JP2002515487A5 - - Google Patents
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- Publication number
- JP2002515487A5 JP2002515487A5 JP2000549591A JP2000549591A JP2002515487A5 JP 2002515487 A5 JP2002515487 A5 JP 2002515487A5 JP 2000549591 A JP2000549591 A JP 2000549591A JP 2000549591 A JP2000549591 A JP 2000549591A JP 2002515487 A5 JP2002515487 A5 JP 2002515487A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- hydrogen
- compound according
- compound
- phenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 description 22
- 229910052739 hydrogen Inorganic materials 0.000 description 17
- 239000001257 hydrogen Substances 0.000 description 17
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 description 9
- 150000002431 hydrogen Chemical group 0.000 description 8
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 description 6
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 description 5
- 229910052736 halogen Inorganic materials 0.000 description 5
- 150000002367 halogens Chemical group 0.000 description 5
- 125000001424 substituent group Chemical group 0.000 description 5
- 125000004189 3,4-dichlorophenyl group Chemical group [H]C1=C([H])C(Cl)=C(Cl)C([H])=C1* 0.000 description 2
- 125000001255 4-fluorophenyl group Chemical group [H]C1=C([H])C(*)=C([H])C([H])=C1F 0.000 description 2
- 0 C[n]1nnnc1* Chemical compound C[n]1nnnc1* 0.000 description 1
- 208000006673 asthma Diseases 0.000 description 1
- 239000003814 drug Substances 0.000 description 1
- 239000003937 drug carrier Substances 0.000 description 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 description 1
- 238000004519 manufacturing process Methods 0.000 description 1
- 239000000203 mixture Substances 0.000 description 1
- 239000008194 pharmaceutical composition Substances 0.000 description 1
- 150000003839 salts Chemical class 0.000 description 1
- 239000002462 tachykinin receptor antagonist Substances 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US7961098A | 1998-05-15 | 1998-05-15 | |
| US09/079,610 | 1998-05-15 | ||
| PCT/US1999/009450 WO1999059972A1 (en) | 1998-05-15 | 1999-04-30 | Carboxy substituted carboxamide derivatives as tachykinin receptor antagonists |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2002515487A JP2002515487A (ja) | 2002-05-28 |
| JP2002515487A5 true JP2002515487A5 (enExample) | 2006-01-05 |
| JP4132671B2 JP4132671B2 (ja) | 2008-08-13 |
Family
ID=22151630
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2000549591A Expired - Lifetime JP4132671B2 (ja) | 1998-05-15 | 1999-04-30 | タキキニン受容体アンタゴニストとしてのカルボキシ置換カルボキサミド誘導体 |
Country Status (20)
| Country | Link |
|---|---|
| EP (1) | EP1077942B1 (enExample) |
| JP (1) | JP4132671B2 (enExample) |
| KR (1) | KR20010043598A (enExample) |
| CN (1) | CN1136191C (enExample) |
| AR (1) | AR015298A1 (enExample) |
| AT (1) | ATE286882T1 (enExample) |
| AU (1) | AU743487B2 (enExample) |
| DE (1) | DE69923173T2 (enExample) |
| DK (1) | DK200001669A (enExample) |
| ES (1) | ES2233042T3 (enExample) |
| HU (1) | HUP0102531A3 (enExample) |
| IL (1) | IL139262A (enExample) |
| MX (1) | MXPA00011204A (enExample) |
| NO (1) | NO319766B1 (enExample) |
| NZ (1) | NZ507432A (enExample) |
| PT (1) | PT1077942E (enExample) |
| SI (1) | SI1077942T1 (enExample) |
| TW (1) | TWI228122B (enExample) |
| WO (1) | WO1999059972A1 (enExample) |
| ZA (1) | ZA200006606B (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20020082421A1 (en) * | 2000-09-14 | 2002-06-27 | Abdel-Magid Ahmed F. | Novel solid salt forms of N-[2-[4-[2-(1- methylethoxy)phenyl]-1-piperazinyl]-2-oxo-1piperidineacetamide |
| US20060128752A1 (en) * | 2002-07-03 | 2006-06-15 | Giuseppe Alvaro | Chemical compounds |
| US8093268B2 (en) | 2007-01-24 | 2012-01-10 | Glaxo Group Limited | Pharmaceutical compositions comprising 2-methoxy-5-(5-trifluoromethyl-tetrazol-1-yl-benzyl)-(2S-phenylpiperidin-3S-yl-) |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9502644D0 (en) * | 1995-02-10 | 1995-03-29 | Zeneca Ltd | Heterocyclic derivatives |
| FR2738245B1 (fr) * | 1995-08-28 | 1997-11-21 | Sanofi Sa | Nouveaux derives de piperidine, procede pour leur obtention et compositions pharmaceutiques les contenant |
-
1999
- 1999-04-30 AU AU37756/99A patent/AU743487B2/en not_active Ceased
- 1999-04-30 DE DE69923173T patent/DE69923173T2/de not_active Expired - Lifetime
- 1999-04-30 IL IL13926299A patent/IL139262A/xx not_active IP Right Cessation
- 1999-04-30 HU HU0102531A patent/HUP0102531A3/hu unknown
- 1999-04-30 NZ NZ507432A patent/NZ507432A/en unknown
- 1999-04-30 AT AT99920201T patent/ATE286882T1/de not_active IP Right Cessation
- 1999-04-30 WO PCT/US1999/009450 patent/WO1999059972A1/en not_active Ceased
- 1999-04-30 EP EP99920201A patent/EP1077942B1/en not_active Expired - Lifetime
- 1999-04-30 JP JP2000549591A patent/JP4132671B2/ja not_active Expired - Lifetime
- 1999-04-30 MX MXPA00011204A patent/MXPA00011204A/es not_active IP Right Cessation
- 1999-04-30 KR KR1020007012743A patent/KR20010043598A/ko not_active Ceased
- 1999-04-30 CN CNB998061891A patent/CN1136191C/zh not_active Expired - Fee Related
- 1999-04-30 SI SI9930752T patent/SI1077942T1/xx unknown
- 1999-04-30 PT PT99920201T patent/PT1077942E/pt unknown
- 1999-04-30 ES ES99920201T patent/ES2233042T3/es not_active Expired - Lifetime
- 1999-05-13 AR ARP990102258A patent/AR015298A1/es active IP Right Grant
- 1999-05-24 TW TW088107935A patent/TWI228122B/zh not_active IP Right Cessation
-
2000
- 2000-11-09 DK DK200001669A patent/DK200001669A/da not_active Application Discontinuation
- 2000-11-14 NO NO20005756A patent/NO319766B1/no unknown
- 2000-11-14 ZA ZA200006606A patent/ZA200006606B/en unknown