JP2007509960A5 - - Google Patents
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- JP2007509960A5 JP2007509960A5 JP2006538253A JP2006538253A JP2007509960A5 JP 2007509960 A5 JP2007509960 A5 JP 2007509960A5 JP 2006538253 A JP2006538253 A JP 2006538253A JP 2006538253 A JP2006538253 A JP 2006538253A JP 2007509960 A5 JP2007509960 A5 JP 2007509960A5
- Authority
- JP
- Japan
- Prior art keywords
- disorders
- pharmaceutical composition
- composition according
- nzojiazepin
- depressive
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
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- 239000008194 pharmaceutical composition Substances 0.000 claims 2
- 206010001488 Aggression Diseases 0.000 claims 1
- 208000019901 Anxiety disease Diseases 0.000 claims 1
- 208000020925 Bipolar disease Diseases 0.000 claims 1
- 206010010904 Convulsion Diseases 0.000 claims 1
- 208000020401 Depressive disease Diseases 0.000 claims 1
- 208000030814 Eating disease Diseases 0.000 claims 1
- 208000019454 Feeding and Eating disease Diseases 0.000 claims 1
- 208000007101 Muscle Cramp Diseases 0.000 claims 1
- 206010049816 Muscle tightness Diseases 0.000 claims 1
- 208000028017 Psychotic disease Diseases 0.000 claims 1
- 208000005392 Spasm Diseases 0.000 claims 1
- 206010047700 Vomiting Diseases 0.000 claims 1
- 230000016571 aggressive behavior Effects 0.000 claims 1
- 208000012761 aggressive behavior Diseases 0.000 claims 1
- 208000010877 cognitive disease Diseases 0.000 claims 1
- 230000003001 depressive effect Effects 0.000 claims 1
- 235000014632 disordered eating Nutrition 0.000 claims 1
- 208000030533 eye disease Diseases 0.000 claims 1
- 230000002401 inhibitory effect Effects 0.000 claims 1
- 230000004770 neurodegeneration Effects 0.000 claims 1
- 230000000626 neurodegenerative effect Effects 0.000 claims 1
- 230000036407 pain Effects 0.000 claims 1
- 208000019116 sleep disease Diseases 0.000 claims 1
- 238000002560 therapeutic procedure Methods 0.000 claims 1
- 230000008673 vomiting Effects 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 description 2
- 238000001727 in vivo Methods 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US51504303P | 2003-10-28 | 2003-10-28 | |
| PCT/US2004/035822 WO2005044818A2 (en) | 2003-10-28 | 2004-10-28 | Imidazo[1,2-a]pyridine anxiolytics |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2007509960A JP2007509960A (ja) | 2007-04-19 |
| JP2007509960A5 true JP2007509960A5 (enExample) | 2007-11-29 |
Family
ID=34572796
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006538253A Withdrawn JP2007509960A (ja) | 2003-10-28 | 2004-10-28 | イミダゾ[1,2−a]ピリジン抗不安薬 |
Country Status (8)
| Country | Link |
|---|---|
| US (3) | US7148353B2 (enExample) |
| EP (1) | EP1682549B1 (enExample) |
| JP (1) | JP2007509960A (enExample) |
| AT (1) | ATE482211T1 (enExample) |
| AU (1) | AU2004287847A1 (enExample) |
| CA (1) | CA2544213A1 (enExample) |
| DE (1) | DE602004029272D1 (enExample) |
| WO (1) | WO2005044818A2 (enExample) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2006327217A1 (en) * | 2005-11-28 | 2007-06-28 | Mallinckrodt Inc. | Improved method of preparation for Imidazolepyridines |
| EP1803722A1 (en) * | 2006-01-03 | 2007-07-04 | Ferrer Internacional, S.A. | Imidazo[1,2-a]pyridin-3-yl-acetic acid hydrazides, processes for their preparation and pharmaceutical uses thereof |
| WO2009143156A2 (en) * | 2008-05-19 | 2009-11-26 | Sepracor Inc. | IMIDAZO[1,2-a]PYRIDINE COMPOUNDS |
| WO2011041713A2 (en) * | 2009-10-02 | 2011-04-07 | Glaxosmithkline Llc | Piperazinyl antiviral agents |
| EP2493889B1 (en) | 2009-10-30 | 2017-09-06 | Janssen Pharmaceutica, N.V. | IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES AND THEIR USE AS PDE10 INHIBITORS |
| AR080754A1 (es) | 2010-03-09 | 2012-05-09 | Janssen Pharmaceutica Nv | Derivados de imidazo (1,2-a) pirazina y su uso como inhibidores de pde10 |
| US9556166B2 (en) * | 2011-05-12 | 2017-01-31 | Proteostasis Therapeutics, Inc. | Proteostasis regulators |
| MX344600B (es) | 2011-06-27 | 2016-12-20 | Janssen Pharmaceutica Nv | Derivados de 1-aril-4-metil-[1,2,4]triazolo[4,3-a]quinoxalina. |
| HK1206250A1 (en) | 2012-06-26 | 2016-01-08 | Janssen Pharmaceutica Nv | Combinations comprising pde 2 inhibitors such as 1-aryl-4-methyl-[1,2,4] triazolo [4,3-a] quinoxaline compounds and ped 10 inhibitors for use in the treatment of neurological or metabolic disorders |
| CN104411314B (zh) | 2012-07-09 | 2017-10-20 | 詹森药业有限公司 | 磷酸二酯酶10的抑制剂 |
| BR112015000675B1 (pt) * | 2012-07-13 | 2022-07-12 | UCB Biopharma SRL | Derivados de imidazopiridina como moduladores da atividade de tnf |
| TWI648281B (zh) * | 2013-10-17 | 2019-01-21 | 日商安斯泰來製藥股份有限公司 | 含硫二環式化合物 |
| TW201601632A (zh) | 2013-11-20 | 2016-01-16 | 杜邦股份有限公司 | 1-芳基-3-烷基吡唑殺蟲劑 |
| AU2015284280C1 (en) | 2014-07-02 | 2020-02-13 | Fmc Corporation | Piperidinone herbicides |
| US9926316B2 (en) * | 2016-03-03 | 2018-03-27 | The Cleveland Clinic Foundation | Antitumor derivatives for differentiation therapy |
| CN107383005B (zh) * | 2017-09-11 | 2020-03-13 | 华东理工大学 | 6-甲基-2-(4-甲基苯基)咪唑并[1,2-a]吡啶-3-乙酸的制备方法 |
| CN113387946B (zh) * | 2021-05-17 | 2023-08-01 | 衡阳师范学院 | 一种超声辅助多组分合成2-苯基-3-芳胺甲基咪唑并吡啶衍生物的方法 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SU522187A1 (ru) * | 1975-03-12 | 1976-07-25 | Военная Краснознаменная академия химической защиты им.Маршала Советского Союза С.К.Тимошенко | Способ получени 3-ацил-2-алкил (арил)-имидазо (1,2 )пиридинов |
| FR2492382A1 (fr) * | 1980-10-22 | 1982-04-23 | Synthelabo | Derives d'imidazo (1,2-a) pyridine, leur preparation et leur application en therapeutique |
| FR2525601A1 (fr) | 1982-04-21 | 1983-10-28 | Synthelabo | Derives d'imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique |
| FR2568880B1 (fr) | 1984-08-07 | 1986-12-12 | Synthelabo | Derives d'acylaminomethyl-3 imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique |
| WO1986007059A2 (en) | 1985-05-25 | 1986-12-04 | Yoshitomi Pharmaceutical Industries, Ltd. | Oxodiazine compounds |
| FR2647451B1 (fr) | 1989-05-26 | 1994-08-05 | Sanofi Sa | Derives d'imidazo(1,2-a)pyridine, procede de preparation, compositions pharmaceutiques les contenant |
| US6514969B2 (en) * | 2000-08-16 | 2003-02-04 | Boehringer Ingelheim Pharma Kg | β-amyloid inhibitors, processes for preparing them, and their use in pharmaceutical compositions |
| DE10040016A1 (de) * | 2000-08-16 | 2002-02-28 | Boehringer Ingelheim Pharma | Neue beta-Amyloid Inhibitoren, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
| SE0100568D0 (sv) | 2001-02-20 | 2001-02-20 | Astrazeneca Ab | Compounds |
| SE0100567D0 (sv) | 2001-02-20 | 2001-02-20 | Astrazeneca Ab | Compounds |
| WO2003000682A1 (en) | 2001-06-25 | 2003-01-03 | Merck & Co., Inc. | (pyrimidyl)(phenyl)substituted fused heteroaryl p38 inhibiting and pkg kinase inhibiting compounds |
| CA2484631A1 (en) | 2002-05-13 | 2003-11-27 | Merck & Co., Inc. | Phenyl substituted imidazopyridines and phenyl substituted benzimidazoles |
-
2004
- 2004-10-28 WO PCT/US2004/035822 patent/WO2005044818A2/en not_active Ceased
- 2004-10-28 AU AU2004287847A patent/AU2004287847A1/en not_active Abandoned
- 2004-10-28 CA CA002544213A patent/CA2544213A1/en not_active Abandoned
- 2004-10-28 AT AT04796657T patent/ATE482211T1/de not_active IP Right Cessation
- 2004-10-28 EP EP04796657A patent/EP1682549B1/en not_active Expired - Lifetime
- 2004-10-28 DE DE602004029272T patent/DE602004029272D1/de not_active Expired - Lifetime
- 2004-10-28 JP JP2006538253A patent/JP2007509960A/ja not_active Withdrawn
- 2004-10-28 US US10/976,331 patent/US7148353B2/en not_active Expired - Lifetime
- 2004-10-28 US US10/595,592 patent/US7723324B2/en active Active
-
2006
- 2006-09-15 US US11/532,402 patent/US7566725B2/en not_active Expired - Lifetime
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