JP2004535444A5 - - Google Patents
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- Publication number
- JP2004535444A5 JP2004535444A5 JP2003508683A JP2003508683A JP2004535444A5 JP 2004535444 A5 JP2004535444 A5 JP 2004535444A5 JP 2003508683 A JP2003508683 A JP 2003508683A JP 2003508683 A JP2003508683 A JP 2003508683A JP 2004535444 A5 JP2004535444 A5 JP 2004535444A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- process according
- thioamide
- halogen
- conversion
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP01115355 | 2001-06-26 | ||
| PCT/EP2002/006644 WO2003002498A1 (en) | 2001-06-26 | 2002-06-17 | Intermediate halophenyl derivatives and their use in a process for preparing azole derivatives |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2004535444A JP2004535444A (ja) | 2004-11-25 |
| JP2004535444A5 true JP2004535444A5 (https=) | 2005-11-17 |
| JP4125672B2 JP4125672B2 (ja) | 2008-07-30 |
Family
ID=8177821
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003508683A Expired - Lifetime JP4125672B2 (ja) | 2001-06-26 | 2002-06-17 | アゾール誘導体製造方法における中間体ハロフェニル誘導体およびそれらの使用 |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US7115643B2 (https=) |
| EP (1) | EP1399402B1 (https=) |
| JP (1) | JP4125672B2 (https=) |
| KR (1) | KR100898887B1 (https=) |
| CN (1) | CN1223564C (https=) |
| AT (1) | ATE482920T1 (https=) |
| AU (1) | AU2002321068B2 (https=) |
| BR (1) | BR0210701A (https=) |
| CA (1) | CA2449800C (https=) |
| CY (1) | CY1111510T1 (https=) |
| DE (1) | DE60237817D1 (https=) |
| DK (1) | DK1399402T3 (https=) |
| ES (1) | ES2349918T3 (https=) |
| MX (1) | MXPA03010914A (https=) |
| PT (1) | PT1399402E (https=) |
| WO (1) | WO2003002498A1 (https=) |
| ZA (1) | ZA200309101B (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8207352B2 (en) * | 2009-10-08 | 2012-06-26 | Drug Process Licensing Associates LLC | Process for the manufacture of enantiomerically pure antifungal azoles as ravuconazole and isavuconazole |
| HUE031679T2 (en) | 2012-08-07 | 2017-07-28 | Basilea Pharmaceutica Ag | Process for the preparation of isavuconazole or ravuconazole |
| US20140371179A1 (en) * | 2013-06-13 | 2014-12-18 | Professional Compounding Centers Of America | Methods and Compositions for Treating Esophageal Diseases |
| CN105801500B (zh) * | 2014-12-31 | 2018-08-24 | 四川科伦药物研究院有限公司 | 拆分艾沙康唑中间化合物消旋体的方法 |
| CN115611822B (zh) * | 2022-10-12 | 2023-09-19 | 四川澄华生物科技有限公司 | 艾沙康唑中间体的制备方法 |
| CN116478103B (zh) * | 2023-03-24 | 2025-07-25 | 四川澄华生物科技有限公司 | 一种拆分艾沙康唑中间体4的方法 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5395942A (en) | 1980-06-02 | 1995-03-07 | Zeneca Limited | Heterocyclic compounds |
| DE3942790A1 (de) * | 1989-12-23 | 1991-06-27 | Hoechst Ag | Verfahren zur herstellung von 2-(4-chlorphenyl)-3-methylbuttersaeure |
| GB9107055D0 (en) | 1991-04-04 | 1991-05-22 | Pfizer Ltd | Triazole antifungal agents |
| JP3471831B2 (ja) * | 1991-12-09 | 2003-12-02 | 富山化学工業株式会社 | 新規なトリアゾール誘導体およびその塩 |
| ES2062941B1 (es) * | 1993-03-15 | 1995-10-01 | Uriach & Cia Sa J | Nuevos derivados de azol activos por via oral. |
| NZ270418A (en) | 1994-02-07 | 1997-09-22 | Eisai Co Ltd | Polycyclic triazole & imidazole derivatives, antifungal compositions |
-
2002
- 2002-06-17 PT PT02754691T patent/PT1399402E/pt unknown
- 2002-06-17 DE DE60237817T patent/DE60237817D1/de not_active Expired - Lifetime
- 2002-06-17 AT AT02754691T patent/ATE482920T1/de active
- 2002-06-17 EP EP02754691A patent/EP1399402B1/en not_active Expired - Lifetime
- 2002-06-17 DK DK02754691.0T patent/DK1399402T3/da active
- 2002-06-17 ES ES02754691T patent/ES2349918T3/es not_active Expired - Lifetime
- 2002-06-17 BR BR0210701-5A patent/BR0210701A/pt not_active IP Right Cessation
- 2002-06-17 CA CA002449800A patent/CA2449800C/en not_active Expired - Fee Related
- 2002-06-17 AU AU2002321068A patent/AU2002321068B2/en not_active Ceased
- 2002-06-17 KR KR1020037016987A patent/KR100898887B1/ko not_active Expired - Fee Related
- 2002-06-17 MX MXPA03010914A patent/MXPA03010914A/es active IP Right Grant
- 2002-06-17 US US10/481,654 patent/US7115643B2/en not_active Expired - Lifetime
- 2002-06-17 CN CNB028126416A patent/CN1223564C/zh not_active Expired - Lifetime
- 2002-06-17 JP JP2003508683A patent/JP4125672B2/ja not_active Expired - Lifetime
- 2002-06-17 WO PCT/EP2002/006644 patent/WO2003002498A1/en not_active Ceased
-
2003
- 2003-11-21 ZA ZA2003/09101A patent/ZA200309101B/en unknown
-
2010
- 2010-12-20 CY CY20101101172T patent/CY1111510T1/el unknown
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