IT1313617B1 - Processo per la preparazione di derivati degli acidi biliari. - Google Patents

Processo per la preparazione di derivati degli acidi biliari.

Info

Publication number
IT1313617B1
IT1313617B1 IT1999MI001856A ITMI991856A IT1313617B1 IT 1313617 B1 IT1313617 B1 IT 1313617B1 IT 1999MI001856 A IT1999MI001856 A IT 1999MI001856A IT MI991856 A ITMI991856 A IT MI991856A IT 1313617 B1 IT1313617 B1 IT 1313617B1
Authority
IT
Italy
Prior art keywords
preparation
acid derivatives
biliary acid
formula
compounds
Prior art date
Application number
IT1999MI001856A
Other languages
English (en)
Inventor
Marino Brocchetta
Chiara Gallotti
Massimo Visigalli
Pier Lucio Anelli
Original Assignee
Bracco Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bracco Spa filed Critical Bracco Spa
Publication of ITMI991856A0 publication Critical patent/ITMI991856A0/it
Priority to IT1999MI001856A priority Critical patent/IT1313617B1/it
Priority to US09/449,998 priority patent/US6307074B1/en
Priority to AU75104/00A priority patent/AU766552B2/en
Priority to PT00964034T priority patent/PT1210359E/pt
Priority to EP00964034A priority patent/EP1210359B1/en
Priority to DE60020130T priority patent/DE60020130T2/de
Priority to CNB008121958A priority patent/CN1174994C/zh
Priority to ES00964034T priority patent/ES2240165T3/es
Priority to KR1020027002496A priority patent/KR100700474B1/ko
Priority to HU0203193A priority patent/HUP0203193A3/hu
Priority to JP2001519719A priority patent/JP4842475B2/ja
Priority to MXPA02002140A priority patent/MXPA02002140A/es
Priority to AT00964034T priority patent/ATE295368T1/de
Priority to IL14840400A priority patent/IL148404A0/xx
Priority to CA002383505A priority patent/CA2383505C/en
Priority to PCT/EP2000/008226 priority patent/WO2001016157A2/en
Priority to SI200030682T priority patent/SI1210359T1/xx
Publication of ITMI991856A1 publication Critical patent/ITMI991856A1/it
Priority to US09/934,603 priority patent/US6479681B2/en
Priority to IL148404A priority patent/IL148404A/en
Priority to NO20020969A priority patent/NO322018B1/no
Application granted granted Critical
Publication of IT1313617B1 publication Critical patent/IT1313617B1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J9/00Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
IT1999MI001856A 1999-08-31 1999-08-31 Processo per la preparazione di derivati degli acidi biliari. IT1313617B1 (it)

Priority Applications (20)

Application Number Priority Date Filing Date Title
IT1999MI001856A IT1313617B1 (it) 1999-08-31 1999-08-31 Processo per la preparazione di derivati degli acidi biliari.
US09/449,998 US6307074B1 (en) 1999-08-31 1999-11-26 Process for the preparation of bile acid derivatives
JP2001519719A JP4842475B2 (ja) 1999-08-31 2000-08-23 胆汁酸誘導体の製造方法
IL14840400A IL148404A0 (en) 1999-08-31 2000-08-23 A process for the preparation of 3-amino bile acid derivatives
EP00964034A EP1210359B1 (en) 1999-08-31 2000-08-23 A process for the preparation of 3-amino bile acid derivatives
DE60020130T DE60020130T2 (de) 1999-08-31 2000-08-23 Verfahren zur herstellung von 3-amino-gallensäure derivaten
CNB008121958A CN1174994C (zh) 1999-08-31 2000-08-23 胆汁酸衍生物的制备方法
ES00964034T ES2240165T3 (es) 1999-08-31 2000-08-23 Procedimiento de preparacion de derivados 3.amino de acidos biliares.
KR1020027002496A KR100700474B1 (ko) 1999-08-31 2000-08-23 3-아미노 바일산 유도체의 제조 방법
HU0203193A HUP0203193A3 (en) 1999-08-31 2000-08-23 Process for the preparation of 3-amino bile acid derivatives
AU75104/00A AU766552B2 (en) 1999-08-31 2000-08-23 A process for the preparation of 3-amino bile acid derivatives
MXPA02002140A MXPA02002140A (es) 1999-08-31 2000-08-23 Proceso para la preparacion de derivados de acido 3-amino biliar.
AT00964034T ATE295368T1 (de) 1999-08-31 2000-08-23 Verfahren zur herstellung 3-amino-gallensaurer derivate
PT00964034T PT1210359E (pt) 1999-08-31 2000-08-23 Processo para a preparacao de derivados do acido 3-amino-biliar
CA002383505A CA2383505C (en) 1999-08-31 2000-08-23 A process for the preparation of 3-amino bile acid derivatives
PCT/EP2000/008226 WO2001016157A2 (en) 1999-08-31 2000-08-23 A process for the preparation of 3-amino bile acid derivatives
SI200030682T SI1210359T1 (it) 1999-08-31 2000-08-23
US09/934,603 US6479681B2 (en) 1999-08-31 2001-08-23 Bile acid salts
IL148404A IL148404A (en) 1999-08-31 2002-02-27 Process for the preparation of 3-amino derivatives of bile acid
NO20020969A NO322018B1 (no) 1999-08-31 2002-02-27 Fremgangsmate ved fremstilling av gallesyrederivater og derivater fremstilt derved.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT1999MI001856A IT1313617B1 (it) 1999-08-31 1999-08-31 Processo per la preparazione di derivati degli acidi biliari.

Publications (3)

Publication Number Publication Date
ITMI991856A0 ITMI991856A0 (it) 1999-08-31
ITMI991856A1 ITMI991856A1 (it) 2001-03-03
IT1313617B1 true IT1313617B1 (it) 2002-09-09

Family

ID=11383568

Family Applications (1)

Application Number Title Priority Date Filing Date
IT1999MI001856A IT1313617B1 (it) 1999-08-31 1999-08-31 Processo per la preparazione di derivati degli acidi biliari.

Country Status (17)

Country Link
US (2) US6307074B1 (it)
EP (1) EP1210359B1 (it)
JP (1) JP4842475B2 (it)
KR (1) KR100700474B1 (it)
CN (1) CN1174994C (it)
AT (1) ATE295368T1 (it)
AU (1) AU766552B2 (it)
CA (1) CA2383505C (it)
DE (1) DE60020130T2 (it)
ES (1) ES2240165T3 (it)
HU (1) HUP0203193A3 (it)
IL (2) IL148404A0 (it)
IT (1) IT1313617B1 (it)
MX (1) MXPA02002140A (it)
NO (1) NO322018B1 (it)
PT (1) PT1210359E (it)
WO (1) WO2001016157A2 (it)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW319763B (it) * 1995-02-01 1997-11-11 Epix Medical Inc
EP1765406A4 (en) * 2004-05-21 2012-11-28 Mediplex Corp ADDITIVES FOR IMPROVED MUCOSAL ABSORPTION OF THERAPEUTIC AGENTS
ES2296463B1 (es) * 2005-07-13 2009-02-16 Universidade De Santiago Compostela Nuevos amidoderivados de acidos billares funcionalizados en la posicion 3 del anillo a. procedimientos para su obtencion y aplicaciones.
KR101139553B1 (ko) * 2009-06-10 2012-04-30 한양대학교 산학협력단 유기 겔과 무기 겔에 의한 나노 복합체의 조성물 및 그의 박막 코팅과 필름 제조방법
CN102153610B (zh) * 2011-02-28 2012-12-12 中国药科大学 一氧化氮供体型胆汁酸衍生物、其制备方法及医药用途
CN102766188B (zh) * 2012-07-24 2016-01-13 上海交通大学 胆固醇衍生物、螯合物、重组高密度脂蛋白及其用途
US20170299379A1 (en) * 2016-04-15 2017-10-19 Lockheed Martin Corporation Precision Hand-Held Scanner
EP3802558B1 (en) * 2018-05-30 2024-09-11 Translate Bio, Inc. Cationic lipids comprising a steroidal moiety
CN114904557B (zh) * 2022-06-13 2024-03-19 南华大学 一种胆酸钠衍生多孔Fe-N-C催化剂及其制备方法和应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0614908B1 (de) * 1993-03-09 1997-05-07 Hoechst Aktiengesellschaft Verfahren zur Herstellung von 3beta-Aminocholansäurederivaten
IT1269839B (it) * 1994-05-26 1997-04-15 Bracco Spa Coniugati di acidi biliari, loro derivati con complessi metallici e relativi usi

Also Published As

Publication number Publication date
HUP0203193A2 (hu) 2003-01-28
MXPA02002140A (es) 2003-03-27
CN1371387A (zh) 2002-09-25
ITMI991856A0 (it) 1999-08-31
ATE295368T1 (de) 2005-05-15
KR20020092903A (ko) 2002-12-12
KR100700474B1 (ko) 2007-03-28
HU0203193D0 (it) 2002-10-28
WO2001016157A2 (en) 2001-03-08
AU7510400A (en) 2001-03-26
US6479681B2 (en) 2002-11-12
EP1210359B1 (en) 2005-05-11
WO2001016157A3 (en) 2001-07-26
IL148404A (en) 2007-03-08
JP2003508407A (ja) 2003-03-04
IL148404A0 (en) 2002-09-12
CA2383505C (en) 2008-03-25
DE60020130D1 (de) 2005-06-16
AU766552B2 (en) 2003-10-16
DE60020130T2 (de) 2006-02-02
ITMI991856A1 (it) 2001-03-03
HUP0203193A3 (en) 2004-07-28
CA2383505A1 (en) 2001-03-08
ES2240165T3 (es) 2005-10-16
EP1210359A2 (en) 2002-06-05
US20020019549A1 (en) 2002-02-14
PT1210359E (pt) 2005-07-29
CN1174994C (zh) 2004-11-10
US6307074B1 (en) 2001-10-23
NO20020969L (no) 2002-04-25
NO322018B1 (no) 2006-08-07
NO20020969D0 (no) 2002-02-27
JP4842475B2 (ja) 2011-12-21

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