JP2000503321A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2000503321A5 JP2000503321A5 JP1997526110A JP52611097A JP2000503321A5 JP 2000503321 A5 JP2000503321 A5 JP 2000503321A5 JP 1997526110 A JP1997526110 A JP 1997526110A JP 52611097 A JP52611097 A JP 52611097A JP 2000503321 A5 JP2000503321 A5 JP 2000503321A5
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/588,711 US5804686A (en) | 1996-01-19 | 1996-01-19 | fused pyrrolecarboxamides; a new class of GABA brain receptor ligands |
| US08/588,711 | 1996-01-19 | ||
| PCT/US1997/000519 WO1997026243A1 (en) | 1996-01-19 | 1997-01-14 | Novel fused pyrrolecarboxamides; a new class of gaba brain receptor ligands |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2000503321A JP2000503321A (ja) | 2000-03-21 |
| JP2000503321A5 true JP2000503321A5 (OSRAM) | 2004-11-18 |
Family
ID=24354983
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP9526110A Ceased JP2000503321A (ja) | 1996-01-19 | 1997-01-14 | 新規な融合ピロールカルボキサミド；新規な種類のｇａｂａ脳リセプタリガンド |
Country Status (26)
| Country | Link |
|---|---|
| US (2) | US5804686A (OSRAM) |
| EP (1) | EP1019372B1 (OSRAM) |
| JP (1) | JP2000503321A (OSRAM) |
| KR (1) | KR100490108B1 (OSRAM) |
| CN (1) | CN1209805A (OSRAM) |
| AP (1) | AP1015A (OSRAM) |
| AT (1) | ATE322480T1 (OSRAM) |
| AU (1) | AU1746697A (OSRAM) |
| BG (1) | BG102634A (OSRAM) |
| BR (1) | BR9707051A (OSRAM) |
| CA (1) | CA2243317C (OSRAM) |
| CZ (1) | CZ215498A3 (OSRAM) |
| DE (1) | DE69735647T2 (OSRAM) |
| ES (1) | ES2263170T3 (OSRAM) |
| HU (1) | HUP9901018A3 (OSRAM) |
| IL (1) | IL125391A (OSRAM) |
| IS (1) | IS4798A (OSRAM) |
| MX (1) | MX9805701A (OSRAM) |
| NO (1) | NO312670B1 (OSRAM) |
| NZ (1) | NZ330861A (OSRAM) |
| OA (1) | OA10811A (OSRAM) |
| PL (1) | PL327936A1 (OSRAM) |
| RU (1) | RU2167151C2 (OSRAM) |
| SK (1) | SK94398A3 (OSRAM) |
| UA (1) | UA49001C2 (OSRAM) |
| WO (1) | WO1997026243A1 (OSRAM) |
Families Citing this family (33)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5750702A (en) * | 1993-10-27 | 1998-05-12 | Neurogen Corporation | Certain pyrrolo pyridine-3-carboxamides; a new class of GABA brain receptor ligands |
| US6211365B1 (en) | 1996-01-19 | 2001-04-03 | Neurogen Corporation | Fused pyrrolecarboxamides; a new class of GABA brain receptor ligands |
| US5804686A (en) * | 1996-01-19 | 1998-09-08 | Neurogen Corporation | fused pyrrolecarboxamides; a new class of GABA brain receptor ligands |
| EP0888300A1 (en) * | 1996-03-22 | 1999-01-07 | Neurogen Corporation | Certain fused pyrrolecarboxamides as gaba brain receptor ligands |
| US5723462A (en) * | 1996-04-26 | 1998-03-03 | Neurogen Corporation | Certain fused pyrrolecarboxamides a new class of GABA brain receptor ligands |
| NZ503916A (en) | 1997-11-13 | 2002-08-28 | Pfizer Prod Inc | Method of synthesis of pyrrole and indole amides |
| GT199800179A (es) * | 1997-11-13 | 2000-05-02 | Procedimiento de sintesis de pirrol amidas. | |
| AU2881199A (en) * | 1998-02-26 | 1999-09-15 | Neurogen Corporation | Substituted 1,4-dihydro-4-oxonicotinic carboxamides: gaba brain receptor ligands |
| GB9812038D0 (en) | 1998-06-04 | 1998-07-29 | Merck Sharp & Dohme | Therapeutic compound |
| AU5444499A (en) * | 1998-09-01 | 2000-03-21 | Nissan Chemical Industries Ltd. | Benzoxazine derivatives |
| PL354513A1 (en) * | 1999-08-31 | 2004-01-26 | Neurogen Corporation | Fused pyrrolecarboxamides: gaba brain receptor ligands |
| US20050014939A1 (en) * | 1999-08-31 | 2005-01-20 | Neurogen Corporation | Fused pyrrolecarboxamides: GABA brain receptor ligands |
| AU2001264932A1 (en) * | 2000-05-26 | 2001-12-11 | Neurogen Corporation | Oxo-imidazopyrimidine-carboxamides and their use as gaba brain receptor ligands |
| EP1315703A1 (en) * | 2000-09-06 | 2003-06-04 | Neurogen Corporation | Aryl substituted tetrahydroindazoles and their use as ligands for the gaba-a receptor |
| CA2419958A1 (en) * | 2000-09-06 | 2002-03-14 | Neurogen Corporation | Substituted fused pyrroleimines and pyrazoleimines |
| JP2004515491A (ja) * | 2000-12-04 | 2004-05-27 | ファイザー・プロダクツ・インク | 縮合ピロールカルボキサミド類の合成 |
| WO2003066634A1 (en) * | 2002-02-07 | 2003-08-14 | Neurogen Corporation | Substituted fused pyrazolecarboxylic acid arylamides and related compounds |
| ATE333455T1 (de) * | 2002-05-17 | 2006-08-15 | Neurogen Corp | Substituierte, ringkondensierte imidazolderivate: gabaa-rezeptorliganden |
| US7678363B2 (en) | 2005-08-26 | 2010-03-16 | Braincells Inc | Methods of treating psychiatric conditions comprising administration of muscarinic agents in combination with SSRIs |
| EP2258359A3 (en) | 2005-08-26 | 2011-04-06 | Braincells, Inc. | Neurogenesis by muscarinic receptor modulation with sabcomelin |
| WO2007047978A2 (en) | 2005-10-21 | 2007-04-26 | Braincells, Inc. | Modulation of neurogenesis by pde inhibition |
| AU2006308889A1 (en) * | 2005-10-31 | 2007-05-10 | Braincells, Inc. | GABA receptor mediated modulation of neurogenesis |
| US20100216734A1 (en) | 2006-03-08 | 2010-08-26 | Braincells, Inc. | Modulation of neurogenesis by nootropic agents |
| WO2007134077A2 (en) | 2006-05-09 | 2007-11-22 | Braincells, Inc. | 5 ht receptor mediated neurogenesis |
| CA2651813A1 (en) | 2006-05-09 | 2007-11-22 | Braincells, Inc. | Neurogenesis by modulating angiotensin |
| CA2662491A1 (en) | 2006-09-08 | 2008-03-13 | Braincells, Inc. | Combinations containing a 4-acylaminopyridine derivative |
| US10954231B2 (en) | 2006-10-16 | 2021-03-23 | Bionomics Limited | Anxiolytic compounds |
| DK2074123T3 (da) | 2006-10-16 | 2013-01-14 | Bionomics Ltd | Nye anxiolytiske forbindelser |
| WO2010099217A1 (en) | 2009-02-25 | 2010-09-02 | Braincells, Inc. | Modulation of neurogenesis using d-cycloserine combinations |
| CR20190244A (es) | 2010-08-31 | 2019-07-11 | Meiji Seika Pharma Co Ltd | Agentes control de plaga |
| EP2681198A4 (en) | 2011-03-02 | 2014-09-03 | Bionomics Ltd | NEW LITTLE MOLECULES AS THERAPIES |
| NZ615466A (en) | 2011-05-12 | 2016-02-26 | Bionomics Ltd | Methods for preparing naphthyridines |
| CN120081825B (zh) * | 2025-05-07 | 2025-09-16 | 天津匠新致成科技有限公司 | 一种化合物及其制备方法和医药用途 |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3455943A (en) * | 1966-10-21 | 1969-07-15 | American Cyanamid Co | Certain 5,8-dihydro-beta-carbolines |
| US4075343A (en) * | 1976-09-13 | 1978-02-21 | Pfizer Inc. | Anti-allergenic 5-alkoxyimidazo[1,2-A]quinoline-2-carboxylic acids and derivatives thereof |
| DE3029980A1 (de) * | 1980-08-08 | 1982-03-11 | Boehringer Mannheim Gmbh, 6800 Mannheim | Indolderivate und verfahren zu ihrer herstellung |
| JPS57123180A (en) * | 1980-12-17 | 1982-07-31 | Schering Ag | 3-substituted beta-carboline, manufacture and psychotropic drug containing same |
| DE3147276A1 (de) * | 1981-11-28 | 1983-06-09 | Boehringer Mannheim Gmbh, 6800 Mannheim | Verfahren zur herstellung von indolderivaten, deren verwendung als wertvolle zwischenprodukte und neue 4-hydroxyindole |
| DE3246932A1 (de) * | 1982-12-16 | 1984-06-20 | Schering AG, 1000 Berlin und 4709 Bergkamen | Substituierte 5h-pyrimido(5,4-b)indole |
| DE3335323A1 (de) * | 1983-09-27 | 1985-04-04 | Schering AG, 1000 Berlin und 4709 Bergkamen | Substituierte ss-carboline, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
| GB8429739D0 (en) * | 1984-11-24 | 1985-01-03 | Fbc Ltd | Fungicides |
| DE3535927A1 (de) * | 1985-10-04 | 1987-04-09 | Schering Ag | 3-vinyl- und 3-ethinyl-ss-carbolinderivate, ihre herstellung und ihre verwendung als arzneimittel |
| DK0552237T3 (da) * | 1990-10-09 | 1993-07-28 | Neurogen Corp | Visse cycloalkyl- og azacycloalkyl-pyrrolopyrimidiner, en klasse af ligander for GABA-receptorer i hjernen |
| US5243049A (en) * | 1992-01-22 | 1993-09-07 | Neurogen Corporation | Certain pyrroloquinolinones: a new class of GABA brain receptor ligands |
| AU3443493A (en) * | 1992-02-19 | 1993-09-13 | Upjohn Company, The | 3-substituted imidazo(1,5-a)quinoxalines and quinazolines with cns activity |
| US5266698A (en) * | 1992-04-30 | 1993-11-30 | Neurogen Corporation | Certain aryl and cycloalkyl fused imidazopyrazinediones; a new class of GABA brain receptor ligands |
| WO1994017095A1 (en) * | 1993-01-29 | 1994-08-04 | Ariad Pharmaceuticals, Inc. | Analogs of receptor tyrosine activation motifs and therapeutic uses thereof |
| FR2705095B1 (fr) * | 1993-05-12 | 1995-06-23 | Adir | Nouveaux indoles substitués, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent. |
| US5484944A (en) * | 1993-10-27 | 1996-01-16 | Neurogen Corporation | Certain fused pyrrolecarboxanilides and their use as GABA brain receptor ligands |
| US5804686A (en) * | 1996-01-19 | 1998-09-08 | Neurogen Corporation | fused pyrrolecarboxamides; a new class of GABA brain receptor ligands |
-
1996
- 1996-01-19 US US08/588,711 patent/US5804686A/en not_active Expired - Fee Related
-
1997
- 1997-01-14 RU RU98115534/04A patent/RU2167151C2/ru not_active IP Right Cessation
- 1997-01-14 EP EP97904754A patent/EP1019372B1/en not_active Expired - Lifetime
- 1997-01-14 CN CN97191759A patent/CN1209805A/zh active Pending
- 1997-01-14 ES ES97904754T patent/ES2263170T3/es not_active Expired - Lifetime
- 1997-01-14 SK SK943-98A patent/SK94398A3/sk unknown
- 1997-01-14 JP JP9526110A patent/JP2000503321A/ja not_active Ceased
- 1997-01-14 NZ NZ330861A patent/NZ330861A/xx unknown
- 1997-01-14 KR KR10-1998-0705446A patent/KR100490108B1/ko not_active Expired - Fee Related
- 1997-01-14 AP APAP/P/1998/001297A patent/AP1015A/en active
- 1997-01-14 CA CA002243317A patent/CA2243317C/en not_active Expired - Fee Related
- 1997-01-14 UA UA98073904A patent/UA49001C2/uk unknown
- 1997-01-14 CZ CZ982154A patent/CZ215498A3/cs unknown
- 1997-01-14 HU HU9901018A patent/HUP9901018A3/hu unknown
- 1997-01-14 IL IL12539197A patent/IL125391A/en not_active IP Right Cessation
- 1997-01-14 WO PCT/US1997/000519 patent/WO1997026243A1/en not_active Ceased
- 1997-01-14 DE DE69735647T patent/DE69735647T2/de not_active Expired - Fee Related
- 1997-01-14 BR BR9707051A patent/BR9707051A/pt not_active Application Discontinuation
- 1997-01-14 AT AT97904754T patent/ATE322480T1/de not_active IP Right Cessation
- 1997-01-14 AU AU17466/97A patent/AU1746697A/en not_active Abandoned
- 1997-01-14 PL PL97327936A patent/PL327936A1/xx unknown
-
1998
- 1998-07-15 BG BG102634A patent/BG102634A/xx unknown
- 1998-07-15 OA OA9800115A patent/OA10811A/en unknown
- 1998-07-15 MX MX9805701A patent/MX9805701A/es not_active IP Right Cessation
- 1998-07-16 IS IS4798A patent/IS4798A/is unknown
- 1998-07-17 NO NO19983315A patent/NO312670B1/no not_active IP Right Cessation
- 1998-09-04 US US09/148,247 patent/US6080873A/en not_active Expired - Fee Related