JP2006502157A - ナフチルエーテル化合物及びそれらの使用 - Google Patents
ナフチルエーテル化合物及びそれらの使用 Download PDFInfo
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- JP2006502157A JP2006502157A JP2004533952A JP2004533952A JP2006502157A JP 2006502157 A JP2006502157 A JP 2006502157A JP 2004533952 A JP2004533952 A JP 2004533952A JP 2004533952 A JP2004533952 A JP 2004533952A JP 2006502157 A JP2006502157 A JP 2006502157A
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- Prior art keywords
- depression
- disorder
- alkyl
- pharmaceutically acceptable
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0202674A SE0202674D0 (sv) | 2002-09-09 | 2002-09-09 | Naphthyl ether compounds and their use |
| SE0301052A SE0301052D0 (sv) | 2003-04-08 | 2003-04-08 | Naphthyl ether compounds and their use |
| PCT/SE2003/001399 WO2004022539A1 (en) | 2002-09-09 | 2003-09-08 | Naphthyl ether compounds and their use |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2006502157A true JP2006502157A (ja) | 2006-01-19 |
| JP2006502157A5 JP2006502157A5 (OSRAM) | 2006-10-19 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004533952A Pending JP2006502157A (ja) | 2002-09-09 | 2003-09-08 | ナフチルエーテル化合物及びそれらの使用 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20050245572A1 (OSRAM) |
| EP (1) | EP1546101A1 (OSRAM) |
| JP (1) | JP2006502157A (OSRAM) |
| AU (1) | AU2003258937A1 (OSRAM) |
| WO (1) | WO2004022539A1 (OSRAM) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7494986B2 (en) * | 2004-07-20 | 2009-02-24 | Bristol-Myers Squibb Company | Cycloalkylamine derivatives as NK-1/SSRI antagonists |
| WO2007003961A2 (en) * | 2005-06-30 | 2007-01-11 | Prosidion Limited | Gpcr agonists |
| US20070249607A1 (en) | 2006-04-17 | 2007-10-25 | Bristol-Myers Squibb Company | Nk-1 and serotonin transporter inhibitors |
| US8071778B2 (en) | 2006-07-27 | 2011-12-06 | Bristol-Myers Squibb Company | Substituted heterocyclic ethers and their use in CNS disorders |
| CN101495470A (zh) * | 2006-07-27 | 2009-07-29 | 百时美施贵宝公司 | 4-芳基烷氧基甲基-4-苯基哌啶及其作为神经激肽受体拮抗剂治疗cns疾病的用途 |
| US8026257B2 (en) * | 2007-07-11 | 2011-09-27 | Bristol-Myers Squibb Company | Substituted heterocyclic ethers and their use in CNS disorders |
| US20090018163A1 (en) * | 2007-07-11 | 2009-01-15 | Bristol-Myers Squibb Company | Substituted Heterocyclic Ethers and Their Use in CNS Disorders |
| US7632861B2 (en) | 2007-11-13 | 2009-12-15 | Bristol-Myers Squibb Company | Substituted heterocyclic ethers and their use in CNS disorders |
| WO2009096941A1 (en) * | 2008-01-28 | 2009-08-06 | Bristol-Myers Squibb Company | Substituted heterocyclic ethers and their use in cns disorders |
| WO2014142761A1 (en) * | 2013-03-15 | 2014-09-18 | Nanyang Technological University | 3-piperidone compounds and their use as neurokinin-1 (nk1) receptor antagonists |
| CN108530262A (zh) * | 2018-06-15 | 2018-09-14 | 贾红琴 | 一种2-溴芴的合成方法 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
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| US5620989A (en) * | 1992-10-28 | 1997-04-15 | Merck Sharp & Dohme Limited | 4-Arylmethyloxymethyl piperidines as tachykinin antagonsits |
| EP0739336B1 (en) * | 1994-01-13 | 1998-08-26 | MERCK SHARP & DOHME LTD. | Gem-disubstituted azacyclic tachykinin antagonists |
| US5491140A (en) * | 1994-06-30 | 1996-02-13 | Eli Lilly And Company | Naphthyl tachykinin receptor antagonists to treat physiological conditions |
| GB9904786D0 (en) * | 1999-03-02 | 1999-04-28 | Merck Sharp & Dohme | Therapeutic agents |
| ATE416162T1 (de) * | 2002-08-29 | 2008-12-15 | Astrazeneca Ab | Naphthamidderivate und deren verwendung |
| AU2003291589A1 (en) * | 2002-12-20 | 2004-07-14 | Astrazeneca Ab | Piperidine amine compounds and their use |
-
2003
- 2003-09-08 AU AU2003258937A patent/AU2003258937A1/en not_active Abandoned
- 2003-09-08 EP EP03794408A patent/EP1546101A1/en not_active Withdrawn
- 2003-09-08 JP JP2004533952A patent/JP2006502157A/ja active Pending
- 2003-09-08 WO PCT/SE2003/001399 patent/WO2004022539A1/en not_active Ceased
- 2003-09-08 US US10/527,280 patent/US20050245572A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2004022539A1 (en) | 2004-03-18 |
| US20050245572A1 (en) | 2005-11-03 |
| AU2003258937A1 (en) | 2004-03-29 |
| EP1546101A1 (en) | 2005-06-29 |
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