IT8424197A0 - Analoghi retro-inverso parzialmente modificati della neurotensina. - Google Patents

Analoghi retro-inverso parzialmente modificati della neurotensina.

Info

Publication number
IT8424197A0
IT8424197A0 IT8424197A IT2419784A IT8424197A0 IT 8424197 A0 IT8424197 A0 IT 8424197A0 IT 8424197 A IT8424197 A IT 8424197A IT 2419784 A IT2419784 A IT 2419784A IT 8424197 A0 IT8424197 A0 IT 8424197A0
Authority
IT
Italy
Prior art keywords
neurotensin
analogues
reverse
partially modified
modified retro
Prior art date
Application number
IT8424197A
Other languages
English (en)
Other versions
IT1178786B (it
Inventor
Fabio Bonelli
Antonello Pessi
Antonio Silvio Verdini
Original Assignee
Anic Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Anic Spa filed Critical Anic Spa
Priority to IT24197/84A priority Critical patent/IT1178786B/it
Publication of IT8424197A0 publication Critical patent/IT8424197A0/it
Priority to AT85115888T priority patent/ATE63317T1/de
Priority to DE8585115888T priority patent/DE3582786D1/de
Priority to EP85115888A priority patent/EP0185320B1/en
Priority to US06/808,617 priority patent/US4716149A/en
Priority to JP60287645A priority patent/JPS61155396A/ja
Application granted granted Critical
Publication of IT1178786B publication Critical patent/IT1178786B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/02Linear peptides containing at least one abnormal peptide link
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
IT24197/84A 1984-12-21 1984-12-21 Analoghi retro-inverso parzialmente modificati della neurotensina IT1178786B (it)

Priority Applications (6)

Application Number Priority Date Filing Date Title
IT24197/84A IT1178786B (it) 1984-12-21 1984-12-21 Analoghi retro-inverso parzialmente modificati della neurotensina
AT85115888T ATE63317T1 (de) 1984-12-21 1985-12-12 Teilweise modifizierte analogen von retroinverso neurotensinen.
DE8585115888T DE3582786D1 (de) 1984-12-21 1985-12-12 Teilweise modifizierte analogen von retroinverso neurotensinen.
EP85115888A EP0185320B1 (en) 1984-12-21 1985-12-12 Partially modified, retro-inverso neurotensin analogs
US06/808,617 US4716149A (en) 1984-12-21 1985-12-13 Partially modified, retro-inverso neurotensin analogs
JP60287645A JPS61155396A (ja) 1984-12-21 1985-12-20 ニユーロテンシン様ペプチド及びその製法

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT24197/84A IT1178786B (it) 1984-12-21 1984-12-21 Analoghi retro-inverso parzialmente modificati della neurotensina

Publications (2)

Publication Number Publication Date
IT8424197A0 true IT8424197A0 (it) 1984-12-21
IT1178786B IT1178786B (it) 1987-09-16

Family

ID=11212494

Family Applications (1)

Application Number Title Priority Date Filing Date
IT24197/84A IT1178786B (it) 1984-12-21 1984-12-21 Analoghi retro-inverso parzialmente modificati della neurotensina

Country Status (6)

Country Link
US (1) US4716149A (it)
EP (1) EP0185320B1 (it)
JP (1) JPS61155396A (it)
AT (1) ATE63317T1 (it)
DE (1) DE3582786D1 (it)
IT (1) IT1178786B (it)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1190389B (it) * 1985-09-19 1988-02-16 Eniricerche Spa Esapeptidi ad attivita' ipotensiva
ES2052517T3 (es) * 1986-07-16 1994-07-16 Eniricerche Spa Analogos de tuftsina parcialmente retroinversos, metodo de preparacion de los mismos y composiciones farmaceuticas que los contienen.
AU3534989A (en) * 1988-04-08 1989-11-03 Scripps Clinic And Research Foundation Polypeptides stabilized by covalent hydrogen bond replacements
US5807979A (en) * 1988-04-08 1998-09-15 The Scripps Research Institute Synthetic, three-dimensionally stabilized polypeptide mimics of HIV
US5374621A (en) * 1991-09-13 1994-12-20 Regents Of The University Of California Neurotensin method for inhibiting vascular leakage
KR20200141986A (ko) 2018-02-12 2020-12-21 다이어비티스-프리, 인크. 개선된 길항성 항-인간 cd40 단클론 항체
WO2020102454A1 (en) 2018-11-13 2020-05-22 Regents Of The University Of Minnesota Cd40 targeted peptides and uses thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3929756A (en) * 1973-11-21 1975-12-30 Univ Brandeis Synthetically produced tridecapeptide having the same activity as the hypothalamic substance, neurotensin
US4110321A (en) * 1976-07-12 1978-08-29 Folkers Karl Synthetic tridecapeptide [Gln4 ]-neurotensin having hormonal activity
US4331661A (en) * 1980-10-03 1982-05-25 The Salk Institute For Biological Studies Bombesin analogs
IT1212508B (it) * 1981-12-22 1989-11-22 Anic Spa Analoghi retro - invertiti dei penta - ed esapeptidi c - terminali della sostanza p. utili come vasodilatatori
IT1190891B (it) * 1982-06-24 1988-02-24 Anic Spa Metodo per la sintesi in fase solida di polipeptidi retroinvertiti
US4439359A (en) * 1982-07-02 1984-03-27 Merck & Co., Inc. Cyclic octapeptide analogs of neurotensin
US4613586A (en) * 1984-04-19 1986-09-23 Board Of Trustees Of The Leland Stanford Junior University Gastrin releasing peptide-like peptides

Also Published As

Publication number Publication date
EP0185320A3 (en) 1988-03-16
DE3582786D1 (de) 1991-06-13
ATE63317T1 (de) 1991-05-15
EP0185320B1 (en) 1991-05-08
JPS61155396A (ja) 1986-07-15
EP0185320A2 (en) 1986-06-25
US4716149A (en) 1987-12-29
IT1178786B (it) 1987-09-16

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