JP2005533804A5 - - Google Patents

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Publication number
JP2005533804A5
JP2005533804A5 JP2004515329A JP2004515329A JP2005533804A5 JP 2005533804 A5 JP2005533804 A5 JP 2005533804A5 JP 2004515329 A JP2004515329 A JP 2004515329A JP 2004515329 A JP2004515329 A JP 2004515329A JP 2005533804 A5 JP2005533804 A5 JP 2005533804A5
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JP
Japan
Prior art keywords
formula
compounds
iii
prepared
phosgene
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2004515329A
Other languages
English (en)
Japanese (ja)
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JP2005533804A (ja
Filing date
Publication date
Priority claimed from SE0201980A external-priority patent/SE0201980D0/xx
Application filed filed Critical
Publication of JP2005533804A publication Critical patent/JP2005533804A/ja
Publication of JP2005533804A5 publication Critical patent/JP2005533804A5/ja
Pending legal-status Critical Current

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JP2004515329A 2002-06-24 2003-06-23 システイン・プロテアーゼ活性に関係する疾患を処置するための新規プリン−もしくはピロール−[2,3−d]ピリミジン−2−カルボニトリル Pending JP2005533804A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0201980A SE0201980D0 (sv) 2002-06-24 2002-06-24 Novel compounds
PCT/SE2003/001079 WO2004000843A1 (en) 2002-06-24 2003-06-23 NOVEL PURINE- OR PYRROLOL[2,3-d]PYRIMIDINE-2-CARBONITILES FOR TREATING DISEASES ASSOCIATED WITH CYSTEINE PROTEASE ACTIVITY

Publications (2)

Publication Number Publication Date
JP2005533804A JP2005533804A (ja) 2005-11-10
JP2005533804A5 true JP2005533804A5 (OSRAM) 2006-08-10

Family

ID=20288336

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2004515329A Pending JP2005533804A (ja) 2002-06-24 2003-06-23 システイン・プロテアーゼ活性に関係する疾患を処置するための新規プリン−もしくはピロール−[2,3−d]ピリミジン−2−カルボニトリル

Country Status (8)

Country Link
US (3) US7439240B2 (OSRAM)
EP (1) EP1532148B1 (OSRAM)
JP (1) JP2005533804A (OSRAM)
AU (1) AU2003243096A1 (OSRAM)
DE (1) DE60311272T2 (OSRAM)
ES (1) ES2279162T3 (OSRAM)
SE (1) SE0201980D0 (OSRAM)
WO (1) WO2004000843A1 (OSRAM)

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WO2009107767A1 (ja) * 2008-02-29 2009-09-03 大日本住友製薬株式会社 H4受容体アンタゴニスト作用を有する新規2環性ピリミジン誘導体
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WO2010059418A1 (en) * 2008-11-19 2010-05-27 The Government Of The U.S.A. As Represented By The Secretary Of The Dept. Of Health & Human Services Substituted triazine and purine compounds, methods of inhibiting cruzain and rhodesain and methods of treating chagas disease and african trypanosomiasis
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CN104837839A (zh) 2012-11-08 2015-08-12 辉瑞公司 作为多巴胺d1配体的杂芳族化合物
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GB0220187D0 (en) * 2002-08-30 2002-10-09 Novartis Ag Organic compounds
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GB0304640D0 (en) 2003-02-28 2003-04-02 Novartis Ag Organic compounds
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