JP2006505533A5 - - Google Patents

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Publication number
JP2006505533A5
JP2006505533A5 JP2004537065A JP2004537065A JP2006505533A5 JP 2006505533 A5 JP2006505533 A5 JP 2006505533A5 JP 2004537065 A JP2004537065 A JP 2004537065A JP 2004537065 A JP2004537065 A JP 2004537065A JP 2006505533 A5 JP2006505533 A5 JP 2006505533A5
Authority
JP
Japan
Prior art keywords
pyrrolidin
urea
methyl
quinolin
diphenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
JP2004537065A
Other languages
English (en)
Japanese (ja)
Other versions
JP2006505533A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2003/010154 external-priority patent/WO2004026836A2/en
Publication of JP2006505533A publication Critical patent/JP2006505533A/ja
Publication of JP2006505533A5 publication Critical patent/JP2006505533A5/ja
Abandoned legal-status Critical Current

Links

JP2004537065A 2002-09-17 2003-09-12 1−ピリジン−4−イル−尿素誘導体 Abandoned JP2006505533A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP0210417 2002-09-17
PCT/EP2003/010154 WO2004026836A2 (en) 2002-09-17 2003-09-12 1-pyridin-4-yl-urea derivatives

Publications (2)

Publication Number Publication Date
JP2006505533A JP2006505533A (ja) 2006-02-16
JP2006505533A5 true JP2006505533A5 (enExample) 2006-10-19

Family

ID=32010909

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2004537065A Abandoned JP2006505533A (ja) 2002-09-17 2003-09-12 1−ピリジン−4−イル−尿素誘導体

Country Status (13)

Country Link
US (1) US20060094716A1 (enExample)
EP (1) EP1554249A2 (enExample)
JP (1) JP2006505533A (enExample)
KR (1) KR20050043967A (enExample)
CN (1) CN1681789A (enExample)
AU (1) AU2003270186A1 (enExample)
BR (1) BR0314353A (enExample)
CA (1) CA2496624A1 (enExample)
MX (1) MXPA05002839A (enExample)
NO (1) NO20050932L (enExample)
RU (1) RU2005111589A (enExample)
WO (1) WO2004026836A2 (enExample)
ZA (1) ZA200502009B (enExample)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004050024A2 (en) 2002-11-27 2004-06-17 Incyte Corporation 3-aminopyrrolidine derivatives as modulators of chemokine receptors
WO2004073634A2 (en) 2003-02-20 2004-09-02 Encysive Pharmaceuticals Inc. Phenylenediamine urotensin-ii receptor antagonists and ccr-9 antagonists
US7288538B2 (en) 2003-02-20 2007-10-30 Encysive Pharmaceuticals, Inc. Phenylenediamine urotensin-II receptor antagonists and CCR-9 antagonists
JP2006519258A (ja) 2003-02-28 2006-08-24 エンサイシブ・ファーマシューティカルズ・インコーポレイテッド ピリジン、ピリミジン、キノリン、キナゾリンおよびナフタレン系のウロテンシン−ii受容体拮抗薬
US7320989B2 (en) 2003-02-28 2008-01-22 Encysive Pharmaceuticals, Inc. Pyridine, pyrimidine, quinoline, quinazoline, and naphthalene urotensin-II receptor antagonists
EP1603899B1 (en) 2003-03-06 2009-08-26 Glaxo Group Limited Heterocyclic urea derivatives for the treatment of pain
US7514562B2 (en) 2003-03-07 2009-04-07 Glaxo Group Limited Urea derivatives and their use as vanilloid receptor antagonists in the treatment of pain
GB0305426D0 (en) 2003-03-08 2003-04-16 Glaxo Group Ltd Novel compounds
WO2004089296A2 (en) 2003-04-03 2004-10-21 The Regents Of The University Of California Improved inhibitors for the soluble epoxide hydrolase
JP4851328B2 (ja) 2003-09-26 2012-01-11 アクテリオン ファーマシューティカルズ リミテッド 新規なピリジン誘導体
EP1765311A4 (en) 2004-03-16 2009-04-29 Univ California REDUCTION OF NEPHROPATHY WITH INHIBITORS OF SOLUBLE EPOXY HYDROLASE AND EPOXYEICOSANOIDS
AR051213A1 (es) * 2004-10-12 2006-12-27 Actelion Pharmaceuticals Ltd 1-(2-(4-bencil-4-hidroxi-piperidin-1-il)-etil)-3-(2-metil-quinolin-4-il)-urea como una sal sulfato cristalina
WO2006045119A2 (en) 2004-10-20 2006-04-27 The Regents Of The University Of California Improved inhibitors for the soluble epoxide hydrolase
NZ566023A (en) 2005-09-21 2010-02-26 Pfizer Ltd Carboxamide derivatives as muscarinic receptor antagonists
AR059826A1 (es) 2006-03-13 2008-04-30 Univ California Inhibidores de urea conformacionalmente restringidos de epoxido hidrolasa soluble
WO2008144268A1 (en) * 2007-05-15 2008-11-27 Boehringer Ingelheim International Gmbh Urotensin ii receptor antagonists
AU2009254738B2 (en) * 2008-06-03 2014-05-08 Idorsia Pharmaceuticals Ltd [4-(1-amino-ethyl) -cyclohexyl] -methyl-amine and [6-(1-amino-ethyl) -tetrahydro- pyran-3-yl] -methyl-amine derivatives as antibacterials
EP2528604B1 (en) 2010-01-29 2017-11-22 The Regents of the University of California Acyl piperidine inhibitors of soluble epoxide hydrolase
EP2552893B1 (en) * 2010-03-31 2014-10-29 Actelion Pharmaceuticals Ltd. Antibacterial isoquinolin-3-ylurea derivatives
CA2826034A1 (en) * 2011-01-28 2012-08-02 University Of Kentucky Research Foundation Stilbene analogs and methods of treating cancer
EP3247692B1 (en) * 2015-01-23 2022-09-07 GVK Biosciences Private Limited Inhibitors of trka kinase
CN107056673B (zh) * 2016-09-09 2019-10-29 南京工业大学 一种3,4-二芳基马来酰亚胺衍生物及其制备方法与应用
CN106432039B (zh) * 2016-09-27 2019-02-22 南京工业大学 3,4-二芳基马来酰亚胺衍生物及其制备方法与应用
WO2020042972A1 (zh) * 2018-08-27 2020-03-05 北京赛特明强医药科技有限公司 脲取代的芳环连二噁烷并喹唑啉或喹啉类化合物、组合物及其应用
PT4097099T (pt) 2020-02-07 2024-07-19 Gasherbrum Bio Inc Agonistas heterocíclicos de glp-1
WO2022052958A1 (en) 2020-09-10 2022-03-17 Gasherbrum Bio, Inc. Heterocyclic glp-1 agonists
KR20250168210A (ko) 2023-02-16 2025-12-02 가셔브룸 바이오, 인크. 헤테로시클릭 glp-1 효능제
CN119219821A (zh) * 2024-12-03 2024-12-31 江苏金杉新材料有限公司 用于湿法冶金的苯乙烯系阴离子树脂及其制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR016817A1 (es) * 1997-08-14 2001-08-01 Smithkline Beecham Plc Derivados de fenilurea o feniltiourea, procedimiento para su preparacion, coleccion de compuestos, compuestos intermediarios, composicion farmaceutica,metodo de tratamiento y uso de dichos compuestos para la manufactura de un medicamento
AUPP003197A0 (en) * 1997-09-03 1997-11-20 Fujisawa Pharmaceutical Co., Ltd. New heterocyclic compounds
DE60013250T2 (de) * 1999-02-12 2005-09-08 Smithkline Beecham P.L.C., Brentford Phenylharnstoff- und Phenylthioharnstoffderivate als Orexinrezeptorantagonisten
JP2004529132A (ja) * 2001-03-27 2004-09-24 アクテリオン ファマシューティカルズ リミテッド 1,2,3,4−テトラヒドロイソキノリン誘導体
CA2473892C (en) * 2001-12-04 2010-09-21 Actelion Pharmaceuticals Ltd Novel quinoline derivatives

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