JP2000503010A5 - - Google Patents
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- Publication number
- JP2000503010A5 JP2000503010A5 JP1997524371A JP52437197A JP2000503010A5 JP 2000503010 A5 JP2000503010 A5 JP 2000503010A5 JP 1997524371 A JP1997524371 A JP 1997524371A JP 52437197 A JP52437197 A JP 52437197A JP 2000503010 A5 JP2000503010 A5 JP 2000503010A5
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Description
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US943195P | 1995-12-29 | 1995-12-29 | |
US60/009,431 | 1995-12-29 | ||
PCT/US1996/020087 WO1997024135A1 (en) | 1995-12-29 | 1996-12-20 | Amidino protease inhibitors |
Publications (2)
Publication Number | Publication Date |
---|---|
JP2000503010A JP2000503010A (ja) | 2000-03-14 |
JP2000503010A5 true JP2000503010A5 (ja) | 2004-11-04 |
Family
ID=21737595
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP09524371A Ceased JP2000503010A (ja) | 1995-12-29 | 1996-12-20 | アミジノプロテアーゼ阻害剤 |
Country Status (19)
Country | Link |
---|---|
US (5) | US6034127A (ja) |
EP (1) | EP0883405B1 (ja) |
JP (1) | JP2000503010A (ja) |
KR (1) | KR19990076817A (ja) |
AT (1) | ATE260112T1 (ja) |
BR (1) | BR9612360A (ja) |
CA (1) | CA2256309C (ja) |
CZ (1) | CZ206698A3 (ja) |
DE (1) | DE69631692T2 (ja) |
DK (1) | DK0883405T3 (ja) |
ES (1) | ES2213786T3 (ja) |
HU (1) | HUP9902256A3 (ja) |
IL (1) | IL124883A0 (ja) |
MX (1) | MX9805152A (ja) |
NO (1) | NO982987L (ja) |
NZ (1) | NZ326076A (ja) |
PL (1) | PL327986A1 (ja) |
PT (1) | PT883405E (ja) |
WO (1) | WO1997024135A1 (ja) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PT883405E (pt) | 1995-12-29 | 2004-06-30 | Dimensional Pharm Inc | Inibidores de amidino-protease |
SE9602646D0 (sv) | 1996-07-04 | 1996-07-04 | Astra Ab | Pharmaceutically-useful compounds |
TW499412B (en) * | 1996-11-26 | 2002-08-21 | Dimensional Pharm Inc | Aminoguanidines and alkoxyguanidines as protease inhibitors |
AU8270698A (en) | 1997-06-26 | 1999-01-19 | Eli Lilly And Company | Antithrombotic agents |
US6740682B2 (en) | 1997-08-29 | 2004-05-25 | Tularik Limited | Meta-benzamidine derivatives as serine protease inhibitors |
WO1999011658A1 (en) * | 1997-08-29 | 1999-03-11 | Proteus Molecular Design Ltd. | Meta-benzamidine derivatives as serin protease inhibitors |
DE69941224D1 (de) * | 1998-11-20 | 2009-09-17 | Fuso Pharmaceutical Ind | Nachweismethode für pankreatitis |
AR023510A1 (es) | 1999-04-21 | 2002-09-04 | Astrazeneca Ab | Un equipo de partes, formulacion farmaceutica y uso de un inhibidor de trombina. |
US6586617B1 (en) | 1999-04-28 | 2003-07-01 | Sumitomo Chemical Takeda Agro Company, Limited | Sulfonamide derivatives |
JP2001026506A (ja) * | 1999-04-28 | 2001-01-30 | Takeda Chem Ind Ltd | スルホンアミド誘導体 |
US6635637B2 (en) | 2000-08-04 | 2003-10-21 | Dimensional Pharmaceuticals, Inc. | Cyclic oxyguanidine protease inhibitors |
WO2002038108A2 (en) * | 2000-11-03 | 2002-05-16 | The J. David Gladstone Institutes | Methods of treating disorders related to apoe |
US8394813B2 (en) | 2000-11-14 | 2013-03-12 | Shire Llc | Active agent delivery systems and methods for protecting and administering active agents |
PT1383756E (pt) * | 2001-04-24 | 2008-06-19 | Aryx Therapeutics | Derivados de cumarina a utilizar como anticoagulantes |
AU2003302238A1 (en) | 2002-12-03 | 2004-06-23 | Axys Pharmaceuticals, Inc. | 2-(2-hydroxybiphenyl-3-yl)-1h-benzoimidazole-5-carboxamidine derivatives as factor viia inhibitors |
EP1751091A2 (en) * | 2004-03-25 | 2007-02-14 | Elan Pharmaceuticals, Inc. | 2-amino- and 2-thio-substituted 1,3-diaminopropanes |
GB0815781D0 (en) * | 2008-08-29 | 2008-10-08 | Xention Ltd | Novel potassium channel blockers |
GB0815782D0 (en) | 2008-08-29 | 2008-10-08 | Xention Ltd | Novel potassium channel blockers |
GB0815784D0 (en) * | 2008-08-29 | 2008-10-08 | Xention Ltd | Novel potassium channel blockers |
RU2019121905A (ru) * | 2010-12-31 | 2019-09-03 | Астразенека Юкей Лимитед | Ингибиторы аргиназы и способы их применения |
EP2989080A1 (en) * | 2013-04-22 | 2016-03-02 | Reuter Chemische Apparatebau KG | Process for preparing enantiomerically enriched 3-hydroxymethylpiperidine |
Family Cites Families (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3577432A (en) * | 1968-12-23 | 1971-05-04 | Robins Co Inc A H | 1-substituted-3-phenoxypyrrolidines |
CH526535A (de) | 1970-02-05 | 1972-08-15 | Sandoz Ag | Verfahren zur Herstellung neuer Pyrrolidin-1-carboxamidinderivate |
JPS537436B2 (ja) * | 1974-04-16 | 1978-03-17 | ||
JPS5175042A (ja) * | 1974-12-26 | 1976-06-29 | Ono Pharmaceutical Co | Guanijinoshibosanamidojudotaino seizohoho |
HU177098B (en) * | 1979-01-04 | 1981-07-28 | Gyogyszerkutato Intezet | Process for producing new peptidyl-n-carboxy-l-arginin-a |
US4316899A (en) | 1979-08-24 | 1982-02-23 | Beecham Group Limited | Chromanone derivatives, a process for their preparation and compositions containing them |
US4433152A (en) * | 1981-05-25 | 1984-02-21 | Nippon Chemiphar Co., Ltd. | Amidinopiperidine derivatives |
JPS58194861A (ja) * | 1982-05-10 | 1983-11-12 | Nippon Chemiphar Co Ltd | 新規ピペリジン誘導体およびその製造法 |
JPS62145060A (ja) | 1985-12-17 | 1987-06-29 | Tanabe Seiyaku Co Ltd | ピペラジン誘導体及びその製法 |
US5039805A (en) * | 1988-12-08 | 1991-08-13 | Hoffmann-La Roche Inc. | Novel benzoic and phenylacetic acid derivatives |
DE3913597A1 (de) | 1989-04-25 | 1990-11-08 | Heumann Pharma Gmbh & Co | Diazinderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
TW201303B (ja) * | 1990-07-05 | 1993-03-01 | Hoffmann La Roche | |
DE4127404A1 (de) | 1991-08-19 | 1993-02-25 | Thomae Gmbh Dr K | Cyclische iminoderivate, diese verbindungen enthaltende arzneimittel und verfahren zu ihrer herstellung |
CA2427890A1 (en) | 1992-02-05 | 1993-08-19 | Ralf Anderskewitz | New amidine derivatives, the preparation and use thereof |
TW223629B (ja) * | 1992-03-06 | 1994-05-11 | Hoffmann La Roche | |
TW257757B (ja) * | 1993-03-03 | 1995-09-21 | Boehringer Mannheim Gmbh | |
US5466811A (en) * | 1994-07-18 | 1995-11-14 | Merck & Co., Inc. | Dioxolenylmethyl carbamates pro moieties for amine drugs |
DE4430755A1 (de) * | 1994-08-30 | 1996-03-07 | Boehringer Mannheim Gmbh | Neue Phosphanoxide, Verfahren zu ihrer Herstellung sowie diese Verbindungen enthaltende Arzneimittel |
DE4430757A1 (de) * | 1994-08-30 | 1996-03-07 | Boehringer Mannheim Gmbh | Neue 4-Aminopyridazine, Verfahren zu ihrer Herstellung sowie diese Verbindungen enthaltende Arzneimittel |
CA2233344A1 (en) * | 1995-09-29 | 1997-04-03 | 3-Dimensional Pharmaceuticals, Inc. | Guanidino protease inhibitors |
PT883405E (pt) | 1995-12-29 | 2004-06-30 | Dimensional Pharm Inc | Inibidores de amidino-protease |
-
1996
- 1996-12-20 PT PT96944847T patent/PT883405E/pt unknown
- 1996-12-20 PL PL96327986A patent/PL327986A1/xx unknown
- 1996-12-20 BR BR9612360A patent/BR9612360A/pt unknown
- 1996-12-20 JP JP09524371A patent/JP2000503010A/ja not_active Ceased
- 1996-12-20 EP EP96944847A patent/EP0883405B1/en not_active Expired - Lifetime
- 1996-12-20 WO PCT/US1996/020087 patent/WO1997024135A1/en not_active Application Discontinuation
- 1996-12-20 DE DE69631692T patent/DE69631692T2/de not_active Expired - Fee Related
- 1996-12-20 IL IL12488396A patent/IL124883A0/xx unknown
- 1996-12-20 NZ NZ326076A patent/NZ326076A/en unknown
- 1996-12-20 ES ES96944847T patent/ES2213786T3/es not_active Expired - Lifetime
- 1996-12-20 DK DK96944847T patent/DK0883405T3/da active
- 1996-12-20 AT AT96944847T patent/ATE260112T1/de not_active IP Right Cessation
- 1996-12-20 CZ CZ982066A patent/CZ206698A3/cs unknown
- 1996-12-20 KR KR1019980704943A patent/KR19990076817A/ko not_active Application Discontinuation
- 1996-12-20 HU HU9902256A patent/HUP9902256A3/hu unknown
- 1996-12-20 CA CA002256309A patent/CA2256309C/en not_active Expired - Fee Related
- 1996-12-27 US US08/782,894 patent/US6034127A/en not_active Expired - Lifetime
-
1998
- 1998-06-24 MX MX9805152A patent/MX9805152A/es unknown
- 1998-06-26 NO NO982987A patent/NO982987L/no not_active Application Discontinuation
-
1999
- 1999-03-16 US US09/270,734 patent/US6133315A/en not_active Expired - Lifetime
-
2000
- 2000-02-11 US US09/502,005 patent/US6281206B1/en not_active Expired - Lifetime
- 2000-08-01 US US09/631,107 patent/US6225302B1/en not_active Expired - Lifetime
-
2001
- 2001-05-09 US US09/851,123 patent/US6414020B2/en not_active Expired - Lifetime