JP2007509960A5 - - Google Patents
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- Publication number
- JP2007509960A5 JP2007509960A5 JP2006538253A JP2006538253A JP2007509960A5 JP 2007509960 A5 JP2007509960 A5 JP 2007509960A5 JP 2006538253 A JP2006538253 A JP 2006538253A JP 2006538253 A JP2006538253 A JP 2006538253A JP 2007509960 A5 JP2007509960 A5 JP 2007509960A5
- Authority
- JP
- Japan
- Prior art keywords
- disorders
- pharmaceutical composition
- composition according
- nzojiazepin
- depressive
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 239000008194 pharmaceutical composition Substances 0.000 claims 2
- 206010001488 Aggression Diseases 0.000 claims 1
- 208000019901 Anxiety disease Diseases 0.000 claims 1
- 208000020925 Bipolar disease Diseases 0.000 claims 1
- 206010010904 Convulsion Diseases 0.000 claims 1
- 208000020401 Depressive disease Diseases 0.000 claims 1
- 208000030814 Eating disease Diseases 0.000 claims 1
- 208000019454 Feeding and Eating disease Diseases 0.000 claims 1
- 208000007101 Muscle Cramp Diseases 0.000 claims 1
- 206010049816 Muscle tightness Diseases 0.000 claims 1
- 208000028017 Psychotic disease Diseases 0.000 claims 1
- 208000005392 Spasm Diseases 0.000 claims 1
- 206010047700 Vomiting Diseases 0.000 claims 1
- 230000016571 aggressive behavior Effects 0.000 claims 1
- 208000012761 aggressive behavior Diseases 0.000 claims 1
- 208000010877 cognitive disease Diseases 0.000 claims 1
- 230000003001 depressive effect Effects 0.000 claims 1
- 235000014632 disordered eating Nutrition 0.000 claims 1
- 208000030533 eye disease Diseases 0.000 claims 1
- 230000002401 inhibitory effect Effects 0.000 claims 1
- 230000004770 neurodegeneration Effects 0.000 claims 1
- 230000000626 neurodegenerative effect Effects 0.000 claims 1
- 230000036407 pain Effects 0.000 claims 1
- 208000019116 sleep disease Diseases 0.000 claims 1
- 238000002560 therapeutic procedure Methods 0.000 claims 1
- 230000008673 vomiting Effects 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 description 2
- 238000001727 in vivo Methods 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US51504303P | 2003-10-28 | 2003-10-28 | |
| PCT/US2004/035822 WO2005044818A2 (en) | 2003-10-28 | 2004-10-28 | Imidazo[1,2-a]pyridine anxiolytics |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2007509960A JP2007509960A (ja) | 2007-04-19 |
| JP2007509960A5 true JP2007509960A5 (enExample) | 2007-11-29 |
Family
ID=34572796
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006538253A Withdrawn JP2007509960A (ja) | 2003-10-28 | 2004-10-28 | イミダゾ[1,2−a]ピリジン抗不安薬 |
Country Status (8)
| Country | Link |
|---|---|
| US (3) | US7723324B2 (enExample) |
| EP (1) | EP1682549B1 (enExample) |
| JP (1) | JP2007509960A (enExample) |
| AT (1) | ATE482211T1 (enExample) |
| AU (1) | AU2004287847A1 (enExample) |
| CA (1) | CA2544213A1 (enExample) |
| DE (1) | DE602004029272D1 (enExample) |
| WO (1) | WO2005044818A2 (enExample) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1966201A1 (en) * | 2005-11-28 | 2008-09-10 | Mallinckrodt, Inc. | Improved method of preparation for imidazolepyridines |
| EP1803722A1 (en) * | 2006-01-03 | 2007-07-04 | Ferrer Internacional, S.A. | Imidazo[1,2-a]pyridin-3-yl-acetic acid hydrazides, processes for their preparation and pharmaceutical uses thereof |
| AU2009249186B2 (en) | 2008-05-19 | 2014-05-22 | Sunovion Pharmaceuticals Inc. | Imidazo [1, 2-a] pyridine compounds as GABA-A receptor modulators |
| WO2011041713A2 (en) * | 2009-10-02 | 2011-04-07 | Glaxosmithkline Llc | Piperazinyl antiviral agents |
| PH12012500778A1 (en) | 2009-10-30 | 2012-11-26 | Janssen Pharmaceutica Nv | IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES AND THEIR USE AS PDE10 INHIBITORS |
| AR080754A1 (es) | 2010-03-09 | 2012-05-09 | Janssen Pharmaceutica Nv | Derivados de imidazo (1,2-a) pirazina y su uso como inhibidores de pde10 |
| TR201906779T4 (tr) * | 2011-05-12 | 2019-05-21 | Proteostasis Therapeutics Inc | Proteostaz regülatörleri. |
| JP6115962B2 (ja) | 2011-06-27 | 2017-04-19 | ヤンセン ファーマシューティカ エヌ.ベー. | 1−アリール−4−メチル−[1,2,4]トリアゾロ[4,3−a]キノキサリン誘導体 |
| WO2014001314A1 (en) | 2012-06-26 | 2014-01-03 | Janssen Pharmaceutica Nv | Combinations comprising pde 2 inhibitors such as 1-aryl-4-methyl- [1,2,4] triazolo [4,3-a] quinoxaline compounds and pde 10 inhibitors for use in the treatment of neurological or metabolic disorders |
| AU2013289284B2 (en) | 2012-07-09 | 2017-03-30 | Janssen Pharmaceutica Nv | Inhibitors of phosphodiesterase 10 enzyme |
| ES2689429T3 (es) * | 2012-07-13 | 2018-11-14 | Ucb Biopharma Sprl | Derivados de imidazopiridina como moduladores de actividad de TNF |
| TWI648281B (zh) * | 2013-10-17 | 2019-01-21 | 日商安斯泰來製藥股份有限公司 | 含硫二環式化合物 |
| TW201601632A (zh) | 2013-11-20 | 2016-01-16 | 杜邦股份有限公司 | 1-芳基-3-烷基吡唑殺蟲劑 |
| UA125012C2 (uk) | 2014-07-02 | 2021-12-29 | ЕфЕмСі КОРПОРЕЙШН | Піперидинонові гербіциди |
| US9926316B2 (en) * | 2016-03-03 | 2018-03-27 | The Cleveland Clinic Foundation | Antitumor derivatives for differentiation therapy |
| CN107383005B (zh) * | 2017-09-11 | 2020-03-13 | 华东理工大学 | 6-甲基-2-(4-甲基苯基)咪唑并[1,2-a]吡啶-3-乙酸的制备方法 |
| CN113387946B (zh) * | 2021-05-17 | 2023-08-01 | 衡阳师范学院 | 一种超声辅助多组分合成2-苯基-3-芳胺甲基咪唑并吡啶衍生物的方法 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SU522187A1 (ru) * | 1975-03-12 | 1976-07-25 | Военная Краснознаменная академия химической защиты им.Маршала Советского Союза С.К.Тимошенко | Способ получени 3-ацил-2-алкил (арил)-имидазо (1,2 )пиридинов |
| FR2492382A1 (fr) | 1980-10-22 | 1982-04-23 | Synthelabo | Derives d'imidazo (1,2-a) pyridine, leur preparation et leur application en therapeutique |
| FR2525601A1 (fr) | 1982-04-21 | 1983-10-28 | Synthelabo | Derives d'imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique |
| FR2568880B1 (fr) * | 1984-08-07 | 1986-12-12 | Synthelabo | Derives d'acylaminomethyl-3 imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique |
| EP0226641B1 (en) | 1985-05-25 | 1989-10-18 | Yoshitomi Pharmaceutical Industries, Ltd. | Oxodiazine compounds |
| FR2647451B1 (fr) * | 1989-05-26 | 1994-08-05 | Sanofi Sa | Derives d'imidazo(1,2-a)pyridine, procede de preparation, compositions pharmaceutiques les contenant |
| DE10040016A1 (de) * | 2000-08-16 | 2002-02-28 | Boehringer Ingelheim Pharma | Neue beta-Amyloid Inhibitoren, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
| US6514969B2 (en) * | 2000-08-16 | 2003-02-04 | Boehringer Ingelheim Pharma Kg | β-amyloid inhibitors, processes for preparing them, and their use in pharmaceutical compositions |
| SE0100568D0 (sv) | 2001-02-20 | 2001-02-20 | Astrazeneca Ab | Compounds |
| SE0100567D0 (sv) | 2001-02-20 | 2001-02-20 | Astrazeneca Ab | Compounds |
| CA2450555A1 (en) | 2001-06-25 | 2003-01-03 | Merck & Co., Inc. | (pyrimidyl)(phenyl)substituted fused heteroaryl p38 inhibiting and pkg kinase inhibiting compounds |
| CA2484631A1 (en) | 2002-05-13 | 2003-11-27 | Merck & Co., Inc. | Phenyl substituted imidazopyridines and phenyl substituted benzimidazoles |
-
2004
- 2004-10-28 US US10/595,592 patent/US7723324B2/en not_active Expired - Lifetime
- 2004-10-28 WO PCT/US2004/035822 patent/WO2005044818A2/en not_active Ceased
- 2004-10-28 EP EP04796657A patent/EP1682549B1/en not_active Expired - Lifetime
- 2004-10-28 AU AU2004287847A patent/AU2004287847A1/en not_active Abandoned
- 2004-10-28 DE DE602004029272T patent/DE602004029272D1/de not_active Expired - Lifetime
- 2004-10-28 AT AT04796657T patent/ATE482211T1/de not_active IP Right Cessation
- 2004-10-28 JP JP2006538253A patent/JP2007509960A/ja not_active Withdrawn
- 2004-10-28 US US10/976,331 patent/US7148353B2/en not_active Expired - Lifetime
- 2004-10-28 CA CA002544213A patent/CA2544213A1/en not_active Abandoned
-
2006
- 2006-09-15 US US11/532,402 patent/US7566725B2/en not_active Expired - Lifetime
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