JP2003525302A - Ｉｌ−８受容体アンタゴニスト - Google Patents
Ｉｌ−８受容体アンタゴニストInfo
- Publication number
- JP2003525302A JP2003525302A JP2001564187A JP2001564187A JP2003525302A JP 2003525302 A JP2003525302 A JP 2003525302A JP 2001564187 A JP2001564187 A JP 2001564187A JP 2001564187 A JP2001564187 A JP 2001564187A JP 2003525302 A JP2003525302 A JP 2003525302A
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- aryl
- heteroaryl
- heterocyclic
- alkenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US18618200P | 2000-03-01 | 2000-03-01 | |
| US60/186,182 | 2000-03-01 | ||
| PCT/US2001/006555 WO2001064691A1 (fr) | 2000-03-01 | 2001-03-01 | Antagonistes du recepteur de l'interleukine 8 (il-8) |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JP2003525302A true JP2003525302A (ja) | 2003-08-26 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| JP2001564187A Withdrawn JP2003525302A (ja) | 2000-03-01 | 2001-03-01 | Ｉｌ−８受容体アンタゴニスト |
Country Status (4)
| Country | Link |
|---|---|
| EP (1) | EP1265905A4 (fr) |
| JP (1) | JP2003525302A (fr) |
| AU (1) | AU2001243351A1 (fr) |
| WO (1) | WO2001064691A1 (fr) |
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|---|---|---|---|---|
| US20040106794A1 (en) | 2001-04-16 | 2004-06-03 | Schering Corporation | 3,4-Di-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands |
| US7132445B2 (en) | 2001-04-16 | 2006-11-07 | Schering Corporation | 3,4-Di-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands |
| CA2462862A1 (fr) | 2001-10-12 | 2003-04-17 | Schering Corporation | Composes de maleimide di-substitues en 3,4, antagonistes du recepteur de la cxc-chimiokine |
| US6878709B2 (en) | 2002-01-04 | 2005-04-12 | Schering Corporation | 3,4-di-substituted pyridazinediones as CXC chemokine receptor antagonists |
| MXPA04009127A (es) | 2002-03-18 | 2005-01-25 | Schering Corp | Tratamiento de enfermedades mediadas por quimiocinas. |
| PE20040570A1 (es) | 2002-10-09 | 2004-08-30 | Pharmacopeia Drug Discovery | Tiadiazoldioxidos y tiadiazoloxidos como ligandos del receptor de cxc- y cc-quimiocina |
| MXPA06007076A (es) | 2003-12-19 | 2006-08-31 | Pharmacopeia Drug Discovery | Tiadiazoles como ligandos del receptor cxc y cc-quimiocina. |
| MXPA06007205A (es) | 2003-12-22 | 2006-08-31 | Schering Corp | Dioxidos de isotiazol como ligandos del receptor cxc y cc-quimiocina. |
| CN1984899B (zh) | 2004-05-12 | 2011-07-27 | 先灵公司 | Cxcr1和cxcr2趋化因子拮抗剂 |
| MX2008000367A (es) | 2005-06-29 | 2008-03-07 | Schering Corp | Oxidiazolopirazinas y tiadiazolopirazinas 5,6-di-sustituidas como ligandos de receptor de quimiocina en la que dos cisternas son separadas por un solo aminoacido. |
| CN101253165A (zh) | 2005-06-29 | 2008-08-27 | 先灵公司 | 作为cxc－化学活素受体配体的二取代的二唑 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1103785A (fr) * | 1954-05-03 | 1955-11-07 | Rhone Poulenc Sa | Nouveaux dérivés de l'acide phosphorique et leurs procédés de préparation |
| US3957923A (en) * | 1973-06-25 | 1976-05-18 | E. I. Du Pont De Nemours & Company | Alkyl and haloalkyl n,n'-dialkyl-n-methylolphosphorodiamidates |
| US4119716A (en) * | 1977-07-27 | 1978-10-10 | Stauffer Chemical Company | Certain diaryldithiophosphorodiamidates and their use as biocides |
| DE3161413D1 (en) * | 1980-04-30 | 1983-12-22 | Ciba Geigy Ag | N-phenylphosphoramidate esters, process for their preparation and their use as coupling components |
| UY25842A1 (es) * | 1998-12-16 | 2001-04-30 | Smithkline Beecham Corp | Antagonistas de receptores de il-8 |
-
2001
- 2001-03-01 WO PCT/US2001/006555 patent/WO2001064691A1/fr not_active Application Discontinuation
- 2001-03-01 AU AU2001243351A patent/AU2001243351A1/en not_active Abandoned
- 2001-03-01 JP JP2001564187A patent/JP2003525302A/ja not_active Withdrawn
- 2001-03-01 EP EP01916312A patent/EP1265905A4/fr not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| WO2001064691A1 (fr) | 2001-09-07 |
| EP1265905A4 (fr) | 2003-03-12 |
| AU2001243351A1 (en) | 2001-09-12 |
| EP1265905A1 (fr) | 2002-12-18 |
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