JP2005506949A - ケモカイン受容体の調節剤としてのジアミン - Google Patents

ケモカイン受容体の調節剤としてのジアミン Download PDF

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JP2005506949A
JP2005506949A JP2002551518A JP2002551518A JP2005506949A JP 2005506949 A JP2005506949 A JP 2005506949A JP 2002551518 A JP2002551518 A JP 2002551518A JP 2002551518 A JP2002551518 A JP 2002551518A JP 2005506949 A JP2005506949 A JP 2005506949A
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amino
methyl
crr
replaced
trifluoromethyl
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JP2005506949A5 (enExample
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パーシー・カーター
ロバート・チャーニー
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Bristol Myers Squibb Pharma Co
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Bristol Myers Squibb Pharma Co
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/63—One oxygen atom
    • C07D213/64—One oxygen atom attached in position 2 or 6
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    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
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JP2002551518A 2000-12-20 2001-12-20 ケモカイン受容体の調節剤としてのジアミン Withdrawn JP2005506949A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25685500P 2000-12-20 2000-12-20
PCT/US2001/050619 WO2002050019A2 (en) 2000-12-20 2001-12-20 Diamines as modulators of chemokine receptor activity

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HUP0303540A2 (hu) 2004-01-28
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