JP2002506014A - 新規な避妊用キット - Google Patents

新規な避妊用キット

Info

Publication number
JP2002506014A
JP2002506014A JP2000535302A JP2000535302A JP2002506014A JP 2002506014 A JP2002506014 A JP 2002506014A JP 2000535302 A JP2000535302 A JP 2000535302A JP 2000535302 A JP2000535302 A JP 2000535302A JP 2002506014 A JP2002506014 A JP 2002506014A
Authority
JP
Japan
Prior art keywords
contraceptive
steroid
steroid compound
compound
structural formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2000535302A
Other languages
English (en)
Japanese (ja)
Inventor
クローステルブール,ヘレニウス・ヤン
デケルス,ホーデフリドス・ヘルマヌス・ヨハンナ
ハーメルスマ,ヨハンネス・アントニウス・マリア
フエルボスト,ピーテル・ミヒエル
クーリニグ・ベンニンク,ヘルマン・ヤン・テイメン
Original Assignee
アクゾ・ノベル・エヌ・ベー
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by アクゾ・ノベル・エヌ・ベー filed Critical アクゾ・ノベル・エヌ・ベー
Publication of JP2002506014A publication Critical patent/JP2002506014A/ja
Withdrawn legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • A61K31/569Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone substituted in position 17 alpha, e.g. ethisterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/575Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Reproductive Health (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
JP2000535302A 1998-03-09 1999-03-03 新規な避妊用キット Withdrawn JP2002506014A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP98200744.5 1998-03-09
EP98200744 1998-03-09
PCT/EP1999/001404 WO1999045886A2 (en) 1998-03-09 1999-03-03 New contraceptive kit for monotherapy

Publications (1)

Publication Number Publication Date
JP2002506014A true JP2002506014A (ja) 2002-02-26

Family

ID=8233452

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2000535302A Withdrawn JP2002506014A (ja) 1998-03-09 1999-03-03 新規な避妊用キット

Country Status (20)

Country Link
EP (1) EP1061928A2 (de)
JP (1) JP2002506014A (de)
KR (1) KR20010041698A (de)
CN (1) CN1292702A (de)
AR (1) AR018313A1 (de)
AU (1) AU756882B2 (de)
BR (1) BR9908605A (de)
CA (1) CA2319765A1 (de)
CO (1) CO5070598A1 (de)
HU (1) HUP0101007A3 (de)
ID (1) ID25621A (de)
IL (1) IL137541A0 (de)
NO (1) NO20004492D0 (de)
NZ (1) NZ506115A (de)
PE (1) PE20000330A1 (de)
PL (1) PL343428A1 (de)
RU (1) RU2225714C2 (de)
TR (1) TR200002593T2 (de)
WO (1) WO1999045886A2 (de)
ZA (1) ZA991851B (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1999051214A2 (en) * 1998-04-07 1999-10-14 Akzo Nobel N.V. Progestogen-only contraceptive kit
NZ517281A (en) 1999-09-06 2003-09-26 Akzo Nobel Nv Non-aromatic estrogenic steroids with a hydrocarbon substituent in position 11
KR20030029640A (ko) 2000-07-28 2003-04-14 악조 노벨 엔.브이. 16 알파-메틸 또는 에틸 치환 에스트로겐
EP1485103A1 (de) * 2002-03-11 2004-12-15 Janssen Pharmaceutica N.V. Kontinuierliches sulfatase-hemmendes progestogen enthaltendes kontrazeptionsschema
WO2003077927A1 (en) * 2002-03-11 2003-09-25 Janssen Pharmaceutica N.V. Sulfatase inhibiting progestogen-only contraceptive regimens
UA89964C2 (ru) 2004-09-08 2010-03-25 Н.В. Органон 15β-ЗАМЕЩЕННЫЕ СТЕРОИДЫ, КОТОРЫЕ ИМЕЮТ СЕЛЕКТИВНУЮ ЭСТРОГЕННУЮ АКТИВНОСТЬ

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7701384A (nl) * 1977-02-10 1978-08-14 Akzo Nv Werkwijze voor het bereiden van nieuwe steroiden van de oestraanreeks.
DE4227989A1 (de) * 1992-08-21 1994-06-09 Schering Ag Mittel zur transdermalen Applikation enthaltend 3-Keto-desogestrel
ZA94715B (en) * 1993-02-08 1994-10-24 Akzo Nv Steroids for treating menopausal complaints

Also Published As

Publication number Publication date
NO20004492L (no) 2000-09-08
AU3143799A (en) 1999-09-27
BR9908605A (pt) 2001-04-24
HUP0101007A3 (en) 2002-02-28
NO20004492D0 (no) 2000-09-08
ID25621A (id) 2000-10-19
AU756882B2 (en) 2003-01-23
PL343428A1 (en) 2001-08-13
ZA991851B (en) 1999-09-22
CN1292702A (zh) 2001-04-25
AR018313A1 (es) 2001-11-14
CA2319765A1 (en) 1999-09-16
PE20000330A1 (es) 2000-05-16
HUP0101007A2 (hu) 2001-12-28
TR200002593T2 (tr) 2000-12-21
RU2225714C2 (ru) 2004-03-20
KR20010041698A (ko) 2001-05-25
WO1999045886A2 (en) 1999-09-16
IL137541A0 (en) 2001-07-24
EP1061928A2 (de) 2000-12-27
WO1999045886A3 (en) 1999-12-02
NZ506115A (en) 2003-07-25
CO5070598A1 (es) 2001-08-28

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Legal Events

Date Code Title Description
A300 Application deemed to be withdrawn because no request for examination was validly filed

Free format text: JAPANESE INTERMEDIATE CODE: A300

Effective date: 20060509