JP2006522834A5 - - Google Patents

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Publication number
JP2006522834A5
JP2006522834A5 JP2006510082A JP2006510082A JP2006522834A5 JP 2006522834 A5 JP2006522834 A5 JP 2006522834A5 JP 2006510082 A JP2006510082 A JP 2006510082A JP 2006510082 A JP2006510082 A JP 2006510082A JP 2006522834 A5 JP2006522834 A5 JP 2006522834A5
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JP
Japan
Prior art keywords
group
composition
disorder
pain
aryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2006510082A
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English (en)
Japanese (ja)
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JP2006522834A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2004/011668 external-priority patent/WO2004091633A1/en
Publication of JP2006522834A publication Critical patent/JP2006522834A/ja
Publication of JP2006522834A5 publication Critical patent/JP2006522834A5/ja
Pending legal-status Critical Current

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JP2006510082A 2003-04-09 2004-04-07 [2−(8,9−ジオキソ−2,6−ジアザビシクロ[5.2.0]ノナ−1(7)−エン−2−イル)アルキル]ホスホン酸および誘導体の鼻腔内投与用医薬組成物およびその使用法 Pending JP2006522834A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US46157103P 2003-04-09 2003-04-09
PCT/US2004/011668 WO2004091633A1 (en) 2003-04-09 2004-04-07 Pharmaceutical compositions for intranasal administration of [2-(8,9-dioxo-2,6-diazabicyclo[5.2.o]non-1 (7)-en-2-yl)alkyl] phosphonic acid and derivatives and methods of use thereof

Publications (2)

Publication Number Publication Date
JP2006522834A JP2006522834A (ja) 2006-10-05
JP2006522834A5 true JP2006522834A5 (https=) 2007-06-14

Family

ID=33299836

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006510082A Pending JP2006522834A (ja) 2003-04-09 2004-04-07 [2−(8,9−ジオキソ−2,6−ジアザビシクロ[5.2.0]ノナ−1(7)−エン−2−イル)アルキル]ホスホン酸および誘導体の鼻腔内投与用医薬組成物およびその使用法

Country Status (12)

Country Link
US (1) US20050004079A1 (https=)
EP (1) EP1622625A1 (https=)
JP (1) JP2006522834A (https=)
CN (1) CN1802161A (https=)
AR (1) AR044014A1 (https=)
AU (1) AU2004229567A1 (https=)
BR (1) BRPI0409088A (https=)
CA (1) CA2521394A1 (https=)
CL (1) CL2004000765A1 (https=)
MX (1) MXPA05010763A (https=)
TW (1) TW200503732A (https=)
WO (1) WO2004091633A1 (https=)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2521313A1 (en) * 2003-04-09 2004-10-28 Wyeth Derivatives of 2-(8,9-dioxo-2,6-diazabicyclo(5.2.o)non-1(7)-3n-2-yl)-al kyl phosphonic acid and their use as n-methyl-d-aspartate (nmda) recetor antagonists
US20050142192A1 (en) * 2003-10-15 2005-06-30 Wyeth Oral administration of [2-(8,9-dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl)alkyl] phosphonic acid and derivatives
GT200400213A (es) * 2003-10-22 2007-09-05 Metodos para la preparacion del acido {2-[(8,9)-dioxo-2,6-diaza-biciclo[5.2.0]-non-1(7)-en-2-il]etil} fosfonico y esteres del mismo
EP2195031A1 (en) * 2007-08-27 2010-06-16 Wyeth a Corporation of the State of Delaware Compositions and methods employing nmda antagonists for achieving an anesthetic-sparing effect
US8784872B2 (en) 2007-11-19 2014-07-22 Comgenrx, Inc. Formulation for decreasing tobacco, alcohol, drug or food consumption
US20090130048A1 (en) * 2007-11-19 2009-05-21 Oronsky Bryan Todd Topical Composition for Treating Pain
WO2009158667A2 (en) * 2008-06-27 2009-12-30 Comgenrx, Inc. Povidone compositions for wound healing
US9757529B2 (en) 2012-12-20 2017-09-12 Otitopic Inc. Dry powder inhaler and methods of use
US9757395B2 (en) 2012-12-20 2017-09-12 Otitopic Inc. Dry powder inhaler and methods of use
HK1218720A1 (zh) 2013-04-30 2017-03-10 欧缇托匹克公司 干粉制剂及使用方法
US10786456B2 (en) 2017-09-22 2020-09-29 Otitopic Inc. Inhaled aspirin and magnesium to treat inflammation
KR102681843B1 (ko) 2017-09-22 2024-07-05 벡추라 인코포레이티드 스테아르산마그네슘을 갖는 건조 분말 조성물

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5624898A (en) * 1989-12-05 1997-04-29 Ramsey Foundation Method for administering neurologic agents to the brain
US5168103A (en) * 1991-01-22 1992-12-01 American Home Products Corporation [[2-(amino-3,4-dioxo-1-cyclobuten-1-yl) amino]alkyl]-acid derivatives
US5124319A (en) * 1991-10-11 1992-06-23 American Home Products Corporation Benzimidazole phosphono-amino acids
TW427904B (en) * 1995-12-07 2001-04-01 American Home Prod Neuroprotective agents
US5990307A (en) * 1997-08-01 1999-11-23 American Home Products Corporation Process for the preparation of [2-((8.9)-Dioxo-2,6-Diazabicyclo [5.2.0]-Non-1(7)-en-2yl) Ethyl]Phosphonic acid
US6225343B1 (en) * 1999-06-16 2001-05-01 Nastech Pharmaceutical Company, Inc. Compositions and methods comprising morphine gluconate
UA78529C2 (en) * 2001-10-10 2007-04-10 Wyeth Corp Derivatives of [[2-(amino-3,4-dioxo-1-cyclobutene-1-yl)amino]alkyl] acid for treating pain
US20040082543A1 (en) * 2002-10-29 2004-04-29 Pharmacia Corporation Compositions of cyclooxygenase-2 selective inhibitors and NMDA receptor antagonists for the treatment or prevention of neuropathic pain
US20050142192A1 (en) * 2003-10-15 2005-06-30 Wyeth Oral administration of [2-(8,9-dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl)alkyl] phosphonic acid and derivatives
GT200400213A (es) * 2003-10-22 2007-09-05 Metodos para la preparacion del acido {2-[(8,9)-dioxo-2,6-diaza-biciclo[5.2.0]-non-1(7)-en-2-il]etil} fosfonico y esteres del mismo

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