IT1219892B - FURANURONIC ACID DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS - Google Patents

FURANURONIC ACID DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS

Info

Publication number
IT1219892B
IT1219892B IT47794/88A IT4779488A IT1219892B IT 1219892 B IT1219892 B IT 1219892B IT 47794/88 A IT47794/88 A IT 47794/88A IT 4779488 A IT4779488 A IT 4779488A IT 1219892 B IT1219892 B IT 1219892B
Authority
IT
Italy
Prior art keywords
medications
preparation
acid derivatives
furanuronic
furanuronic acid
Prior art date
Application number
IT47794/88A
Other languages
Italian (it)
Other versions
IT8847794A0 (en
Inventor
Fulvio Gadient
Arnold Vogel
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of IT8847794A0 publication Critical patent/IT8847794A0/en
Application granted granted Critical
Publication of IT1219892B publication Critical patent/IT1219892B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16Purine radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IT47794/88A 1987-04-06 1988-03-30 FURANURONIC ACID DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS IT1219892B (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE3711561 1987-04-06
DE3711563 1987-04-06
DE3711564 1987-04-06
DE3711562 1987-04-06

Publications (2)

Publication Number Publication Date
IT8847794A0 IT8847794A0 (en) 1988-03-30
IT1219892B true IT1219892B (en) 1990-05-24

Family

ID=27433888

Family Applications (1)

Application Number Title Priority Date Filing Date
IT47794/88A IT1219892B (en) 1987-04-06 1988-03-30 FURANURONIC ACID DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS

Country Status (22)

Country Link
JP (1) JPS63258892A (en)
KR (1) KR880012629A (en)
AT (1) AT393507B (en)
AU (1) AU609109B2 (en)
BE (1) BE1002151A5 (en)
CA (1) CA1326017C (en)
CH (1) CH676121A5 (en)
DK (1) DK183488A (en)
ES (1) ES2007177A6 (en)
FI (1) FI87463C (en)
FR (1) FR2613367A1 (en)
GB (1) GB2203149B (en)
HU (1) HU201955B (en)
IL (1) IL85969A (en)
IT (1) IT1219892B (en)
LU (1) LU87181A1 (en)
MY (1) MY102323A (en)
NL (1) NL8800862A (en)
NZ (1) NZ224131A (en)
PH (1) PH25424A (en)
PT (1) PT87153B (en)
SE (1) SE8801236A0 (en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4755594A (en) * 1986-01-31 1988-07-05 Warner-Lambert Company N6 -substituted adenosines
US4954504A (en) * 1986-11-14 1990-09-04 Ciba-Geigy Corporation N9 -cyclopentyl-substituted adenine derivatives having adenosine-2 receptor stimulating activity
US5063233A (en) * 1986-11-14 1991-11-05 Ciba-Geigy Corporation N9 -cyclopentyl-substituted adenine derivatives useful as adenosine receptor agonists
NL8702926A (en) * 1986-12-15 1988-07-01 Sandoz Ag NEW FURANURONIC ACID DERIVATIVES AND METHODS FOR PREPARING AND USING THESE DERIVATIVES.
US4968697A (en) * 1987-02-04 1990-11-06 Ciba-Geigy Corporation 2-substituted adenosine 5'-carboxamides as antihypertensive agents
FI880405A (en) * 1987-02-04 1988-08-05 Ciba Geigy Ag Adenosine-5'-KARBOXAMIDDERIVAT.
USRE36494E (en) * 1990-02-20 2000-01-11 Discovery Therapeutics, Inc. 2-aralkoxy and 2-alkoxy adenosine derivatives as coronary vasodilators and antihypertensive agents
US5140015A (en) * 1990-02-20 1992-08-18 Whitby Research, Inc. 2-aralkoxy and 2-alkoxy adenosine derivatives as coronary vasodilators and antihypertensive agents
IT1254915B (en) * 1992-04-24 1995-10-11 Gloria Cristalli ADENOSINE DERIVATIVES FOR ACTIVITY A2 AGONIST
GB9301000D0 (en) * 1993-01-20 1993-03-10 Glaxo Group Ltd Chemical compounds
TW528755B (en) 1996-12-24 2003-04-21 Glaxo Group Ltd 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives
YU44900A (en) 1998-01-31 2003-01-31 Glaxo Group Limited 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives
HUP0103025A3 (en) 1998-06-23 2002-04-29 Glaxo Group Ltd A2a agonist 2-(purin-9-yl)tetrahydrofuran-3,4-diol derivatives, medicaments containing the same, process for producing them and the useful intermediates
US6593078B1 (en) 1999-04-16 2003-07-15 Schering Corporation Use of azetidinone compounds
US20050033044A1 (en) 2003-05-19 2005-02-10 Bristol-Myers Squibb Pharma Company Methods for preparing 2-alkynyladenosine derivatives
AR049384A1 (en) 2004-05-24 2006-07-26 Glaxo Group Ltd PURINA DERIVATIVES
BRPI0515506A (en) * 2004-09-20 2008-07-29 Inotek Pharmaceuticals Corp purine derivatives and methods of use thereof
GB0514809D0 (en) 2005-07-19 2005-08-24 Glaxo Group Ltd Compounds

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH606084A5 (en) * 1975-02-18 1978-10-13 Hoffmann La Roche (Di) nitrates of adenosine -5'-carboxylic acid derivs
US4167565A (en) * 1976-11-08 1979-09-11 Abbott Laboratories Adenosine-5'-carboxamides and method of use
DE3406533A1 (en) * 1984-02-23 1985-08-29 Boehringer Mannheim Gmbh, 6800 Mannheim USE OF ADENOSINE DERIVATIVES AS ANTIALLERGICA AND MEDICINAL PRODUCTS CONTAINING THEM
NL8702926A (en) * 1986-12-15 1988-07-01 Sandoz Ag NEW FURANURONIC ACID DERIVATIVES AND METHODS FOR PREPARING AND USING THESE DERIVATIVES.
FI880405A (en) * 1987-02-04 1988-08-05 Ciba Geigy Ag Adenosine-5'-KARBOXAMIDDERIVAT.

Also Published As

Publication number Publication date
PT87153B (en) 1992-07-31
FR2613367A1 (en) 1988-10-07
ES2007177A6 (en) 1989-06-01
AT393507B (en) 1991-11-11
LU87181A1 (en) 1988-11-17
DK183488D0 (en) 1988-04-05
NL8800862A (en) 1988-11-01
PH25424A (en) 1991-07-01
CA1326017C (en) 1994-01-11
IL85969A (en) 1992-03-29
AU1415188A (en) 1988-10-06
KR880012629A (en) 1988-11-28
CH676121A5 (en) 1990-12-14
FI881571A0 (en) 1988-04-05
FI881571A (en) 1988-10-07
HUT48902A (en) 1989-07-28
PT87153A (en) 1988-05-01
NZ224131A (en) 1991-12-23
FI87463C (en) 1993-01-11
IL85969A0 (en) 1988-09-30
GB2203149A (en) 1988-10-12
FI87463B (en) 1992-09-30
MY102323A (en) 1992-05-28
IT8847794A0 (en) 1988-03-30
DK183488A (en) 1988-10-07
BE1002151A5 (en) 1990-08-07
AU609109B2 (en) 1991-04-26
SE8801236L (en) 1988-10-17
ATA87388A (en) 1991-04-15
JPS63258892A (en) 1988-10-26
GB2203149B (en) 1991-02-13
HU201955B (en) 1991-01-28
SE8801236D0 (en) 1988-04-05
GB8807750D0 (en) 1988-05-05
SE8801236A0 (en) 1988-10-17

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Legal Events

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TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19940328