JP2006506369A - メチレン架橋選択的アンドロゲン受容体調節剤及びその使用方法 - Google Patents
メチレン架橋選択的アンドロゲン受容体調節剤及びその使用方法 Download PDFInfo
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- JP2006506369A JP2006506369A JP2004544890A JP2004544890A JP2006506369A JP 2006506369 A JP2006506369 A JP 2006506369A JP 2004544890 A JP2004544890 A JP 2004544890A JP 2004544890 A JP2004544890 A JP 2004544890A JP 2006506369 A JP2006506369 A JP 2006506369A
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- C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
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- C07C235/38—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring
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- C07C255/00—Carboxylic acid nitriles
- C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
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- C07C255/60—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton at least one of the singly-bound nitrogen atoms being acylated
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- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| US41816602P | 2002-10-15 | 2002-10-15 | |
| PCT/US2003/032511 WO2004035738A2 (en) | 2002-10-15 | 2003-10-14 | Methylene-bridged selective androgen receptor modulators and methods of use thereof |
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| JP2006506369A true JP2006506369A (ja) | 2006-02-23 |
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| US (2) | US7253210B2 (cg-RX-API-DMAC7.html) |
| EP (1) | EP1562594A4 (cg-RX-API-DMAC7.html) |
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| TW (1) | TW200503711A (cg-RX-API-DMAC7.html) |
| WO (1) | WO2004035738A2 (cg-RX-API-DMAC7.html) |
Cited By (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2010539181A (ja) * | 2007-09-11 | 2010-12-16 | ユニバーシティ オブ テネシー リサーチ ファウンデーション | 選択的アンドロゲン受容体調節因子の固体形態 |
| JP2011503130A (ja) * | 2007-11-13 | 2011-01-27 | プロシマ ゲーエムベーハー | 治療上の使用のためのｃ−１９ステロイド |
| JP2014532686A (ja) * | 2011-11-04 | 2014-12-08 | ガルデルマ・リサーチ・アンド・デヴェロップメント | Ｎ−（ピリド−４−イル）アミドおよびｎ−（ピリミジン−４−イル）アミド、ならびにそれらの医薬的および美容的使用関連出願 |
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| JP2023514455A (ja) * | 2020-02-25 | 2023-04-05 | ユニバーシティ オブ テネシー リサーチ ファウンデーション | 選択的アンドロゲン受容体共有結合性アンタゴニスト（ｓａｒｃａ）およびその使用方法 |
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| JP2010539181A (ja) * | 2007-09-11 | 2010-12-16 | ユニバーシティ オブ テネシー リサーチ ファウンデーション | 選択的アンドロゲン受容体調節因子の固体形態 |
| JP2012067118A (ja) * | 2007-09-11 | 2012-04-05 | Univ Of Tennessee Research Foundation | 選択的アンドロゲン受容体調節因子の固体形態 |
| JP2014133744A (ja) * | 2007-09-11 | 2014-07-24 | Gtx Inc | 選択的アンドロゲン受容体調節因子の固体形態 |
| JP2011503130A (ja) * | 2007-11-13 | 2011-01-27 | プロシマ ゲーエムベーハー | 治療上の使用のためのｃ−１９ステロイド |
| JP2014532686A (ja) * | 2011-11-04 | 2014-12-08 | ガルデルマ・リサーチ・アンド・デヴェロップメント | Ｎ−（ピリド−４−イル）アミドおよびｎ−（ピリミジン−４−イル）アミド、ならびにそれらの医薬的および美容的使用関連出願 |
| JP2018513182A (ja) * | 2015-04-21 | 2018-05-24 | ジーティーエックス・インコーポレイテッド | 選択的アンドロゲン受容体分解剤（ｓａｒｄ）リガンド及びその使用方法 |
| JP2019522644A (ja) * | 2016-06-10 | 2019-08-15 | ユニバーシティ オブ テネシー リサーチ ファウンデーション | 選択的アンドロゲン受容体分解剤（ｓａｒｄ）リガンドおよびその使用方法 |
| JP2021138780A (ja) * | 2016-06-10 | 2021-09-16 | ユニバーシティ オブ テネシー リサーチ ファウンデーション | 選択的アンドロゲン受容体分解剤（ｓａｒｄ）リガンドおよびその使用方法 |
| JP7382987B2 (ja) | 2016-06-10 | 2023-11-17 | ユニバーシティ オブ テネシー リサーチ ファウンデーション | 選択的アンドロゲン受容体分解剤（ｓａｒｄ）リガンドおよびその使用方法 |
| JP2023514455A (ja) * | 2020-02-25 | 2023-04-05 | ユニバーシティ オブ テネシー リサーチ ファウンデーション | 選択的アンドロゲン受容体共有結合性アンタゴニスト（ｓａｒｃａ）およびその使用方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| AU2003287077A1 (en) | 2004-05-04 |
| EP1562594A4 (en) | 2008-12-17 |
| EP1562594A2 (en) | 2005-08-17 |
| CN1726034A (zh) | 2006-01-25 |
| CA2502209A1 (en) | 2004-04-29 |
| WO2004035738A2 (en) | 2004-04-29 |
| TW200503711A (en) | 2005-02-01 |
| US20040147550A1 (en) | 2004-07-29 |
| AU2003287077B2 (en) | 2007-09-20 |
| WO2004035738A3 (en) | 2004-07-15 |
| US20080319009A1 (en) | 2008-12-25 |
| US7253210B2 (en) | 2007-08-07 |
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