AU2001283237B2 - Pyridine derivatives as inhibitors of p38 - Google Patents
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- AU2001283237B2 AU2001283237B2 AU2001283237A AU2001283237A AU2001283237B2 AU 2001283237 B2 AU2001283237 B2 AU 2001283237B2 AU 2001283237 A AU2001283237 A AU 2001283237A AU 2001283237 A AU2001283237 A AU 2001283237A AU 2001283237 B2 AU2001283237 B2 AU 2001283237B2
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Classifications
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Landscapes
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Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AU2007249154A AU2007249154A1 (en) | 2000-08-11 | 2007-12-20 | Pyridine Derivatives as Inhibitors of p38 |
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| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US22471900P | 2000-08-11 | 2000-08-11 | |
| US60/224,719 | 2000-08-11 | ||
| PCT/US2001/025015 WO2002014281A1 (en) | 2000-08-11 | 2001-08-10 | Pyridine derivatives as inhibitors of p38 |
Related Child Applications (1)
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|---|---|---|---|
| AU2007249154A Division AU2007249154A1 (en) | 2000-08-11 | 2007-12-20 | Pyridine Derivatives as Inhibitors of p38 |
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| AU2001283237A1 AU2001283237A1 (en) | 2002-05-23 |
| AU2001283237B2 true AU2001283237B2 (en) | 2007-09-20 |
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| AU8323701A Pending AU8323701A (en) | 2000-08-11 | 2001-08-10 | Inhibitors of p38 |
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| Application Number | Title | Priority Date | Filing Date |
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| AU8323701A Pending AU8323701A (en) | 2000-08-11 | 2001-08-10 | Inhibitors of p38 |
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| EP (1) | EP1309560B1 (https=) |
| JP (2) | JP4993838B2 (https=) |
| AU (2) | AU2001283237B2 (https=) |
| CA (1) | CA2418389A1 (https=) |
| MX (1) | MXPA03001256A (https=) |
| WO (1) | WO2002014281A1 (https=) |
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| AR023659A1 (es) * | 1998-09-18 | 2002-09-04 | Vertex Pharma | Un compuesto inhibidor de p38, una composicion farmaceutica que lo comprende y el uso de dicha composicion en el tratamiento y prevencion de estados patologicos |
| ATE538794T1 (de) | 1999-01-13 | 2012-01-15 | Bayer Healthcare Llc | Gamma carboxyarylsubstituierte diphenylharnstoffverbindungen als p38 kinasehemmer |
| US7351834B1 (en) | 1999-01-13 | 2008-04-01 | Bayer Pharmaceuticals Corporation | ω-Carboxyaryl substituted diphenyl ureas as raf kinase inhibitors |
| US8124630B2 (en) | 1999-01-13 | 2012-02-28 | Bayer Healthcare Llc | ω-carboxyaryl substituted diphenyl ureas as raf kinase inhibitors |
| WO2003068229A1 (en) | 2002-02-11 | 2003-08-21 | Bayer Pharmaceuticals Corporation | Pyridine, quinoline, and isoquinoline n-oxides as kinase inhibitors |
| MXPA04007832A (es) | 2002-02-11 | 2005-09-08 | Bayer Pharmaceuticals Corp | Aril-ureas con actividad inhibitoria de angiogenesis. |
| US7329502B2 (en) | 2002-04-25 | 2008-02-12 | The United States Of America As Represented By The Department Of Health And Human Services | ZAP-70 expression as a marker for chronic lymphocytic leukemia/small lymphocytic lymphoma (CLL/SLL) |
| MXPA05001804A (es) * | 2002-08-14 | 2005-05-27 | Vertex Pharma | Inhibidores de proteinas cinasas y usos de los mismos. |
| CN101723891A (zh) * | 2003-02-10 | 2010-06-09 | 沃泰克斯药物股份有限公司 | 通过使n-芳基氨基甲酸酯与卤代杂芳基反应制备n-杂芳基-n-芳基胺的方法和类似方法 |
| WO2004113274A2 (en) | 2003-05-20 | 2004-12-29 | Bayer Pharmaceuticals Corporation | Diaryl ureas with kinase inhibiting activity |
| EA010485B1 (ru) | 2003-07-23 | 2008-10-30 | Байер Фамэсьютиклс Копэрейшн | Производное n,n'-дифенилмочевины, фармацевтическая композиция (варианты) и способ лечения и предупреждения заболеваний и состояний с его использованием (варианты) |
| CN101010315A (zh) | 2004-04-30 | 2007-08-01 | 拜耳制药公司 | 用于治疗癌症的取代的吡唑基脲衍生物 |
| WO2006021848A1 (en) * | 2004-08-27 | 2006-03-02 | Ranbaxy Laboratories Limited | Anti-inflammatory agents |
| CA2681420A1 (en) * | 2007-03-20 | 2008-09-25 | Cadila Pharmaceuticals Limited | P38 inhibitors |
| GB0908317D0 (en) * | 2009-05-14 | 2009-06-24 | Argenta Discovery Ltd | Pharmaceutical compounds and compositions |
| NZ620174A (en) * | 2009-09-16 | 2016-08-26 | Celgene Avilomics Res Inc | Protein kinase conjugates and inhibitors |
| EP2799537B1 (en) | 2011-12-28 | 2021-09-22 | Kyoto Prefectural Public University Corporation | Normalization of culture of corneal endothelial cells |
| WO2015072580A1 (ja) | 2013-11-14 | 2015-05-21 | 学校法人同志社 | 細胞増殖促進または細胞障害抑制による角膜内皮治療薬 |
| WO2021152587A1 (en) * | 2020-01-30 | 2021-08-05 | Yeda Research And Development Co. Ltd. | Treating acute liver disease with tlr-mik inhibitors |
| AU2021269065A1 (en) * | 2020-05-08 | 2022-12-15 | Georgiamune, Inc. | Akt3 modulators and methods of use thereof |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1999058502A1 (en) * | 1998-05-11 | 1999-11-18 | Vertex Pharmaceuticals Incorporated | Heterocyclic inhibitors of p38 |
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|---|---|---|---|---|
| US6147080A (en) * | 1996-12-18 | 2000-11-14 | Vertex Pharmaceuticals Incorporated | Inhibitors of p38 |
| US6608060B1 (en) * | 1996-12-18 | 2003-08-19 | Vertex Pharmaceuticals Incorporated | Inhibitors of p38 |
| US5945418A (en) * | 1996-12-18 | 1999-08-31 | Vertex Pharmaceuticals Incorporated | Inhibitors of p38 |
| AR023659A1 (es) * | 1998-09-18 | 2002-09-04 | Vertex Pharma | Un compuesto inhibidor de p38, una composicion farmaceutica que lo comprende y el uso de dicha composicion en el tratamiento y prevencion de estados patologicos |
| CA2403828A1 (en) * | 2000-03-22 | 2001-09-27 | Vertex Pharmaceuticals Incorporated | Inhibitors of p38 |
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2001
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- 2001-08-10 WO PCT/US2001/025015 patent/WO2002014281A1/en not_active Ceased
- 2001-08-10 CA CA002418389A patent/CA2418389A1/en not_active Abandoned
- 2001-08-10 AU AU2001283237A patent/AU2001283237B2/en not_active Ceased
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- 2001-08-10 EP EP01962021A patent/EP1309560B1/en not_active Expired - Lifetime
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2003
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2011
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Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1999058502A1 (en) * | 1998-05-11 | 1999-11-18 | Vertex Pharmaceuticals Incorporated | Heterocyclic inhibitors of p38 |
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| EP1309560A1 (en) | 2003-05-14 |
| WO2002014281A8 (en) | 2002-04-04 |
| EP1309560B1 (en) | 2012-10-03 |
| WO2002014281A1 (en) | 2002-02-21 |
| US7186737B2 (en) | 2007-03-06 |
| JP2004506042A (ja) | 2004-02-26 |
| US20110160163A1 (en) | 2011-06-30 |
| US20090318452A1 (en) | 2009-12-24 |
| US7919513B2 (en) | 2011-04-05 |
| MXPA03001256A (es) | 2004-12-06 |
| US7598277B2 (en) | 2009-10-06 |
| US20040044002A1 (en) | 2004-03-04 |
| JP2012149085A (ja) | 2012-08-09 |
| JP4993838B2 (ja) | 2012-08-08 |
| US20070142334A1 (en) | 2007-06-21 |
| AU8323701A (en) | 2002-02-25 |
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