JP2003531119A5 - - Google Patents

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Publication number
JP2003531119A5
JP2003531119A5 JP2001572528A JP2001572528A JP2003531119A5 JP 2003531119 A5 JP2003531119 A5 JP 2003531119A5 JP 2001572528 A JP2001572528 A JP 2001572528A JP 2001572528 A JP2001572528 A JP 2001572528A JP 2003531119 A5 JP2003531119 A5 JP 2003531119A5
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JP
Japan
Prior art keywords
compound
embedded image
providing
dimethyl
chemical
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JP2001572528A
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English (en)
Japanese (ja)
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JP4845320B2 (ja
JP2003531119A (ja
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Priority claimed from PCT/US2001/010293 external-priority patent/WO2001074839A2/en
Publication of JP2003531119A publication Critical patent/JP2003531119A/ja
Publication of JP2003531119A5 publication Critical patent/JP2003531119A5/ja
Application granted granted Critical
Publication of JP4845320B2 publication Critical patent/JP4845320B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2001572528A 2000-03-31 2001-03-30 (7α,11β)−ジメチル−17β−ヒドロキシ−4−エストレン−3−オンの4−N−ブチルシクロヘキサン酸エステル及びウンデカン酸エステルの製造方法及びそれらの医学用途 Expired - Fee Related JP4845320B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US19353000P 2000-03-31 2000-03-31
US60/193,530 2000-03-31
US19444000P 2000-04-04 2000-04-04
US60/194,440 2000-04-04
PCT/US2001/010293 WO2001074839A2 (en) 2000-03-31 2001-03-30 Methods of making the 4-n-butylcyclohexanoic and the undecanoic acid esters of (7 alpha, 11 beta)-dimethyl-17 beta-hydroxy-4-estren-3-one and their medical use

Publications (3)

Publication Number Publication Date
JP2003531119A JP2003531119A (ja) 2003-10-21
JP2003531119A5 true JP2003531119A5 (https=) 2008-05-01
JP4845320B2 JP4845320B2 (ja) 2011-12-28

Family

ID=26889099

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2001572528A Expired - Fee Related JP4845320B2 (ja) 2000-03-31 2001-03-30 (7α,11β)−ジメチル−17β−ヒドロキシ−4−エストレン−3−オンの4−N−ブチルシクロヘキサン酸エステル及びウンデカン酸エステルの製造方法及びそれらの医学用途

Country Status (8)

Country Link
US (1) US7196074B2 (https=)
EP (1) EP1272196B1 (https=)
JP (1) JP4845320B2 (https=)
AT (1) ATE334682T1 (https=)
AU (2) AU2001249661B2 (https=)
CA (1) CA2402524C (https=)
DE (1) DE60121928T2 (https=)
WO (1) WO2001074839A2 (https=)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5952319A (en) 1997-11-26 1999-09-14 Research Triangle Institute Androgenic steroid compounds and a method of making and using the same
US20030069215A1 (en) * 2001-03-30 2003-04-10 The Government Of The United States Of America, Methods of making and using 7a,11b-dimethyl-17b-hydroxy-4-estren-3-one 17b-trans-4-n-butylcyclohexane carboxylate and 7a,11b-dimethyl-17b-hydroxyestr-4-en-3-one 17-undecanoate
GB0025221D0 (en) * 2000-10-14 2000-11-29 Astrazeneca Ab New process
AU2006211907B2 (en) * 2005-02-04 2011-09-08 Government Of The United States Of America, Represented By The Secretary, Department Of Health And Human Services Nandrolone 17beta-carbonates
WO2008039482A2 (en) * 2006-09-26 2008-04-03 The Regents Of The University Of California Methods and compositions for cancer prevention and treatment
US9517240B2 (en) 2006-09-26 2016-12-13 The Regents Of The University Of California Methods and compositions for cancer prevention and treatment
BR112014012444B1 (pt) 2011-11-23 2021-12-14 Therapeuticsmd, Inc Composição farmacêutica compreendendo estradiol solubilizado, progesterona e um agente de solubilização, bem como usos desta para tratar um sintoma relacionado à menopausa em uma mulher
US9301920B2 (en) 2012-06-18 2016-04-05 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
US10806740B2 (en) 2012-06-18 2020-10-20 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
US20150196640A1 (en) 2012-06-18 2015-07-16 Therapeuticsmd, Inc. Progesterone formulations having a desirable pk profile
US20130338122A1 (en) 2012-06-18 2013-12-19 Therapeuticsmd, Inc. Transdermal hormone replacement therapies
US10806697B2 (en) 2012-12-21 2020-10-20 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US9180091B2 (en) 2012-12-21 2015-11-10 Therapeuticsmd, Inc. Soluble estradiol capsule for vaginal insertion
US10568891B2 (en) 2012-12-21 2020-02-25 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10471072B2 (en) 2012-12-21 2019-11-12 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10537581B2 (en) 2012-12-21 2020-01-21 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US11266661B2 (en) 2012-12-21 2022-03-08 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US11246875B2 (en) 2012-12-21 2022-02-15 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10050658B2 (en) 2014-02-24 2018-08-14 National Products, Inc. Docking sleeve with electrical adapter
RU2016143081A (ru) 2014-05-22 2018-06-26 Терапьютиксмд, Инк. Натуральные комбинированные гормонозаместительные составы и терапии
US10328087B2 (en) 2015-07-23 2019-06-25 Therapeuticsmd, Inc. Formulations for solubilizing hormones
US10286077B2 (en) 2016-04-01 2019-05-14 Therapeuticsmd, Inc. Steroid hormone compositions in medium chain oils
US9931349B2 (en) 2016-04-01 2018-04-03 Therapeuticsmd, Inc. Steroid hormone pharmaceutical composition
US11633405B2 (en) 2020-02-07 2023-04-25 Therapeuticsmd, Inc. Steroid hormone pharmaceutical formulations
US20230227492A1 (en) * 2020-06-11 2023-07-20 The Usa As Represented By The Secretary, Department Of Health And Human Services Monomeric and oligomeric compound embodiments as contraceptives and therapies and methods of making and using the same

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2837517A (en) * 1955-08-08 1958-06-03 Upjohn Co 9, 11beta-epoxy-17-alkyltestosterones
US3160644A (en) * 1955-08-08 1964-12-08 Upjohn Co 1-dehydro-11-keto-9alpha-fluoro-17alpha-methyl testosterones
US2806863A (en) * 1956-03-19 1957-09-17 Upjohn Co 9alpha-halo-11beta, 17beta-dihydroxy-17alpha-methylandrostane-3-ones
US3438783A (en) * 1965-08-16 1969-04-15 Monsanto Co Improving egg quality in poultry by orally administering androgens
US3577410A (en) 1968-07-30 1971-05-04 American Home Prod 13beta-alkyl-17-hydroxygona-4,14-dien-3-ones
DE2031849C3 (de) 1970-06-27 1978-11-16 Bosch Gmbh Robert Flüssigkeitsdichte Verbindung eines Deckels aus thermoplastischem Material mit einem Kasten aus thermoplastischem Material
ZA712312B (en) 1970-04-28 1972-01-26 Ochsner Med Found Alton 4,14-estradiene compounds
IL36628A (en) 1970-04-28 1978-08-31 Ochsner Med Found Alton 4, 14-estradiene compounds and processes for their preparation
ES2053714T3 (es) * 1987-12-12 1994-08-01 Akzo Nv Proceso para la preparacion de 11-arilesteroides.
FR2747680B1 (fr) * 1996-04-18 1998-07-03 Roussel Uclaf Nouveaux steroides, leur application a titre de medicaments, leur procede de preparation, les intermediaires de ce procede et les compositions pharmaceutiques les renfermant
DE19619045C1 (de) 1996-05-02 1997-11-13 Jenapharm Gmbh Verwendung von Kombinationspräparaten zur Behandlung hypogonadaler Männer sowie Männern mit Hypophysenerkrankungen
US5952319A (en) * 1997-11-26 1999-09-14 Research Triangle Institute Androgenic steroid compounds and a method of making and using the same
TW548277B (en) 1999-07-16 2003-08-21 Akzo Nobel Nv Orally active androgens

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