JP2001506986A5 - - Google Patents

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Publication number
JP2001506986A5
JP2001506986A5 JP1998525838A JP52583898A JP2001506986A5 JP 2001506986 A5 JP2001506986 A5 JP 2001506986A5 JP 1998525838 A JP1998525838 A JP 1998525838A JP 52583898 A JP52583898 A JP 52583898A JP 2001506986 A5 JP2001506986 A5 JP 2001506986A5
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JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP1998525838A
Other languages
English (en)
Japanese (ja)
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JP2001506986A (ja
JP4094066B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US1997/022355 external-priority patent/WO1998024804A2/en
Publication of JP2001506986A publication Critical patent/JP2001506986A/ja
Publication of JP2001506986A5 publication Critical patent/JP2001506986A5/ja
Application granted granted Critical
Publication of JP4094066B2 publication Critical patent/JP4094066B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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JP52583898A 1996-12-06 1997-12-05 インターロイキン−1β変換酵素のインヒビター Expired - Lifetime JP4094066B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US3212996P 1996-12-06 1996-12-06
US60/032,129 1996-12-06
US4193897P 1997-04-04 1997-04-04
US60/041,938 1997-04-04
US5079697P 1997-06-26 1997-06-26
US60/050,796 1997-06-26
PCT/US1997/022355 WO1998024804A2 (en) 1996-12-06 1997-12-05 INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME

Publications (3)

Publication Number Publication Date
JP2001506986A JP2001506986A (ja) 2001-05-29
JP2001506986A5 true JP2001506986A5 (enExample) 2005-08-11
JP4094066B2 JP4094066B2 (ja) 2008-06-04

Family

ID=27364031

Family Applications (1)

Application Number Title Priority Date Filing Date
JP52583898A Expired - Lifetime JP4094066B2 (ja) 1996-12-06 1997-12-05 インターロイキン−1β変換酵素のインヒビター

Country Status (8)

Country Link
US (1) US6350741B1 (enExample)
EP (1) EP0942925B1 (enExample)
JP (1) JP4094066B2 (enExample)
AT (1) ATE346085T1 (enExample)
AU (1) AU7624798A (enExample)
CA (1) CA2274250A1 (enExample)
DE (1) DE69736984T2 (enExample)
WO (1) WO1998024804A2 (enExample)

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CA2740885C (en) 2008-10-16 2018-04-03 The Regents Of The University Of California Fused ring heteroaryl kinase inhibitors
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WO2011047384A2 (en) 2009-10-16 2011-04-21 The Regents Of The University Of California Methods of inhibiting ire1
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JP2013545749A (ja) 2010-11-10 2013-12-26 インフィニティー ファーマシューティカルズ, インコーポレイテッド 複素環化合物及びその使用
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JP6130305B2 (ja) 2011-02-23 2017-05-17 インテリカイン, エルエルシー キナーゼ阻害剤の組み合わせおよびそれらの使用
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JP7398391B2 (ja) 2018-04-20 2023-12-14 エフ. ホフマン-ラ ロシュ アーゲー N-[4-オキソ-2,3-ジヒドロ-1,5-ベンズオキサゼピン-3-イル]-5,6-ジヒドロ-4H-ピロロ[1,2-b]ピラゾール-2-カルボキサミド誘導体及び例えば過敏性腸症候群(IBS)を処置するためのRIP1キナーゼ阻害剤としての関連化合物
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WO2026082873A1 (en) 2024-10-17 2026-04-23 Institut National de la Santé et de la Recherche Médicale Use of caspase-1 inhibitors for treating ineffective erythropoiesis in patients suffering from sickle cell disease

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US6204261B1 (en) * 1995-12-20 2001-03-20 Vertex Pharmaceuticals Incorporated Inhibitors of interleukin-1β Converting enzyme inhibitors
WO1994026723A2 (en) * 1993-05-14 1994-11-24 Genentech, Inc. ras FARNESYL TRANSFERASE INHIBITORS
US5580979A (en) * 1994-03-15 1996-12-03 Trustees Of Tufts University Phosphotyrosine peptidomimetics for inhibiting SH2 domain interactions
US5716929A (en) * 1994-06-17 1998-02-10 Vertex Pharmaceuticals, Inc. Inhibitors of interleukin-1β converting enzyme
JPH09295996A (ja) * 1996-03-06 1997-11-18 Takeda Chem Ind Ltd システインプロテアーゼ阻害化合物

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