JP2004536049A5 - - Google Patents
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- Publication number
- JP2004536049A5 JP2004536049A5 JP2002581366A JP2002581366A JP2004536049A5 JP 2004536049 A5 JP2004536049 A5 JP 2004536049A5 JP 2002581366 A JP2002581366 A JP 2002581366A JP 2002581366 A JP2002581366 A JP 2002581366A JP 2004536049 A5 JP2004536049 A5 JP 2004536049A5
- Authority
- JP
- Japan
- Prior art keywords
- substituted
- unsubstituted
- alkyl
- aryl
- heterocyclic group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 125000003118 aryl group Chemical group 0.000 claims 47
- 125000000217 alkyl group Chemical group 0.000 claims 45
- 125000000623 heterocyclic group Chemical group 0.000 claims 41
- 150000001875 compounds Chemical class 0.000 claims 36
- 125000003710 aryl alkyl group Chemical group 0.000 claims 35
- RTZKZFJDLAIYFH-UHFFFAOYSA-N ether Substances CCOCC RTZKZFJDLAIYFH-UHFFFAOYSA-N 0.000 claims 25
- 150000002170 ethers Chemical class 0.000 claims 25
- 125000004404 heteroalkyl group Chemical group 0.000 claims 22
- 150000003568 thioethers Chemical class 0.000 claims 22
- -1 phosphinoyl Chemical group 0.000 claims 13
- 125000005843 halogen group Chemical group 0.000 claims 11
- 229910052739 hydrogen Inorganic materials 0.000 claims 10
- 239000001257 hydrogen Substances 0.000 claims 10
- 125000000467 secondary amino group Chemical class [H]N([*:1])[*:2] 0.000 claims 10
- 150000003512 tertiary amines Chemical class 0.000 claims 10
- 150000002431 hydrogen Chemical class 0.000 claims 9
- UEZVMMHDMIWARA-UHFFFAOYSA-M phosphonate Chemical class [O-]P(=O)=O UEZVMMHDMIWARA-UHFFFAOYSA-M 0.000 claims 8
- 229920000642 polymer Polymers 0.000 claims 8
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims 8
- 150000003839 salts Chemical class 0.000 claims 8
- 150000002148 esters Chemical class 0.000 claims 7
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 7
- 229910052757 nitrogen Inorganic materials 0.000 claims 7
- 125000004433 nitrogen atom Chemical group N* 0.000 claims 7
- 150000002576 ketones Chemical class 0.000 claims 6
- 150000003457 sulfones Chemical class 0.000 claims 6
- 239000012453 solvate Substances 0.000 claims 5
- UCKMPCXJQFINFW-UHFFFAOYSA-N Sulphide Chemical compound [S-2] UCKMPCXJQFINFW-UHFFFAOYSA-N 0.000 claims 3
- 125000005073 adamantyl group Chemical group C12(CC3CC(CC(C1)C3)C2)* 0.000 claims 3
- 150000003008 phosphonic acid esters Chemical class 0.000 claims 3
- 150000003462 sulfoxides Chemical class 0.000 claims 3
- 229910052782 aluminium Inorganic materials 0.000 claims 2
- 229910052788 barium Inorganic materials 0.000 claims 2
- 229910052794 bromium Inorganic materials 0.000 claims 2
- 229910052793 cadmium Inorganic materials 0.000 claims 2
- 229910052801 chlorine Inorganic materials 0.000 claims 2
- 150000004696 coordination complex Chemical class 0.000 claims 2
- 229910052802 copper Inorganic materials 0.000 claims 2
- PXBRQCKWGAHEHS-UHFFFAOYSA-N dichlorodifluoromethane Chemical compound FC(F)(Cl)Cl PXBRQCKWGAHEHS-UHFFFAOYSA-N 0.000 claims 2
- 125000001072 heteroaryl group Chemical group 0.000 claims 2
- 229910052738 indium Inorganic materials 0.000 claims 2
- 229910052740 iodine Inorganic materials 0.000 claims 2
- 229910052744 lithium Inorganic materials 0.000 claims 2
- 229910052749 magnesium Inorganic materials 0.000 claims 2
- 229910052748 manganese Inorganic materials 0.000 claims 2
- 239000002184 metal Substances 0.000 claims 2
- 229910052751 metal Inorganic materials 0.000 claims 2
- 229910052700 potassium Inorganic materials 0.000 claims 2
- 229910052708 sodium Inorganic materials 0.000 claims 2
- 229910052717 sulfur Inorganic materials 0.000 claims 2
- 125000004434 sulfur atom Chemical group 0.000 claims 2
- 125000000999 tert-butyl group Chemical group [H]C([H])([H])C(*)(C([H])([H])[H])C([H])([H])[H] 0.000 claims 2
- 229910052719 titanium Inorganic materials 0.000 claims 2
- 125000005039 triarylmethyl group Chemical group 0.000 claims 2
- 229910052725 zinc Inorganic materials 0.000 claims 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 1
- 239000002253 acid Substances 0.000 claims 1
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims 1
- 125000000475 sulfinyl group Chemical group [*:2]S([*:1])=O 0.000 claims 1
- 229940124530 sulfonamide Drugs 0.000 claims 1
- 150000003456 sulfonamides Chemical class 0.000 claims 1
- 125000001302 tertiary amino group Chemical group 0.000 claims 1
- 125000003944 tolyl group Chemical group 0.000 claims 1
- 239000013638 trimer Substances 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US28333701P | 2001-04-13 | 2001-04-13 | |
| PCT/US2002/011471 WO2002083608A2 (en) | 2001-04-13 | 2002-04-12 | Methods of preparing sulfinamide and sulfoxides |
| US10/120,541 US7064214B2 (en) | 2001-04-13 | 2002-04-12 | Methods of preparing sulfinamides and sulfoxides |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2004536049A JP2004536049A (ja) | 2004-12-02 |
| JP2004536049A5 true JP2004536049A5 (enExample) | 2005-12-22 |
Family
ID=26818471
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002581366A Pending JP2004536049A (ja) | 2001-04-13 | 2002-04-12 | スルフィンアミドおよびスルホキシドの製造方法 |
Country Status (4)
| Country | Link |
|---|---|
| US (3) | US7064214B2 (enExample) |
| JP (1) | JP2004536049A (enExample) |
| AU (1) | AU2002338655A1 (enExample) |
| WO (1) | WO2002083608A2 (enExample) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2002083608A2 (en) * | 2001-04-13 | 2002-10-24 | Apsinterm Llc | Methods of preparing sulfinamide and sulfoxides |
| MXPA04009843A (es) * | 2002-04-10 | 2005-08-16 | Apsinterm Llc | Metodo para la preparacion de estereoisomeros de amina. |
| JP2006514108A (ja) * | 2002-12-19 | 2006-04-27 | テバ ファーマシューティカル インダストリーズ リミティド | パントプラゾールナトリウムの固体状態、それらの調製方法、及び公知のパントプラゾールナトリウム水和物の調製方法 |
| US20040235904A1 (en) * | 2003-03-12 | 2004-11-25 | Nina Finkelstein | Crystalline and amorphous solids of pantoprazole and processes for their preparation |
| WO2004111029A2 (en) * | 2003-06-10 | 2004-12-23 | Teva Pharmaceutical Industries Ltd. | Process for preparing 2-[(pyridinyl)methyl]sulfinyl-substituted benzimidazoles and novel chlorinated derivatives of pantoprazole |
| US7582634B2 (en) | 2005-02-18 | 2009-09-01 | Wyeth | 7-substituted imidazo[4,5-c]pyridine antagonists of gonadotropin releasing hormone receptor |
| US7534796B2 (en) | 2005-02-18 | 2009-05-19 | Wyeth | Imidazo[4,5-b]pyridine antagonists of gonadotropin releasing hormone receptor |
| US7538113B2 (en) | 2005-02-18 | 2009-05-26 | Wyeth | 4-substituted imidazo[4,5-c]pyridine antagonists of gonadotropin releasing hormone receptor |
| US7531542B2 (en) | 2005-05-18 | 2009-05-12 | Wyeth | Benzooxazole and benzothiazole antagonists of gonadotropin releasing hormone receptor |
| US7582636B2 (en) | 2005-05-26 | 2009-09-01 | Wyeth | Piperazinylimidazopyridine and piperazinyltriazolopyridine antagonists of Gonadotropin Releasing Hormone receptor |
| JP6030752B2 (ja) | 2012-05-09 | 2016-11-24 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | オキセタン−３−イルメタンアミンの製造方法 |
| EP2922835B1 (en) * | 2012-11-21 | 2017-08-09 | Boehringer Ingelheim International GmbH | Process for making n-sulfinyl alpha-amino amides |
| US20140275582A1 (en) * | 2013-03-14 | 2014-09-18 | Texas Tech University | Chiral 2-arylpropyl-2-sulfinamide and chiral n-2-arylpropyl-2-sulfinylimines and synthesis thereof |
| US9731985B2 (en) | 2015-06-03 | 2017-08-15 | Lg Nanoh2O, Inc. | Chemical additives for enhancement of water flux of a membrane |
| US9695065B2 (en) | 2015-06-03 | 2017-07-04 | Lg Nanoh2O, Inc. | Combination of chemical additives for enhancement of water flux of a membrane |
| US9724651B2 (en) | 2015-07-14 | 2017-08-08 | Lg Nanoh2O, Inc. | Chemical additives for water flux enhancement |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3311636A1 (de) | 1983-03-30 | 1984-10-04 | Bayer Ag, 5090 Leverkusen | Neue fuenfgliedrige stickstoffhaltige heterocyclen, verfahren zu ihrer herstellung sowie ihre verwendung als schaedlingsbekaempfungsmittel |
| US5271812A (en) | 1991-06-19 | 1993-12-21 | Sepracor, Inc. | Electrocatalytic oxidation method for the production of cyclic sulfates and sulfamidates |
| SE9301830D0 (sv) * | 1993-05-28 | 1993-05-28 | Ab Astra | New compounds |
| AU2395095A (en) * | 1994-04-29 | 1995-11-29 | G.D. Searle & Co. | Method of using (h+/k+) atpase inhibitors as antiviral agents |
| SE504459C2 (sv) * | 1994-07-15 | 1997-02-17 | Astra Ab | Förfarande för framställning av substituerade sulfoxider |
| GB9423968D0 (en) * | 1994-11-28 | 1995-01-11 | Astra Ab | Resolution |
| WO2002083608A2 (en) * | 2001-04-13 | 2002-10-24 | Apsinterm Llc | Methods of preparing sulfinamide and sulfoxides |
| MXPA04009843A (es) | 2002-04-10 | 2005-08-16 | Apsinterm Llc | Metodo para la preparacion de estereoisomeros de amina. |
-
2002
- 2002-04-12 WO PCT/US2002/011471 patent/WO2002083608A2/en not_active Ceased
- 2002-04-12 US US10/120,541 patent/US7064214B2/en not_active Expired - Fee Related
- 2002-04-12 JP JP2002581366A patent/JP2004536049A/ja active Pending
- 2002-04-12 AU AU2002338655A patent/AU2002338655A1/en not_active Abandoned
-
2006
- 2006-01-27 US US11/340,551 patent/US7256297B2/en not_active Expired - Fee Related
-
2007
- 2007-07-30 US US11/830,166 patent/US20070293682A1/en not_active Abandoned
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