukotrienes or prostaglandins
    • A61K31/558Eicosanoids, e.g. leukotrienes or prostaglandins having heterocyclic rings containing oxygen as the only ring hetero atom, e.g. thromboxanes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/10Laxatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nutrition Science (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrane Compounds (AREA)
KR1020077004900A 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체 Ceased KR20070048221A (ko)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US60652104P 2004-09-02 2004-09-02
US60/606,521 2004-09-02
US66631705P 2005-03-30 2005-03-30
US60/666,317 2005-03-30
US66659305P 2005-03-31 2005-03-31
US60/666,593 2005-03-31

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1020137034994A Division KR20140019006A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체

Publications (1)

Publication Number Publication Date
KR20070048221A true KR20070048221A (ko) 2007-05-08

Family

ID=35229739

Family Applications (4)

Application Number Title Priority Date Filing Date
KR1020077004900A Ceased KR20070048221A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체
KR1020137034994A Ceased KR20140019006A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체
KR1020167036382A Ceased KR20170003712A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체
KR1020187008381A Ceased KR20180033310A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체

Family Applications After (3)

Application Number Title Priority Date Filing Date
KR1020137034994A Ceased KR20140019006A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체
KR1020167036382A Ceased KR20170003712A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체
KR1020187008381A Ceased KR20180033310A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체

Country Status (16)

Country Link
US (2) US8748481B2 (cg-RX-API-DMAC7.html)
EP (1) EP1791545B1 (cg-RX-API-DMAC7.html)
JP (4) JP2008511541A (cg-RX-API-DMAC7.html)
KR (4) KR20070048221A (cg-RX-API-DMAC7.html)
CN (1) CN102885821A (cg-RX-API-DMAC7.html)
AR (1) AR050626A1 (cg-RX-API-DMAC7.html)
AU (1) AU2005278323B2 (cg-RX-API-DMAC7.html)
BR (1) BRPI0514891A (cg-RX-API-DMAC7.html)
CA (1) CA2577284A1 (cg-RX-API-DMAC7.html)
ES (1) ES2603381T3 (cg-RX-API-DMAC7.html)
IL (1) IL181332A (cg-RX-API-DMAC7.html)
MX (1) MX2007002602A (cg-RX-API-DMAC7.html)
NO (1) NO340989B1 (cg-RX-API-DMAC7.html)
NZ (1) NZ553434A (cg-RX-API-DMAC7.html)
TW (1) TWI387454B (cg-RX-API-DMAC7.html)
WO (1) WO2006025599A1 (cg-RX-API-DMAC7.html)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1562604E (pt) * 2002-10-23 2012-04-09 Sucampo Ag Compostos de prostaglandina para o tratamento de obesidade
EP1641462B1 (en) * 2003-07-03 2010-11-24 Sucampo AG Enteric coated composition comprising prostaglandin analogs as chloride channel opener
EP1984027B1 (en) 2006-01-24 2015-12-30 R-Tech Ueno, Ltd. Pharmaceutical composition comprising a bi-cyclic compound and method for stabilizing the bi-cyclic compound
US20090030072A1 (en) * 2007-07-03 2009-01-29 Sucampo Ag Pharmaceutical combination of opioid and prostaglandin compound
CA2870252A1 (en) * 2012-04-23 2013-10-31 Sucampo Ag Method for treating irritable bowel syndrome with diarrhea
AU2014213251B2 (en) * 2013-02-04 2017-07-20 Taisho Pharmaceutical Co., Ltd. Prophylactic or therapeutic drug for constipation
WO2014159679A1 (en) 2013-03-12 2014-10-02 The United States Of America, As Represented By The Secretary, Department Of Health & Human Services Methods for using lubiprostone to absorb fluid from the subretinal space

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5166174A (en) 1987-01-28 1992-11-24 K.K. Ueno Seiyaku Oyo Kenkyujo Prostaglandins E and anti-ulcers containing same
US5380709A (en) 1987-01-28 1995-01-10 K.K. Ueno Seiyaku Oyo Kenkyujo Prostaglandins E and anti ulcers containing same
US5225439A (en) 1987-01-28 1993-07-06 K.K. Ueno Seiyaku Oyo Kenkyujo Prostaglandins E and anti ulcers containing same
US5317032A (en) * 1987-10-02 1994-05-31 Kabushiki Kaisha Ueno Seiyaku Oyo Kenkyujo Prostaglandin cathartic
JP4332316B2 (ja) 1999-10-15 2009-09-16 スキャンポ・アーゲー 二環式化合物組成物およびその安定化方法
US6414016B1 (en) * 2000-09-05 2002-07-02 Sucampo, A.G. Anti-constipation composition
TWI302100B (en) 2001-05-02 2008-10-21 Sucampo Ag Composition for treating drug-induced constipation
PT1389116E (pt) 2001-05-18 2008-04-11 Sucampo Ag Composição de indução catártica
BR0212233A (pt) * 2001-08-31 2004-10-05 Sucampo Ag Abridor de canal de cloreto
AR037524A1 (es) * 2001-11-14 2004-11-17 Sucampo Ag Unidad de dosificacion que comprende un analogo de prostaglandina para el tratamiento de la constipacion
US7732487B2 (en) 2001-11-19 2010-06-08 Sucampo Ag Method for treating a disease or condition responsive to opening of C1C-2 channel
KR101164838B1 (ko) * 2002-12-27 2012-07-11 수캄포 아게 복부 불쾌감 치료용 프로스타글랜딘의 유도체
EP1641462B1 (en) 2003-07-03 2010-11-24 Sucampo AG Enteric coated composition comprising prostaglandin analogs as chloride channel opener

Also Published As

Publication number Publication date
CN102885821A (zh) 2013-01-23
ES2603381T3 (es) 2017-02-27
US8748481B2 (en) 2014-06-10
TWI387454B (zh) 2013-03-01
AR050626A1 (es) 2006-11-08
IL181332A0 (en) 2007-07-04
NZ553434A (en) 2010-01-29
NO340989B1 (no) 2017-07-31
JP6408426B2 (ja) 2018-10-17
US20060063830A1 (en) 2006-03-23
AU2005278323A1 (en) 2006-03-09
JP2008511541A (ja) 2008-04-17
BRPI0514891A (pt) 2008-06-24
KR20170003712A (ko) 2017-01-09
KR20180033310A (ko) 2018-04-02
EP1791545B1 (en) 2016-08-31
WO2006025599A1 (en) 2006-03-09
MX2007002602A (es) 2007-04-25
JP2018150354A (ja) 2018-09-27
JP2015166377A (ja) 2015-09-24
AU2005278323B2 (en) 2011-03-17
NO20071704L (no) 2007-05-31
EP1791545A1 (en) 2007-06-06
JP2013049688A (ja) 2013-03-14
US20140315994A1 (en) 2014-10-23
CA2577284A1 (en) 2006-03-09
IL181332A (en) 2015-09-24
KR20140019006A (ko) 2014-02-13
TW200612901A (en) 2006-05-01

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