JP2006515841A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2006515841A5 JP2006515841A5 JP2004559734A JP2004559734A JP2006515841A5 JP 2006515841 A5 JP2006515841 A5 JP 2006515841A5 JP 2004559734 A JP2004559734 A JP 2004559734A JP 2004559734 A JP2004559734 A JP 2004559734A JP 2006515841 A5 JP2006515841 A5 JP 2006515841A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- atom
- chlorine
- fluorine
- represented
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 229910052801 chlorine Inorganic materials 0.000 claims 77
- 229910052731 fluorine Inorganic materials 0.000 claims 75
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 62
- 125000004435 hydrogen atom Chemical group [H]* 0.000 claims 61
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical group [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 claims 60
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims 58
- 125000005843 halogen group Chemical group 0.000 claims 49
- 125000001153 fluoro group Chemical group F* 0.000 claims 47
- -1 - haloalkyl group Chemical group 0.000 claims 46
- 125000001309 chloro group Chemical group Cl* 0.000 claims 46
- 239000000460 chlorine Substances 0.000 claims 31
- 239000011737 fluorine Substances 0.000 claims 29
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 claims 28
- YCKRFDGAMUMZLT-UHFFFAOYSA-N Fluorine atom Chemical compound [F] YCKRFDGAMUMZLT-UHFFFAOYSA-N 0.000 claims 28
- 125000004093 cyano group Chemical group *C#N 0.000 claims 28
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 claims 27
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 claims 27
- 125000001028 difluoromethyl group Chemical group [H]C(F)(F)* 0.000 claims 23
- 125000001246 bromo group Chemical group Br* 0.000 claims 21
- 125000003866 trichloromethyl group Chemical group ClC(Cl)(Cl)* 0.000 claims 21
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims 16
- ZCYVEMRRCGMTRW-UHFFFAOYSA-N 7553-56-2 Chemical group [I] ZCYVEMRRCGMTRW-UHFFFAOYSA-N 0.000 claims 16
- 229910052740 iodine Inorganic materials 0.000 claims 16
- 125000003277 amino group Chemical group 0.000 claims 15
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims 10
- GTKIGDZXPDCIKR-UHFFFAOYSA-N 2-phenylbenzamide Chemical compound NC(=O)C1=CC=CC=C1C1=CC=CC=C1 GTKIGDZXPDCIKR-UHFFFAOYSA-N 0.000 claims 9
- 125000001301 ethoxy group Chemical group [H]C([H])([H])C([H])([H])O* 0.000 claims 9
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims 9
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims 9
- 125000002816 methylsulfanyl group Chemical group [H]C([H])([H])S[*] 0.000 claims 9
- 125000004705 ethylthio group Chemical group C(C)S* 0.000 claims 8
- 125000001188 haloalkyl group Chemical group 0.000 claims 8
- 239000002253 acid Substances 0.000 claims 7
- 125000000217 alkyl group Chemical group 0.000 claims 7
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 7
- 239000011230 binding agent Substances 0.000 claims 6
- 239000003085 diluting agent Substances 0.000 claims 6
- 125000005034 trifluormethylthio group Chemical group FC(S*)(F)F 0.000 claims 6
- 125000000876 trifluoromethoxy group Chemical group FC(F)(F)O* 0.000 claims 6
- 125000004786 difluoromethoxy group Chemical group [H]C(F)(F)O* 0.000 claims 5
- 244000005700 microbiome Species 0.000 claims 5
- 125000000999 tert-butyl group Chemical group [H]C([H])([H])C(*)(C([H])([H])[H])C([H])([H])[H] 0.000 claims 5
- 125000004784 trichloromethoxy group Chemical group ClC(O*)(Cl)Cl 0.000 claims 5
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims 4
- WGLLSSPDPJPLOR-UHFFFAOYSA-N 2,3-dimethylbut-2-ene Chemical group CC(C)=C(C)C WGLLSSPDPJPLOR-UHFFFAOYSA-N 0.000 claims 4
- KZBUYRJDOAKODT-UHFFFAOYSA-N Chlorine Chemical compound ClCl KZBUYRJDOAKODT-UHFFFAOYSA-N 0.000 claims 4
- 239000003054 catalyst Substances 0.000 claims 4
- 125000004995 haloalkylthio group Chemical group 0.000 claims 4
- 125000004029 hydroxymethyl group Chemical group [H]OC([H])([H])* 0.000 claims 4
- 125000000959 isobutyl group Chemical group [H]C([H])([H])C([H])(C([H])([H])[H])C([H])([H])* 0.000 claims 4
- 125000004108 n-butyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])C([H])([H])* 0.000 claims 4
- 125000004123 n-propyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])* 0.000 claims 4
- 125000002914 sec-butyl group Chemical group [H]C([H])([H])C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims 4
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 claims 3
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims 3
- 150000003857 carboxamides Chemical class 0.000 claims 3
- 125000001559 cyclopropyl group Chemical group [H]C1([H])C([H])([H])C1([H])* 0.000 claims 3
- PXBRQCKWGAHEHS-UHFFFAOYSA-N dichlorodifluoromethane Chemical compound FC(F)(Cl)Cl PXBRQCKWGAHEHS-UHFFFAOYSA-N 0.000 claims 3
- 125000004438 haloalkoxy group Chemical group 0.000 claims 3
- 238000004519 manufacturing process Methods 0.000 claims 3
- 125000004170 methylsulfonyl group Chemical group [H]C([H])([H])S(*)(=O)=O 0.000 claims 3
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 3
- 229910052717 sulfur Inorganic materials 0.000 claims 3
- 239000011593 sulfur Substances 0.000 claims 3
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 claims 2
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims 2
- KDLHZDBZIXYQEI-UHFFFAOYSA-N Palladium Chemical compound [Pd] KDLHZDBZIXYQEI-UHFFFAOYSA-N 0.000 claims 2
- 150000001642 boronic acid derivatives Chemical class 0.000 claims 2
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Substances BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 claims 2
- 229910052794 bromium Inorganic materials 0.000 claims 2
- 239000004067 bulking agent Substances 0.000 claims 2
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 claims 2
- 125000002147 dimethylamino group Chemical group [H]C([H])([H])N(*)C([H])([H])[H] 0.000 claims 2
- 125000000250 methylamino group Chemical group [H]N(*)C([H])([H])[H] 0.000 claims 2
- BASFCYQUMIYNBI-UHFFFAOYSA-N platinum Chemical compound [Pt] BASFCYQUMIYNBI-UHFFFAOYSA-N 0.000 claims 2
- 239000004094 surface-active agent Substances 0.000 claims 2
- 125000006583 (C1-C3) haloalkyl group Chemical group 0.000 claims 1
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims 1
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims 1
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 claims 1
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims 1
- 125000004209 (C1-C8) alkyl group Chemical group 0.000 claims 1
- YFTHTJAPODJVSL-UHFFFAOYSA-N 2-(1-benzothiophen-5-yl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane Chemical compound O1C(C)(C)C(C)(C)OB1C1=CC=C(SC=C2)C2=C1 YFTHTJAPODJVSL-UHFFFAOYSA-N 0.000 claims 1
- 125000004974 2-butenyl group Chemical group C(C=CC)* 0.000 claims 1
- 125000000069 2-butynyl group Chemical group [H]C([H])([H])C#CC([H])([H])* 0.000 claims 1
- 125000003903 2-propenyl group Chemical group [H]C([*])([H])C([H])=C([H])[H] 0.000 claims 1
- 125000001494 2-propynyl group Chemical group [H]C#CC([H])([H])* 0.000 claims 1
- 125000000474 3-butynyl group Chemical group [H]C#CC([H])([H])C([H])([H])* 0.000 claims 1
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims 1
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 claims 1
- 125000004448 alkyl carbonyl group Chemical group 0.000 claims 1
- 125000004390 alkyl sulfonyl group Chemical group 0.000 claims 1
- 125000004414 alkyl thio group Chemical group 0.000 claims 1
- 125000000304 alkynyl group Chemical group 0.000 claims 1
- 125000004397 aminosulfonyl group Chemical group NS(=O)(=O)* 0.000 claims 1
- 125000002490 anilino group Chemical class [H]N(*)C1=C([H])C([H])=C([H])C([H])=C1[H] 0.000 claims 1
- 125000004429 atom Chemical group 0.000 claims 1
- 125000003236 benzoyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C(*)=O 0.000 claims 1
- 125000006268 biphenyl-3-yl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C1=C([H])C(*)=C([H])C([H])=C1[H] 0.000 claims 1
- 150000001732 carboxylic acid derivatives Chemical class 0.000 claims 1
- 125000000113 cyclohexyl group Chemical group [H]C1([H])C([H])([H])C([H])([H])C([H])(*)C([H])([H])C1([H])[H] 0.000 claims 1
- 125000004210 cyclohexylmethyl group Chemical group [H]C([H])(*)C1([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C1([H])[H] 0.000 claims 1
- 125000001511 cyclopentyl group Chemical group [H]C1([H])C([H])([H])C([H])([H])C([H])(*)C1([H])[H] 0.000 claims 1
- 125000004851 cyclopentylmethyl group Chemical group C1(CCCC1)C* 0.000 claims 1
- 125000004186 cyclopropylmethyl group Chemical group [H]C([H])(*)C1([H])C([H])([H])C1([H])[H] 0.000 claims 1
- 125000006263 dimethyl aminosulfonyl group Chemical group [H]C([H])([H])N(C([H])([H])[H])S(*)(=O)=O 0.000 claims 1
- 125000005745 ethoxymethyl group Chemical group [H]C([H])([H])C([H])([H])OC([H])([H])* 0.000 claims 1
- 125000004216 fluoromethyl group Chemical group [H]C([H])(F)* 0.000 claims 1
- 229910052736 halogen Inorganic materials 0.000 claims 1
- 229910052739 hydrogen Inorganic materials 0.000 claims 1
- 239000001257 hydrogen Substances 0.000 claims 1
- 125000005394 methallyl group Chemical group 0.000 claims 1
- 238000000034 method Methods 0.000 claims 1
- 125000004184 methoxymethyl group Chemical group [H]C([H])([H])OC([H])([H])* 0.000 claims 1
- 125000006216 methylsulfinyl group Chemical group [H]C([H])([H])S(*)=O 0.000 claims 1
- 229910052763 palladium Inorganic materials 0.000 claims 1
- 125000003170 phenylsulfonyl group Chemical group C1(=CC=CC=C1)S(=O)(=O)* 0.000 claims 1
- 229910052697 platinum Inorganic materials 0.000 claims 1
- 125000001844 prenyl group Chemical group [H]C([*])([H])C([H])=C(C([H])([H])[H])C([H])([H])[H] 0.000 claims 1
- 0 CC(C1*)OC(C)=C1*#C Chemical compound CC(C1*)OC(C)=C1*#C 0.000 description 10
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10258314A DE10258314A1 (de) | 2002-12-13 | 2002-12-13 | Biphenyloximether |
| PCT/EP2003/013498 WO2004054982A1 (de) | 2002-12-13 | 2003-12-01 | Biphenylcarboxamide |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2006515841A JP2006515841A (ja) | 2006-06-08 |
| JP2006515841A5 true JP2006515841A5 (enExample) | 2010-07-22 |
| JP4555085B2 JP4555085B2 (ja) | 2010-09-29 |
Family
ID=32336291
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004559734A Expired - Fee Related JP4555085B2 (ja) | 2002-12-13 | 2003-12-01 | ビフェニルカルボキサミド |
Country Status (8)
| Country | Link |
|---|---|
| US (2) | US7728019B2 (enExample) |
| EP (1) | EP1572663B1 (enExample) |
| JP (1) | JP4555085B2 (enExample) |
| CN (1) | CN100391947C (enExample) |
| AU (1) | AU2003298156A1 (enExample) |
| BR (1) | BR0317290B1 (enExample) |
| DE (1) | DE10258314A1 (enExample) |
| WO (1) | WO2004054982A1 (enExample) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10354607A1 (de) * | 2003-11-21 | 2005-06-16 | Bayer Cropscience Ag | Siylierte Carboxamide |
| DE102004005786A1 (de) * | 2004-02-06 | 2005-08-25 | Bayer Cropscience Ag | Haloalkylcarboxamide |
| DE102004005785A1 (de) * | 2004-02-06 | 2005-08-25 | Bayer Cropscience Ag | 2-Halogenfuryl/thienyl-3-carboxamide |
| TWI372752B (en) * | 2005-12-22 | 2012-09-21 | Nihon Nohyaku Co Ltd | Pyrazinecarboxamide derivatives and plant disease controlling agents containing the same |
| RU2425036C2 (ru) * | 2005-12-22 | 2011-07-27 | Нихон Нохияку Ко., Лтд. | Производные пиразинкарбоксамида и средства, содержащие их, для подавления болезней растений |
| ZA200804816B (en) * | 2005-12-22 | 2009-10-28 | Nihon Nohyaku Co Ltd | Pyrazinecarboxamide derivatives and plant disease controlling agents containing the same |
| EP2662363A1 (en) * | 2012-05-09 | 2013-11-13 | Bayer CropScience AG | 5-Halogenopyrazole biphenylcarboxamides |
| AR105929A1 (es) | 2015-09-07 | 2017-11-22 | Bayer Cropscience Ag | Derivados de 2-difluorometil-nicotin(tio)carboxanilida sustituidos y su uso como fungicidas |
| KR20200040348A (ko) | 2018-10-08 | 2020-04-20 | 한국화학연구원 | 티오펜 카르복사미드계 유도체 및 이를 함유하는 식물 병해 방제제 |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5045554A (en) * | 1988-11-29 | 1991-09-03 | Monsanto Company | Substituted thiazoles and their use as fungicides |
| AU6049590A (en) | 1989-07-25 | 1991-02-22 | Monsanto Company | Substituted carboxanilidothiazoles and their use as fungicides |
| IN172842B (enExample) * | 1990-05-17 | 1993-12-11 | Boots Pharmaceuticals Limited | |
| CA2081935C (en) * | 1991-11-22 | 2004-05-25 | Karl Eicken | Anilide derivatives and their use for combating botrytis |
| US5223526A (en) * | 1991-12-06 | 1993-06-29 | Monsanto Company | Pyrazole carboxanilide fungicides and use |
| ATE172597T1 (de) * | 1992-07-15 | 1998-11-15 | Basf Ag | Substituierte oximether und ihre verwendung zur bekämpfung von schädlingen |
| DE4231517A1 (de) * | 1992-09-21 | 1994-03-24 | Basf Ag | Carbonsäureanilide, Verfahren zu ihrer Herstellung und sie enthaltende Mittel zur Bekämpfung von Schadpilzen |
| DE4231519A1 (de) * | 1992-09-21 | 1994-03-24 | Basf Ag | Cyclohex(en)ylcarbonsäureamide, Verfahren zu ihrer Herstellung und sie enthaltende Mittel zur Bekämpfung von Schadpilzen |
| GB9510459D0 (en) * | 1995-05-24 | 1995-07-19 | Zeneca Ltd | Bicyclic amines |
| IL130058A0 (en) * | 1996-11-26 | 2000-02-29 | Zeneca Ltd | 8-Azabicyclo(3.2.1)octane-8-azabicyclo(3.2.1)oct-6-ene-9-azabicyclo(3.3.1)nonane-9-aza-3-oxabicyclo (3.3.1)nonane- and 9-aza-3-thiabicyclo(3.3.1)nonane derivatives their preparation and their use as insecticides |
| GB9624611D0 (en) * | 1996-11-26 | 1997-01-15 | Zeneca Ltd | Bicyclic amine compounds |
| DE19735224A1 (de) * | 1997-08-15 | 1999-02-18 | Basf Ag | Biphenylamide |
| DE19840322A1 (de) * | 1998-09-04 | 2000-03-09 | Bayer Ag | Pyrazol-carboxanilide |
| WO2002008197A1 (de) * | 2000-07-24 | 2002-01-31 | Bayer Cropscience Ag | Biphenylcarboxamide |
| US6992098B2 (en) | 2000-07-24 | 2006-01-31 | Bayer Cropscience Ag | Pyrazolyl biphenyl carboxamides and the use thereof for controlling undesired microorganisms |
| DK1599460T3 (da) * | 2003-02-14 | 2008-03-25 | Bayer Cropscience Ag | Oxathiincarboxamider |
-
2002
- 2002-12-13 DE DE10258314A patent/DE10258314A1/de not_active Withdrawn
-
2003
- 2003-12-01 EP EP03795860A patent/EP1572663B1/de not_active Expired - Lifetime
- 2003-12-01 CN CNB2003801095719A patent/CN100391947C/zh not_active Expired - Fee Related
- 2003-12-01 AU AU2003298156A patent/AU2003298156A1/en not_active Abandoned
- 2003-12-01 US US10/538,242 patent/US7728019B2/en not_active Expired - Fee Related
- 2003-12-01 WO PCT/EP2003/013498 patent/WO2004054982A1/de not_active Ceased
- 2003-12-01 BR BRPI0317290-2A patent/BR0317290B1/pt not_active IP Right Cessation
- 2003-12-01 JP JP2004559734A patent/JP4555085B2/ja not_active Expired - Fee Related
-
2010
- 2010-04-30 US US12/771,285 patent/US20100216849A1/en not_active Abandoned
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2005530694A5 (enExample) | ||
| JP2006515841A5 (enExample) | ||
| JP4448327B2 (ja) | 新規置換１ｈ−ジヒドロピラゾール、それらの製造および使用 | |
| JP2010536767A5 (enExample) | ||
| JP2007508305A5 (enExample) | ||
| RU2010109881A (ru) | Способ получения производных 5-галогеналкил-4,5-дигидроизоксазола | |
| CA2587528A1 (en) | Method for preparing n-phenylpyrazole-1-carboxamides | |
| BRPI0608732A2 (pt) | composto ou um sal, hidrato, solvato, complexo ou pró-droga farmaceuticamente aceitável do mesmo, sal de um composto, processo para a preparação de um composto, uso de um composto, composição farmacêutica, e, produto | |
| JP2012519693A5 (enExample) | ||
| JP2008523069A5 (enExample) | ||
| JP2005531549A5 (enExample) | ||
| PT91620B (pt) | Processo para a preparacao de compostos antifungicos a base de amidas com grupo fenilo e de composicoes fungicidas que os contem | |
| CN104245665B (zh) | 烷基化芳香族酰胺衍生物的制造方法 | |
| BR112019023012A2 (pt) | 4-difluorometil benzoil amidas com ação herbicida | |
| AR063048A1 (es) | Derivados de n-cicloaquil-carboxamida, tiocarboxamida y carboximidamida n-sustituida fungicidas | |
| CN1107672C (zh) | 用于制备吡唑衍生物的中间体 | |
| TW201215594A (en) | Intermediate compound for the preparation of a 2-pyridylethylcarboxamide derivative | |
| JP2008540658A5 (enExample) | ||
| JP2012176950A5 (enExample) | ||
| JP2012149082A5 (enExample) | ||
| CN102858735B (zh) | N-甲氧羰基-n-甲氧基-(2-氯甲基)苯胺、其制备及其作为制备2-(吡唑-3＇-基氧基亚甲基)酰替苯胺的前体的用途 | |
| CN101166728B (zh) | 制备烷基n-酰基苯胺的方法 | |
| JP2004504383A5 (enExample) | ||
| CN103420884B (zh) | 具有光学活性和几何异构的双酰胺衍生物与制备及应用 | |
| JP2007502312A5 (enExample) |