JP2003535864A5 - - Google Patents

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Publication number
JP2003535864A5
JP2003535864A5 JP2002501899A JP2002501899A JP2003535864A5 JP 2003535864 A5 JP2003535864 A5 JP 2003535864A5 JP 2002501899 A JP2002501899 A JP 2002501899A JP 2002501899 A JP2002501899 A JP 2002501899A JP 2003535864 A5 JP2003535864 A5 JP 2003535864A5
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JP
Japan
Prior art keywords
group
hydroxy
unsubstituted
alkylamino
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2002501899A
Other languages
English (en)
Japanese (ja)
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JP2003535864A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/EP2001/006306 external-priority patent/WO2001094350A1/en
Publication of JP2003535864A publication Critical patent/JP2003535864A/ja
Publication of JP2003535864A5 publication Critical patent/JP2003535864A5/ja
Withdrawn legal-status Critical Current

Links

JP2002501899A 2000-06-07 2001-06-01 6−フェニルピロロピリミジンジオン誘導体 Withdrawn JP2003535864A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
ES200001436 2000-06-07
ES200001436 2000-06-07
PCT/EP2001/006306 WO2001094350A1 (en) 2000-06-07 2001-06-01 6-phenylpyrrolopyrimidinedione derivatives

Publications (2)

Publication Number Publication Date
JP2003535864A JP2003535864A (ja) 2003-12-02
JP2003535864A5 true JP2003535864A5 (cg-RX-API-DMAC7.html) 2008-07-17

Family

ID=8493813

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002501899A Withdrawn JP2003535864A (ja) 2000-06-07 2001-06-01 6−フェニルピロロピリミジンジオン誘導体

Country Status (12)

Country Link
US (1) US6943253B2 (cg-RX-API-DMAC7.html)
EP (1) EP1286997B1 (cg-RX-API-DMAC7.html)
JP (1) JP2003535864A (cg-RX-API-DMAC7.html)
AR (1) AR030424A1 (cg-RX-API-DMAC7.html)
AT (1) ATE273980T1 (cg-RX-API-DMAC7.html)
AU (1) AU2001281802A1 (cg-RX-API-DMAC7.html)
CA (1) CA2411013A1 (cg-RX-API-DMAC7.html)
DE (1) DE60105020T2 (cg-RX-API-DMAC7.html)
ES (1) ES2222389T3 (cg-RX-API-DMAC7.html)
MY (1) MY133995A (cg-RX-API-DMAC7.html)
PE (1) PE20020219A1 (cg-RX-API-DMAC7.html)
WO (1) WO2001094350A1 (cg-RX-API-DMAC7.html)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2193839B1 (es) * 2001-06-22 2005-02-16 Almirall Prodesfarma, S.A. Nuevos derivados de 6-fenildihidropirrolpirimidindiona.
ES2208063B1 (es) 2002-04-01 2005-10-01 Almirall Prodesfarma, S.A. Nuevos derivados de la 4-(pirrolopirimidin-6-il)bencenosulfonamida.
DE10229778A1 (de) * 2002-07-03 2004-01-29 Bayer Ag Neue Verwendung von Imidazotriazinonen
PL1644021T3 (pl) * 2003-06-13 2013-01-31 Ironwood Pharmaceuticals Inc Sposoby i kompozycje do leczenia zaburzeń żołądkowo-jelitowych
US7449473B2 (en) 2003-10-31 2008-11-11 Cv Therapeutics, Inc. Substituted pyrrolo[3,2-d]pyrimidin-2,4-diones as A2b adenosine receptor antagonists
EP2275096A3 (en) 2005-08-26 2011-07-13 Braincells, Inc. Neurogenesis via modulation of the muscarinic receptors
EP2258358A3 (en) 2005-08-26 2011-09-07 Braincells, Inc. Neurogenesis with acetylcholinesterase inhibitor
AU2006304787A1 (en) 2005-10-21 2007-04-26 Braincells, Inc. Modulation of neurogenesis by PDE inhibition
CA2625210A1 (en) 2005-10-31 2007-05-10 Braincells, Inc. Gaba receptor mediated modulation of neurogenesis
US20100216734A1 (en) 2006-03-08 2010-08-26 Braincells, Inc. Modulation of neurogenesis by nootropic agents
AU2007249399A1 (en) 2006-05-09 2007-11-22 Braincells, Inc. Neurogenesis by modulating angiotensin
AU2007249435A1 (en) 2006-05-09 2007-11-22 Braincells, Inc. 5 HT receptor mediated neurogenesis
BRPI0716604A2 (pt) 2006-09-08 2013-04-09 Braincells Inc combinaÇÕes contendo um derivado de 4-acilaminopiridina
US20100184806A1 (en) 2006-09-19 2010-07-22 Braincells, Inc. Modulation of neurogenesis by ppar agents
US20100216805A1 (en) 2009-02-25 2010-08-26 Braincells, Inc. Modulation of neurogenesis using d-cycloserine combinations
AR077898A1 (es) * 2009-08-26 2011-09-28 Nycomed Gmbh Metilpirrolopirimidincarboxamidas
AR079451A1 (es) 2009-12-18 2012-01-25 Nycomed Gmbh Compuestos 3,4,4a,10b-tetrahidro-1h-tiopirano[4,3-c]isoquinolina
AT512084A1 (de) * 2011-10-20 2013-05-15 Univ Wien Tech Diazabicyclo- und diazaspiro-alkanderivate als phosphodiesterase-5 inhibitoren
WO2013106547A1 (en) 2012-01-10 2013-07-18 President And Fellows Of Harvard College Beta-cell replication promoting compounds and methods of their use
TWI698436B (zh) 2014-12-30 2020-07-11 美商佛瑪治療公司 作為泛素特異性蛋白酶7抑制劑之吡咯并及吡唑并嘧啶
MA41291A (fr) 2014-12-30 2017-11-07 Forma Therapeutics Inc Dérivés de la pyrrolotriazinone et de l'imidazotriazinone en tant qu'inhibiteurs de la protéase spécifique de l'ubiquitine n° 7 (usp7) pour le traitement d'un cancer
US9932351B2 (en) 2015-02-05 2018-04-03 Forma Therapeutics, Inc. Thienopyrimidinones as ubiquitin-specific protease 7 inhibitors
JP2018504430A (ja) 2015-02-05 2018-02-15 フォーマ セラピューティクス,インコーポレイテッド ユビキチン特異的プロテアーゼ7阻害物質としてのキナゾリノン及びアザキナゾリノン
US9938300B2 (en) 2015-02-05 2018-04-10 Forma Therapeutics, Inc. Isothiazolopyrimidinones, pyrazolopyrimidinones, and pyrrolopyrimidinones as ubiquitin-specific protease 7 inhibitors

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5260322A (en) 1990-10-08 1993-11-09 Merck & Co., Inc. Angiotension II antagonists in the treatment of hyperuricemia
FR2737494B1 (fr) * 1995-08-04 1997-08-29 Synthelabo Derives de benzenesulfonamide, leur preparation et leur application en therapeutique
AU4501199A (en) * 1998-06-03 1999-12-20 Almirall Prodesfarma S.A. 8-phenylxanthine derivatives and their use as phosphodiesterase inhibitors

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