JP2004506042A5 - - Google Patents

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Publication number
JP2004506042A5
JP2004506042A5 JP2002519424A JP2002519424A JP2004506042A5 JP 2004506042 A5 JP2004506042 A5 JP 2004506042A5 JP 2002519424 A JP2002519424 A JP 2002519424A JP 2002519424 A JP2002519424 A JP 2002519424A JP 2004506042 A5 JP2004506042 A5 JP 2004506042A5
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JP
Japan
Prior art keywords
independently selected
embedded image
disease
compound
aromatic
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2002519424A
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English (en)
Japanese (ja)
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JP2004506042A (ja
JP4993838B2 (ja
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Publication date
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Priority claimed from PCT/US2001/025015 external-priority patent/WO2002014281A1/en
Publication of JP2004506042A publication Critical patent/JP2004506042A/ja
Publication of JP2004506042A5 publication Critical patent/JP2004506042A5/ja
Application granted granted Critical
Publication of JP4993838B2 publication Critical patent/JP4993838B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2002519424A 2000-08-11 2001-08-10 P38のインヒビターとしてのピリジン誘導体 Expired - Fee Related JP4993838B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US22471900P 2000-08-11 2000-08-11
US60/224,719 2000-08-11
PCT/US2001/025015 WO2002014281A1 (en) 2000-08-11 2001-08-10 Pyridine derivatives as inhibitors of p38

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2012077626A Division JP2012149085A (ja) 2000-08-11 2012-03-29 P38のインヒビターとしてのピリジン誘導体

Publications (3)

Publication Number Publication Date
JP2004506042A JP2004506042A (ja) 2004-02-26
JP2004506042A5 true JP2004506042A5 (https=) 2008-10-02
JP4993838B2 JP4993838B2 (ja) 2012-08-08

Family

ID=22841879

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2002519424A Expired - Fee Related JP4993838B2 (ja) 2000-08-11 2001-08-10 P38のインヒビターとしてのピリジン誘導体
JP2012077626A Withdrawn JP2012149085A (ja) 2000-08-11 2012-03-29 P38のインヒビターとしてのピリジン誘導体

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2012077626A Withdrawn JP2012149085A (ja) 2000-08-11 2012-03-29 P38のインヒビターとしてのピリジン誘導体

Country Status (7)

Country Link
US (4) US7186737B2 (https=)
EP (1) EP1309560B1 (https=)
JP (2) JP4993838B2 (https=)
AU (2) AU2001283237B2 (https=)
CA (1) CA2418389A1 (https=)
MX (1) MXPA03001256A (https=)
WO (1) WO2002014281A1 (https=)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR023659A1 (es) * 1998-09-18 2002-09-04 Vertex Pharma Un compuesto inhibidor de p38, una composicion farmaceutica que lo comprende y el uso de dicha composicion en el tratamiento y prevencion de estados patologicos
ATE538794T1 (de) 1999-01-13 2012-01-15 Bayer Healthcare Llc Gamma carboxyarylsubstituierte diphenylharnstoffverbindungen als p38 kinasehemmer
US7351834B1 (en) 1999-01-13 2008-04-01 Bayer Pharmaceuticals Corporation ω-Carboxyaryl substituted diphenyl ureas as raf kinase inhibitors
US8124630B2 (en) 1999-01-13 2012-02-28 Bayer Healthcare Llc ω-carboxyaryl substituted diphenyl ureas as raf kinase inhibitors
WO2003068229A1 (en) 2002-02-11 2003-08-21 Bayer Pharmaceuticals Corporation Pyridine, quinoline, and isoquinoline n-oxides as kinase inhibitors
MXPA04007832A (es) 2002-02-11 2005-09-08 Bayer Pharmaceuticals Corp Aril-ureas con actividad inhibitoria de angiogenesis.
US7329502B2 (en) 2002-04-25 2008-02-12 The United States Of America As Represented By The Department Of Health And Human Services ZAP-70 expression as a marker for chronic lymphocytic leukemia/small lymphocytic lymphoma (CLL/SLL)
MXPA05001804A (es) * 2002-08-14 2005-05-27 Vertex Pharma Inhibidores de proteinas cinasas y usos de los mismos.
CN101723891A (zh) * 2003-02-10 2010-06-09 沃泰克斯药物股份有限公司 通过使n-芳基氨基甲酸酯与卤代杂芳基反应制备n-杂芳基-n-芳基胺的方法和类似方法
WO2004113274A2 (en) 2003-05-20 2004-12-29 Bayer Pharmaceuticals Corporation Diaryl ureas with kinase inhibiting activity
EA010485B1 (ru) 2003-07-23 2008-10-30 Байер Фамэсьютиклс Копэрейшн Производное n,n'-дифенилмочевины, фармацевтическая композиция (варианты) и способ лечения и предупреждения заболеваний и состояний с его использованием (варианты)
CN101010315A (zh) 2004-04-30 2007-08-01 拜耳制药公司 用于治疗癌症的取代的吡唑基脲衍生物
WO2006021848A1 (en) * 2004-08-27 2006-03-02 Ranbaxy Laboratories Limited Anti-inflammatory agents
CA2681420A1 (en) * 2007-03-20 2008-09-25 Cadila Pharmaceuticals Limited P38 inhibitors
GB0908317D0 (en) * 2009-05-14 2009-06-24 Argenta Discovery Ltd Pharmaceutical compounds and compositions
NZ620174A (en) * 2009-09-16 2016-08-26 Celgene Avilomics Res Inc Protein kinase conjugates and inhibitors
EP2799537B1 (en) 2011-12-28 2021-09-22 Kyoto Prefectural Public University Corporation Normalization of culture of corneal endothelial cells
WO2015072580A1 (ja) 2013-11-14 2015-05-21 学校法人同志社 細胞増殖促進または細胞障害抑制による角膜内皮治療薬
WO2021152587A1 (en) * 2020-01-30 2021-08-05 Yeda Research And Development Co. Ltd. Treating acute liver disease with tlr-mik inhibitors
AU2021269065A1 (en) * 2020-05-08 2022-12-15 Georgiamune, Inc. Akt3 modulators and methods of use thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6147080A (en) * 1996-12-18 2000-11-14 Vertex Pharmaceuticals Incorporated Inhibitors of p38
US6608060B1 (en) * 1996-12-18 2003-08-19 Vertex Pharmaceuticals Incorporated Inhibitors of p38
US5945418A (en) * 1996-12-18 1999-08-31 Vertex Pharmaceuticals Incorporated Inhibitors of p38
MY132496A (en) * 1998-05-11 2007-10-31 Vertex Pharma Inhibitors of p38
AR023659A1 (es) * 1998-09-18 2002-09-04 Vertex Pharma Un compuesto inhibidor de p38, una composicion farmaceutica que lo comprende y el uso de dicha composicion en el tratamiento y prevencion de estados patologicos
CA2403828A1 (en) * 2000-03-22 2001-09-27 Vertex Pharmaceuticals Incorporated Inhibitors of p38

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