IT1130300B - PROCEDURE FOR PREPARING 1,1-PENICILLANIC ACID DIOXIDE AND ITS ESTERS - Google Patents

PROCEDURE FOR PREPARING 1,1-PENICILLANIC ACID DIOXIDE AND ITS ESTERS

Info

Publication number
IT1130300B
IT1130300B IT20367/80A IT2036780A IT1130300B IT 1130300 B IT1130300 B IT 1130300B IT 20367/80 A IT20367/80 A IT 20367/80A IT 2036780 A IT2036780 A IT 2036780A IT 1130300 B IT1130300 B IT 1130300B
Authority
IT
Italy
Prior art keywords
esters
preparing
procedure
penicillanic acid
acid dioxide
Prior art date
Application number
IT20367/80A
Other languages
Italian (it)
Other versions
IT8020367A0 (en
Inventor
Bernard S Moore
Ronnie D Carrol
Robert A Volkmann
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IT8020367A0 publication Critical patent/IT8020367A0/en
Application granted granted Critical
Publication of IT1130300B publication Critical patent/IT1130300B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
IT20367/80A 1979-03-05 1980-03-05 PROCEDURE FOR PREPARING 1,1-PENICILLANIC ACID DIOXIDE AND ITS ESTERS IT1130300B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1780879A 1979-03-05 1979-03-05
US1781079A 1979-03-05 1979-03-05

Publications (2)

Publication Number Publication Date
IT8020367A0 IT8020367A0 (en) 1980-03-05
IT1130300B true IT1130300B (en) 1986-06-11

Family

ID=26690337

Family Applications (1)

Application Number Title Priority Date Filing Date
IT20367/80A IT1130300B (en) 1979-03-05 1980-03-05 PROCEDURE FOR PREPARING 1,1-PENICILLANIC ACID DIOXIDE AND ITS ESTERS

Country Status (36)

Country Link
KR (1) KR850001339B1 (en)
AR (1) AR225031A1 (en)
AT (1) AT366693B (en)
AU (1) AU522572B2 (en)
BG (1) BG33292A3 (en)
CH (1) CH644608A5 (en)
CS (1) CS215130B2 (en)
DD (1) DD149367A5 (en)
DE (1) DE3008257C2 (en)
DK (2) DK159852C (en)
EG (1) EG14437A (en)
ES (1) ES489185A0 (en)
FI (1) FI70024C (en)
FR (1) FR2450836B1 (en)
GB (1) GB2045755B (en)
GR (1) GR67234B (en)
HK (1) HK66587A (en)
HU (1) HU186304B (en)
IE (1) IE49535B1 (en)
IL (1) IL59515A (en)
IN (1) IN153685B (en)
IT (1) IT1130300B (en)
KE (1) KE3464A (en)
LU (1) LU82215A1 (en)
MX (1) MX6032E (en)
MY (1) MY8500319A (en)
NL (1) NL180317C (en)
NO (2) NO800618L (en)
PL (1) PL125197B1 (en)
PT (1) PT70897A (en)
RO (1) RO80112A (en)
SE (2) SE449103B (en)
SG (1) SG55884G (en)
SU (1) SU1192626A3 (en)
UA (1) UA6342A1 (en)
YU (1) YU42328B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4419284A (en) * 1981-03-23 1983-12-06 Pfizer Inc. Preparation of halomethyl esters (and related esters) of penicillanic acid 1,1-dioxide
IN159362B (en) * 1981-03-23 1987-05-09 Pfizer
PT76527B (en) * 1982-04-19 1985-12-09 Gist Brocades Nv A process for the preparation of penicillanic acid 1,1-dioxide and derivatives thereof
IT1190897B (en) * 1982-06-29 1988-02-24 Opos Biochimica Srl PROCEDURE FOR THE PREPARATION OF THE 1-ETHOXYCARBONYLOXYETHYL ACID ACID 6- (D (-) - ALPHA AMINOALPHA-PHENYLACETAMIDE) -PENICILLANIC
US4606865A (en) * 1982-09-20 1986-08-19 Astra Lakemedel Aktiebolag Methods for the preparation of α-bromodiethylcarbonate
EP0139048A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the dehalogenation of 6,6-dibromopenicillanic acid 1,1-dioxide
EP0139047A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the preparation of 6,6-dibromopenicillanic acid 1,1-dioxide
US4596677A (en) * 1984-04-06 1986-06-24 Bristol-Myers Company Anhydropenicillin intermediates

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN149747B (en) * 1977-06-07 1982-04-03 Pfizer
CA1158639A (en) * 1978-12-11 1983-12-13 Eric M. Gordon 6-bromopenicillanic acid sulfone
DE3068390D1 (en) * 1979-01-10 1984-08-09 Beecham Group Plc Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
IE49880B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives

Also Published As

Publication number Publication date
IT8020367A0 (en) 1980-03-05
HU186304B (en) 1985-07-29
DE3008257A1 (en) 1980-09-11
KR850001339B1 (en) 1985-09-19
LU82215A1 (en) 1980-09-24
FR2450836B1 (en) 1986-03-21
DD149367A5 (en) 1981-07-08
NO823127L (en) 1980-09-08
SG55884G (en) 1985-03-08
FI800661A (en) 1980-09-06
RO80112A (en) 1982-10-26
HK66587A (en) 1987-09-25
MX6032E (en) 1984-10-04
PT70897A (en) 1980-04-01
AT366693B (en) 1982-04-26
PL125197B1 (en) 1983-04-30
UA6342A1 (en) 1994-12-29
YU58580A (en) 1983-02-28
AU522572B2 (en) 1982-06-17
DK166353C (en) 1993-09-06
CS215130B2 (en) 1982-07-30
IL59515A (en) 1983-02-23
SE8000512L (en) 1980-09-06
GB2045755A (en) 1980-11-05
EG14437A (en) 1984-09-30
KE3464A (en) 1984-10-12
DK166353B (en) 1993-04-13
BG33292A3 (en) 1983-01-14
ATA119080A (en) 1981-09-15
IN153685B (en) 1984-08-04
IL59515A0 (en) 1980-06-30
IE49535B1 (en) 1985-10-16
FI70024B (en) 1986-01-31
FR2450836A1 (en) 1980-10-03
MY8500319A (en) 1985-12-31
DK145690D0 (en) 1990-06-14
DK92680A (en) 1980-09-06
FI70024C (en) 1986-09-12
NO800618L (en) 1980-09-08
DE3008257C2 (en) 1984-03-01
ES8103094A1 (en) 1981-02-16
AR225031A1 (en) 1982-02-15
DK159852B (en) 1990-12-17
DK159852C (en) 1991-05-06
GR67234B (en) 1981-06-25
DK145690A (en) 1990-06-14
PL222448A1 (en) 1981-01-02
CH644608A5 (en) 1984-08-15
NL180317B (en) 1986-09-01
NL8001285A (en) 1980-09-09
SU1192626A3 (en) 1985-11-15
IE800429L (en) 1980-09-05
ES489185A0 (en) 1981-02-16
YU42328B (en) 1988-08-31
SE8603309D0 (en) 1986-08-04
AU5610480A (en) 1980-09-11
GB2045755B (en) 1983-01-26
NL180317C (en) 1987-02-02
SE8603309L (en) 1986-08-04
SE449103B (en) 1987-04-06

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Legal Events

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TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19970127