JP2004506042A5 - - Google Patents

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Publication number
JP2004506042A5
JP2004506042A5 JP2002519424A JP2002519424A JP2004506042A5 JP 2004506042 A5 JP2004506042 A5 JP 2004506042A5 JP 2002519424 A JP2002519424 A JP 2002519424A JP 2002519424 A JP2002519424 A JP 2002519424A JP 2004506042 A5 JP2004506042 A5 JP 2004506042A5
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JP
Japan
Prior art keywords
independently selected
embedded image
disease
compound
aromatic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2002519424A
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English (en)
Japanese (ja)
Other versions
JP4993838B2 (ja
JP2004506042A (ja
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Publication date
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Priority claimed from PCT/US2001/025015 external-priority patent/WO2002014281A1/en
Publication of JP2004506042A publication Critical patent/JP2004506042A/ja
Publication of JP2004506042A5 publication Critical patent/JP2004506042A5/ja
Application granted granted Critical
Publication of JP4993838B2 publication Critical patent/JP4993838B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2002519424A 2000-08-11 2001-08-10 P38のインヒビターとしてのピリジン誘導体 Expired - Fee Related JP4993838B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US22471900P 2000-08-11 2000-08-11
US60/224,719 2000-08-11
PCT/US2001/025015 WO2002014281A1 (en) 2000-08-11 2001-08-10 Pyridine derivatives as inhibitors of p38

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2012077626A Division JP2012149085A (ja) 2000-08-11 2012-03-29 P38のインヒビターとしてのピリジン誘導体

Publications (3)

Publication Number Publication Date
JP2004506042A JP2004506042A (ja) 2004-02-26
JP2004506042A5 true JP2004506042A5 (https=) 2008-10-02
JP4993838B2 JP4993838B2 (ja) 2012-08-08

Family

ID=22841879

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2002519424A Expired - Fee Related JP4993838B2 (ja) 2000-08-11 2001-08-10 P38のインヒビターとしてのピリジン誘導体
JP2012077626A Withdrawn JP2012149085A (ja) 2000-08-11 2012-03-29 P38のインヒビターとしてのピリジン誘導体

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2012077626A Withdrawn JP2012149085A (ja) 2000-08-11 2012-03-29 P38のインヒビターとしてのピリジン誘導体

Country Status (7)

Country Link
US (4) US7186737B2 (https=)
EP (1) EP1309560B1 (https=)
JP (2) JP4993838B2 (https=)
AU (2) AU2001283237B2 (https=)
CA (1) CA2418389A1 (https=)
MX (1) MXPA03001256A (https=)
WO (1) WO2002014281A1 (https=)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR023659A1 (es) * 1998-09-18 2002-09-04 Vertex Pharma Un compuesto inhibidor de p38, una composicion farmaceutica que lo comprende y el uso de dicha composicion en el tratamiento y prevencion de estados patologicos
ME00275B (me) 1999-01-13 2011-02-10 Bayer Corp ω-KARBOKSIARIL SUPSTITUISANI DIFENIL KARBAMIDI KAO INHIBITORI RAF KINAZE
EP1158985B1 (en) 1999-01-13 2011-12-28 Bayer HealthCare LLC OMEGA-CARBOXY ARYL SUBSTITUTED DIPHENYL UREAS AS p38 KINASE INHIBITORS
US8124630B2 (en) 1999-01-13 2012-02-28 Bayer Healthcare Llc ω-carboxyaryl substituted diphenyl ureas as raf kinase inhibitors
SI1478358T1 (sl) 2002-02-11 2013-09-30 Bayer Healthcare Llc Sorafenib tozilat za zdravljenje bolezni, značilnih po abnormalni angiogenezi
WO2003068229A1 (en) 2002-02-11 2003-08-21 Bayer Pharmaceuticals Corporation Pyridine, quinoline, and isoquinoline n-oxides as kinase inhibitors
CA2413475C (en) 2002-04-25 2010-07-27 The Government Of The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services Zap-70 expression as a marker for chronic lymphocytic leukemia/small lymphocytic lymphoma (cll/sll)
AU2003262642B2 (en) * 2002-08-14 2010-06-17 Vertex Pharmaceuticals Incorporated Protein kinase inhibitors and uses thereof
RU2351590C2 (ru) 2003-02-10 2009-04-10 Вертекс Фармасьютикалз Инкорпорейтед Способ получения диариламина
EP1636585B2 (en) 2003-05-20 2012-06-13 Bayer HealthCare LLC Diaryl ureas with kinase inhibiting activity
EP1663978B1 (en) 2003-07-23 2007-11-28 Bayer Pharmaceuticals Corporation Fluoro substituted omega-carboxyaryl diphenyl urea for the treatment and prevention of diseases and conditions
EP2295426A1 (en) 2004-04-30 2011-03-16 Bayer HealthCare, LLC Substituted pyrazolyl urea derivatives useful in the treatment of cancer
WO2006021848A1 (en) * 2004-08-27 2006-03-02 Ranbaxy Laboratories Limited Anti-inflammatory agents
US20100104536A1 (en) * 2007-03-20 2010-04-29 Indravadan Ambalal Modi P38 inhibitors
GB0908317D0 (en) * 2009-05-14 2009-06-24 Argenta Discovery Ltd Pharmaceutical compounds and compositions
US9556426B2 (en) 2009-09-16 2017-01-31 Celgene Avilomics Research, Inc. Protein kinase conjugates and inhibitors
ES2897740T3 (es) 2011-12-28 2022-03-02 Kyoto Prefectural Public Univ Corp Normalización del cultivo de células endoteliales de la córnea
WO2015072580A1 (ja) 2013-11-14 2015-05-21 学校法人同志社 細胞増殖促進または細胞障害抑制による角膜内皮治療薬
EP4096647A1 (en) * 2020-01-30 2022-12-07 Yeda Research and Development Co. Ltd Treating acute liver disease with tlr-mik inhibitors
EP4146196A4 (en) * 2020-05-08 2024-06-26 Georgiamune Inc. AKT3 MODULATORS AND METHODS OF USE THEREOF

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6608060B1 (en) 1996-12-18 2003-08-19 Vertex Pharmaceuticals Incorporated Inhibitors of p38
US6147080A (en) * 1996-12-18 2000-11-14 Vertex Pharmaceuticals Incorporated Inhibitors of p38
US5945418A (en) 1996-12-18 1999-08-31 Vertex Pharmaceuticals Incorporated Inhibitors of p38
MY132496A (en) * 1998-05-11 2007-10-31 Vertex Pharma Inhibitors of p38
AR023659A1 (es) 1998-09-18 2002-09-04 Vertex Pharma Un compuesto inhibidor de p38, una composicion farmaceutica que lo comprende y el uso de dicha composicion en el tratamiento y prevencion de estados patologicos
AU2001247700A1 (en) * 2000-03-22 2001-10-03 Vertex Pharmaceuticals Incorporated Inhibitors of p38

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