JP2002516313A5 - - Google Patents
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- Publication number
- JP2002516313A5 JP2002516313A5 JP2000550831A JP2000550831A JP2002516313A5 JP 2002516313 A5 JP2002516313 A5 JP 2002516313A5 JP 2000550831 A JP2000550831 A JP 2000550831A JP 2000550831 A JP2000550831 A JP 2000550831A JP 2002516313 A5 JP2002516313 A5 JP 2002516313A5
- Authority
- JP
- Japan
- Prior art keywords
- erythro
- carbon atoms
- formula
- embedded image
- salt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 *C(*)[C@@]1NCCCC1 Chemical compound *C(*)[C@@]1NCCCC1 0.000 description 4
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/792,661 US5965734A (en) | 1997-01-31 | 1997-01-31 | Processes and intermediates for preparing 2-substituted piperidine stereoisomers |
| PCT/US1998/010599 WO1999061425A1 (en) | 1997-01-31 | 1998-05-26 | Processes and intermediates for preparing 2-substituted piperidine stereoisomers |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2002516313A JP2002516313A (ja) | 2002-06-04 |
| JP2002516313A5 true JP2002516313A5 (https=) | 2006-01-05 |
| JP4491135B2 JP4491135B2 (ja) | 2010-06-30 |
Family
ID=26794135
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2000550831A Expired - Fee Related JP4491135B2 (ja) | 1997-01-31 | 1998-05-26 | ２−置換ピペリジン立体異性体を製造するための方法及び中間体 |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US5965734A (https=) |
| EP (2) | EP1082307B1 (https=) |
| JP (1) | JP4491135B2 (https=) |
| AT (2) | ATE304531T1 (https=) |
| AU (1) | AU765194B2 (https=) |
| CA (1) | CA2333089C (https=) |
| CY (1) | CY1108818T1 (https=) |
| DE (2) | DE69831611T2 (https=) |
| DK (2) | DK1082307T3 (https=) |
| ES (2) | ES2320012T3 (https=) |
| PT (1) | PT1612207E (https=) |
| WO (1) | WO1999061425A1 (https=) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5922736A (en) * | 1995-12-04 | 1999-07-13 | Celegene Corporation | Chronic, bolus administration of D-threo methylphenidate |
| US5837284A (en) * | 1995-12-04 | 1998-11-17 | Mehta; Atul M. | Delivery of multiple doses of medications |
| US6486177B2 (en) * | 1995-12-04 | 2002-11-26 | Celgene Corporation | Methods for treatment of cognitive and menopausal disorders with D-threo methylphenidate |
| US6962997B1 (en) * | 1997-05-22 | 2005-11-08 | Celgene Corporation | Process and intermediates for resolving piperidyl acetamide steroisomers |
| US6359139B1 (en) * | 2000-11-07 | 2002-03-19 | Celgene Corporation | Methods for production of piperidyl acetamide stereoisomers |
| US20020187192A1 (en) * | 2001-04-30 | 2002-12-12 | Yatindra Joshi | Pharmaceutical composition which reduces or eliminates drug abuse potential |
| US20030073681A1 (en) * | 2001-08-21 | 2003-04-17 | Hauske James R. | 2-substituted piperidines that are ligands for monoamine receptors and transporters |
| US6638533B2 (en) | 2002-01-03 | 2003-10-28 | George Krsek | Pulse dosage formulations of methylphenidate and method to prepare same |
| US20050239830A1 (en) * | 2004-04-26 | 2005-10-27 | Vikram Khetani | Methods of diminishing co-abuse potential |
| CA2591247A1 (en) * | 2004-12-09 | 2006-06-15 | Celgene Corporation | Treatment of patients suffering from a disease having a family history or diagnosis of tics or tourette's syndrome with d-threo methylphenidate |
| ITMI20042415A1 (it) * | 2004-12-17 | 2005-03-17 | Clariant Lsm Italia Spa | Sintesi di alfa-aril-alfa-piperid-2-il-acetammidi e loro idrolisi acida |
| US9233924B2 (en) | 2014-03-11 | 2016-01-12 | Ampac Fine Chemicals Llc | Methods for preparing D-threo methylphenidate using diazomethane, and compositions thereof |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2507631A (en) * | 1944-01-19 | 1950-05-16 | Ciba Pharm Prod Inc | Pyridine and piperidine compounds and process of making same |
| US2957880A (en) * | 1953-12-23 | 1960-10-25 | Ciba Pharm Prod Inc | Process for the conversion of stereoisomers |
| JPS5630978A (en) * | 1979-08-24 | 1981-03-28 | Kyowa Hakko Kogyo Co Ltd | Novel mitomycin and its preparation |
| US4978744A (en) * | 1989-01-27 | 1990-12-18 | Arizona Board Of Regents | Synthesis of dolastatin 10 |
| US5075315A (en) * | 1990-05-17 | 1991-12-24 | Mcneilab, Inc. | Antipsychotic hexahydro-2H-indeno[1,2-c]pyridine derivatives |
| AU670939B2 (en) * | 1992-03-16 | 1996-08-08 | Merck Sharp & Dohme Limited | Benzodiazepine derivatives, compositions containing them and their use in therapy |
| AU681924B2 (en) * | 1993-11-22 | 1997-09-11 | Merck & Co., Inc. | 3-acylaminobenzazepines |
| DK0771789T3 (da) * | 1995-10-30 | 2000-06-13 | Hoffmann La Roche | 1 alpha, 26-dihydroxy-D-homo-vitamin D3 |
| DE19615119A1 (de) * | 1996-04-17 | 1997-10-23 | Bayer Ag | Neue Arylessigsäureamide |
-
1997
- 1997-01-31 US US08/792,661 patent/US5965734A/en not_active Expired - Lifetime
-
1998
- 1998-05-26 DK DK98923727T patent/DK1082307T3/da active
- 1998-05-26 PT PT05077084T patent/PT1612207E/pt unknown
- 1998-05-26 JP JP2000550831A patent/JP4491135B2/ja not_active Expired - Fee Related
- 1998-05-26 DE DE69831611T patent/DE69831611T2/de not_active Expired - Lifetime
- 1998-05-26 AT AT98923727T patent/ATE304531T1/de active
- 1998-05-26 DK DK05077084T patent/DK1612207T3/da active
- 1998-05-26 AU AU75950/98A patent/AU765194B2/en not_active Expired
- 1998-05-26 EP EP98923727A patent/EP1082307B1/en not_active Expired - Lifetime
- 1998-05-26 EP EP05077084A patent/EP1612207B1/en not_active Expired - Lifetime
- 1998-05-26 WO PCT/US1998/010599 patent/WO1999061425A1/en not_active Ceased
- 1998-05-26 ES ES05077084T patent/ES2320012T3/es not_active Expired - Lifetime
- 1998-05-26 DE DE69840457T patent/DE69840457D1/de not_active Expired - Lifetime
- 1998-05-26 AT AT05077084T patent/ATE420073T1/de active
- 1998-05-26 CA CA002333089A patent/CA2333089C/en not_active Expired - Lifetime
- 1998-05-26 ES ES98923727T patent/ES2249830T3/es not_active Expired - Lifetime
-
2009
- 2009-02-26 CY CY20091100223T patent/CY1108818T1/el unknown
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