JP2000511528A5 - - Google Patents

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Publication number
JP2000511528A5
JP2000511528A5 JP1997542371A JP54237197A JP2000511528A5 JP 2000511528 A5 JP2000511528 A5 JP 2000511528A5 JP 1997542371 A JP1997542371 A JP 1997542371A JP 54237197 A JP54237197 A JP 54237197A JP 2000511528 A5 JP2000511528 A5 JP 2000511528A5
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JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP1997542371A
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English (en)
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JP2000511528A (ja
JP3897363B2 (ja
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Publication date
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Priority claimed from PCT/US1997/006602 external-priority patent/WO1997045397A1/en
Publication of JP2000511528A publication Critical patent/JP2000511528A/ja
Publication of JP2000511528A5 publication Critical patent/JP2000511528A5/ja
Application granted granted Critical
Publication of JP3897363B2 publication Critical patent/JP3897363B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Description

Figure 2000511528
Figure 2000511528
Figure 2000511528
Figure 2000511528
Figure 2000511528
Figure 2000511528
Figure 2000511528
Figure 2000511528
Figure 2000511528
Figure 2000511528
JP54237197A 1996-05-30 1997-04-24 アルキルオキシアミノ置換フルオレノンおよびプロテインキナーゼc阻害剤としてのその使用 Expired - Fee Related JP3897363B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US65553796A 1996-05-30 1996-05-30
US65558496A 1996-05-30 1996-05-30
US08/655,584 1996-05-30
US08/655,537 1996-05-30
PCT/US1997/006602 WO1997045397A1 (en) 1996-05-30 1997-04-24 Alkyloxyamino substituted fluorenones and their use as protein kinase c inhibitors

Publications (3)

Publication Number Publication Date
JP2000511528A JP2000511528A (ja) 2000-09-05
JP2000511528A5 true JP2000511528A5 (ja) 2005-01-13
JP3897363B2 JP3897363B2 (ja) 2007-03-22

Family

ID=27096988

Family Applications (1)

Application Number Title Priority Date Filing Date
JP54237197A Expired - Fee Related JP3897363B2 (ja) 1996-05-30 1997-04-24 アルキルオキシアミノ置換フルオレノンおよびプロテインキナーゼc阻害剤としてのその使用

Country Status (18)

Country Link
EP (1) EP0906268B1 (ja)
JP (1) JP3897363B2 (ja)
CN (1) CN1160309C (ja)
AR (1) AR008375A1 (ja)
AT (1) ATE209626T1 (ja)
AU (1) AU737073B2 (ja)
BR (1) BR9709406B1 (ja)
CA (1) CA2257136C (ja)
DE (1) DE69708629T2 (ja)
DK (1) DK0906268T3 (ja)
ES (1) ES2170390T3 (ja)
HK (1) HK1019147A1 (ja)
HU (1) HUP9901621A3 (ja)
IL (1) IL126873A (ja)
NO (1) NO312457B1 (ja)
NZ (1) NZ332597A (ja)
PT (1) PT906268E (ja)
WO (1) WO1997045397A1 (ja)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6103712A (en) * 1998-03-05 2000-08-15 Eli Lilly And Company Therapeutic treatment for asthma
US6103713A (en) * 1998-03-05 2000-08-15 Eli Lilly And Company Therapeutic treatment for autoimmune diseases
DE19908504C2 (de) * 1999-02-26 2003-04-30 Boehringer Ingelheim Pharma Großtechnisches Verfahren zur Herstellung von Derivaten der Biphenyl-2-carbonsäure durch Verseifen eines (2-Oxazolinyl)-2-biphenyl-Derivats mit Salzsäure
DE19917990A1 (de) * 1999-04-20 2000-11-02 Florian Lang Arzneimittel enthaltend Hemmstoffe der zellvolumenregulierten humanen Kinase h-sgk
ES2238463T3 (es) * 2000-08-18 2005-09-01 Agouron Pharmaceuticals, Inc. Hidroxiimino-fluorenos heterociclicos y uso para inhibir proteina-quinasas.
US7365193B2 (en) 2004-02-04 2008-04-29 Abbott Laboratories Amino-substituted tricyclic derivatives and methods of use
US20050171079A1 (en) * 2004-02-04 2005-08-04 Schrimpf Michael R. Amino-substituted tricyclic derivatives and methods of use
CA2786854A1 (en) * 2010-01-11 2011-07-14 Healor Ltd. Method for treatment of inflammatory disease and disorder
CN103204781B (zh) * 2013-03-14 2015-04-01 武汉大学 2,7–二取代芴酮衍生物及其制备方法与应用
CN109053435A (zh) * 2018-08-03 2018-12-21 上海华堇生物技术有限责任公司 2,3-二甲氧基苯甲酰氯的制备方法
CN115590964A (zh) * 2022-09-14 2023-01-13 苏州大学(Cn) 蛋白激酶c抑制剂在制备抗肿瘤转移药物中的应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL33573A (en) * 1968-12-30 1973-10-25 Richardson Merrell Inc Bis-basic ethers and thioethers of fluorenone,fluorenol and fluorene
US5034384A (en) * 1990-08-01 1991-07-23 Merck & Co., Inc. 2-(9-fluorenonyl)-carbapenem antibacterial agents

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