JP2004536049A - スルフィンアミドおよびスルホキシドの製造方法 - Google Patents

スルフィンアミドおよびスルホキシドの製造方法 Download PDF

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Publication number
JP2004536049A
JP2004536049A JP2002581366A JP2002581366A JP2004536049A JP 2004536049 A JP2004536049 A JP 2004536049A JP 2002581366 A JP2002581366 A JP 2002581366A JP 2002581366 A JP2002581366 A JP 2002581366A JP 2004536049 A JP2004536049 A JP 2004536049A
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JP
Japan
Prior art keywords
substituted
unsubstituted
formula
aryl
compound
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Pending
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JP2002581366A
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English (en)
Japanese (ja)
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JP2004536049A5 (https=
Inventor
クリス・ヒュー・セナナエイク
ジェンユ・ハン
ディリープクマー・クリシュナマーシー
デレク・フラム
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Apsinterm LLC
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Apsinterm LLC
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Application filed by Apsinterm LLC filed Critical Apsinterm LLC
Publication of JP2004536049A publication Critical patent/JP2004536049A/ja
Publication of JP2004536049A5 publication Critical patent/JP2004536049A5/ja
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D291/00—Heterocyclic compounds containing rings having nitrogen, oxygen and sulfur atoms as the only ring hetero atoms
    • C07D291/02—Heterocyclic compounds containing rings having nitrogen, oxygen and sulfur atoms as the only ring hetero atoms not condensed with other rings
    • C07D291/04—Five-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C313/00—Sulfinic acids; Sulfenic acids; Halides, esters or anhydrides thereof; Amides of sulfinic or sulfenic acids, i.e. compounds having singly-bound oxygen atoms of sulfinic or sulfenic groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C313/02—Sulfinic acids; Derivatives thereof
    • C07C313/04—Sulfinic acids; Esters thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C315/00—Preparation of sulfones; Preparation of sulfoxides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/02—Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to acyclic carbon atoms
    • C07C317/04—Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/28—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D291/00—Heterocyclic compounds containing rings having nitrogen, oxygen and sulfur atoms as the only ring hetero atoms
    • C07D291/08—Heterocyclic compounds containing rings having nitrogen, oxygen and sulfur atoms as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00—Systems containing two condensed rings
    • C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
    • C07C2602/04—One of the condensed rings being a six-membered aromatic ring
    • C07C2602/08—One of the condensed rings being a six-membered aromatic ring the other ring being five-membered, e.g. indane

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP2002581366A 2001-04-13 2002-04-12 スルフィンアミドおよびスルホキシドの製造方法 Pending JP2004536049A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US28333701P 2001-04-13 2001-04-13
US10/120,541 US7064214B2 (en) 2001-04-13 2002-04-12 Methods of preparing sulfinamides and sulfoxides
PCT/US2002/011471 WO2002083608A2 (en) 2001-04-13 2002-04-12 Methods of preparing sulfinamide and sulfoxides

Publications (2)

Publication Number Publication Date
JP2004536049A true JP2004536049A (ja) 2004-12-02
JP2004536049A5 JP2004536049A5 (https=) 2005-12-22

Family

ID=26818471

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002581366A Pending JP2004536049A (ja) 2001-04-13 2002-04-12 スルフィンアミドおよびスルホキシドの製造方法

Country Status (4)

Country Link
US (3) US7064214B2 (https=)
JP (1) JP2004536049A (https=)
AU (1) AU2002338655A1 (https=)
WO (1) WO2002083608A2 (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005522525A (ja) * 2002-04-10 2005-07-28 アプシンターム・リミテッド・ライアビリティ・カンパニー アミン立体異性体の製造方法

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002083608A2 (en) * 2001-04-13 2002-10-24 Apsinterm Llc Methods of preparing sulfinamide and sulfoxides
US7507829B2 (en) * 2002-12-19 2009-03-24 Teva Pharmaceuticals Industries, Ltd Solid states of pantoprazole sodium, processes for preparing them and processes for preparing known pantoprazole sodium hydrates
WO2004080961A2 (en) * 2003-03-12 2004-09-23 Teva Pharmaceutical Industries Ltd. Crystalline and amorphous solids of pantoprazole and processes for their preparation
US7683177B2 (en) * 2003-06-10 2010-03-23 Teva Pharmaceutical Industries Ltd Process for preparing 2-[(pyridinyl)methyl]sulfinyl-substituted benzimidazoles and novel chlorinated derivatives of pantoprazole
US7582634B2 (en) 2005-02-18 2009-09-01 Wyeth 7-substituted imidazo[4,5-c]pyridine antagonists of gonadotropin releasing hormone receptor
US7534796B2 (en) 2005-02-18 2009-05-19 Wyeth Imidazo[4,5-b]pyridine antagonists of gonadotropin releasing hormone receptor
US7538113B2 (en) 2005-02-18 2009-05-26 Wyeth 4-substituted imidazo[4,5-c]pyridine antagonists of gonadotropin releasing hormone receptor
US7531542B2 (en) 2005-05-18 2009-05-12 Wyeth Benzooxazole and benzothiazole antagonists of gonadotropin releasing hormone receptor
US7582636B2 (en) 2005-05-26 2009-09-01 Wyeth Piperazinylimidazopyridine and piperazinyltriazolopyridine antagonists of Gonadotropin Releasing Hormone receptor
WO2013169531A1 (en) 2012-05-09 2013-11-14 Boehringer Ingelheim International Gmbh Methods for making oxetan-3-ylmethanamines
WO2014081558A1 (en) * 2012-11-21 2014-05-30 Boehringer Ingelheim International Gmbh PROCESS FOR MAKING N-SULFINYL a-AMINO AMIDES
US20140275582A1 (en) * 2013-03-14 2014-09-18 Texas Tech University Chiral 2-arylpropyl-2-sulfinamide and chiral n-2-arylpropyl-2-sulfinylimines and synthesis thereof
US9695065B2 (en) 2015-06-03 2017-07-04 Lg Nanoh2O, Inc. Combination of chemical additives for enhancement of water flux of a membrane
US9731985B2 (en) 2015-06-03 2017-08-15 Lg Nanoh2O, Inc. Chemical additives for enhancement of water flux of a membrane
US9724651B2 (en) 2015-07-14 2017-08-08 Lg Nanoh2O, Inc. Chemical additives for water flux enhancement

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3311636A1 (de) 1983-03-30 1984-10-04 Bayer Ag, 5090 Leverkusen Neue fuenfgliedrige stickstoffhaltige heterocyclen, verfahren zu ihrer herstellung sowie ihre verwendung als schaedlingsbekaempfungsmittel
US5271812A (en) 1991-06-19 1993-12-21 Sepracor, Inc. Electrocatalytic oxidation method for the production of cyclic sulfates and sulfamidates
SE9301830D0 (sv) * 1993-05-28 1993-05-28 Ab Astra New compounds
WO1995029897A1 (en) * 1994-04-29 1995-11-09 G.D. Searle & Co. METHOD OF USING (H+/K+) ATPase INHIBITORS AS ANTIVIRAL AGENTS
SE504459C2 (sv) 1994-07-15 1997-02-17 Astra Ab Förfarande för framställning av substituerade sulfoxider
GB9423968D0 (en) 1994-11-28 1995-01-11 Astra Ab Resolution
WO2002083608A2 (en) * 2001-04-13 2002-10-24 Apsinterm Llc Methods of preparing sulfinamide and sulfoxides
CN101613310A (zh) 2002-04-10 2009-12-30 艾普辛特姆有限责任公司 胺立体异构体的制备方法

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005522525A (ja) * 2002-04-10 2005-07-28 アプシンターム・リミテッド・ライアビリティ・カンパニー アミン立体異性体の製造方法

Also Published As

Publication number Publication date
US20070293682A1 (en) 2007-12-20
US7064214B2 (en) 2006-06-20
WO2002083608A2 (en) 2002-10-24
US20060128767A1 (en) 2006-06-15
US20030083517A1 (en) 2003-05-01
US7256297B2 (en) 2007-08-14
WO2002083608A3 (en) 2003-10-16
AU2002338655A1 (en) 2002-10-28

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