DK92680A - PROCEDURE FOR PENICILLANIC ACID-1,1-DIOXIDE E AND ESTERS THEREOF AND INTERMEDIATES USED IN THE PRESENT PROCEDURE - Google Patents

PROCEDURE FOR PENICILLANIC ACID-1,1-DIOXIDE E AND ESTERS THEREOF AND INTERMEDIATES USED IN THE PRESENT PROCEDURE

Info

Publication number
DK92680A
DK92680A DK92680A DK92680A DK92680A DK 92680 A DK92680 A DK 92680A DK 92680 A DK92680 A DK 92680A DK 92680 A DK92680 A DK 92680A DK 92680 A DK92680 A DK 92680A
Authority
DK
Denmark
Prior art keywords
procedure
esters
dioxide
intermediates used
penicillanic acid
Prior art date
Application number
DK92680A
Other languages
Danish (da)
Other versions
DK159852B (en
DK159852C (en
Inventor
B S Moore
R D Carroll
R A Volkmann
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK92680A publication Critical patent/DK92680A/en
Publication of DK159852B publication Critical patent/DK159852B/en
Application granted granted Critical
Publication of DK159852C publication Critical patent/DK159852C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Cosmetics (AREA)
DK092680A 1979-03-05 1980-03-04 PROCEDURE FOR THE PREPARATION OF PENICILLANIC ACID-1,1-DIOXIDE OR BASIC SALTS OR IN VIVO EASY HYDRAULIZABLE ESTERS DK159852C (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US1780879A 1979-03-05 1979-03-05
US1781079A 1979-03-05 1979-03-05
US1781079 1979-03-05
US1780879 1979-03-05

Publications (3)

Publication Number Publication Date
DK92680A true DK92680A (en) 1980-09-06
DK159852B DK159852B (en) 1990-12-17
DK159852C DK159852C (en) 1991-05-06

Family

ID=26690337

Family Applications (2)

Application Number Title Priority Date Filing Date
DK092680A DK159852C (en) 1979-03-05 1980-03-04 PROCEDURE FOR THE PREPARATION OF PENICILLANIC ACID-1,1-DIOXIDE OR BASIC SALTS OR IN VIVO EASY HYDRAULIZABLE ESTERS
DK145690A DK166353C (en) 1979-03-05 1990-06-14 Penicillanic acid 1,1-dioxide DERIVATIVES

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK145690A DK166353C (en) 1979-03-05 1990-06-14 Penicillanic acid 1,1-dioxide DERIVATIVES

Country Status (36)

Country Link
KR (1) KR850001339B1 (en)
AR (1) AR225031A1 (en)
AT (1) AT366693B (en)
AU (1) AU522572B2 (en)
BG (1) BG33292A3 (en)
CH (1) CH644608A5 (en)
CS (1) CS215130B2 (en)
DD (1) DD149367A5 (en)
DE (1) DE3008257C2 (en)
DK (2) DK159852C (en)
EG (1) EG14437A (en)
ES (1) ES8103094A1 (en)
FI (1) FI70024C (en)
FR (1) FR2450836B1 (en)
GB (1) GB2045755B (en)
GR (1) GR67234B (en)
HK (1) HK66587A (en)
HU (1) HU186304B (en)
IE (1) IE49535B1 (en)
IL (1) IL59515A (en)
IN (1) IN153685B (en)
IT (1) IT1130300B (en)
KE (1) KE3464A (en)
LU (1) LU82215A1 (en)
MX (1) MX6032E (en)
MY (1) MY8500319A (en)
NL (1) NL180317C (en)
NO (2) NO800618L (en)
PL (1) PL125197B1 (en)
PT (1) PT70897A (en)
RO (1) RO80112A (en)
SE (2) SE449103B (en)
SG (1) SG55884G (en)
SU (1) SU1192626A3 (en)
UA (1) UA6342A1 (en)
YU (1) YU42328B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4419284A (en) * 1981-03-23 1983-12-06 Pfizer Inc. Preparation of halomethyl esters (and related esters) of penicillanic acid 1,1-dioxide
IN159362B (en) * 1981-03-23 1987-05-09 Pfizer
PT76526B (en) * 1982-04-19 1986-01-21 Gist Brocades Nv Preparation of 6-alpha-bromo- and/or 6,6-dibromopenicillanic acid 1,1-dioxides
IT1190897B (en) * 1982-06-29 1988-02-24 Opos Biochimica Srl PROCEDURE FOR THE PREPARATION OF THE 1-ETHOXYCARBONYLOXYETHYL ACID ACID 6- (D (-) - ALPHA AMINOALPHA-PHENYLACETAMIDE) -PENICILLANIC
US4606865A (en) * 1982-09-20 1986-08-19 Astra Lakemedel Aktiebolag Methods for the preparation of α-bromodiethylcarbonate
EP0139048A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the dehalogenation of 6,6-dibromopenicillanic acid 1,1-dioxide
EP0139047A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the preparation of 6,6-dibromopenicillanic acid 1,1-dioxide
US4596677A (en) * 1984-04-06 1986-06-24 Bristol-Myers Company Anhydropenicillin intermediates

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN149747B (en) * 1977-06-07 1982-04-03 Pfizer
CA1158639A (en) * 1978-12-11 1983-12-13 Eric M. Gordon 6-bromopenicillanic acid sulfone
DE3068390D1 (en) * 1979-01-10 1984-08-09 Beecham Group Plc Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates

Also Published As

Publication number Publication date
KR850001339B1 (en) 1985-09-19
GB2045755B (en) 1983-01-26
FR2450836B1 (en) 1986-03-21
NL8001285A (en) 1980-09-09
NO800618L (en) 1980-09-08
DK166353C (en) 1993-09-06
LU82215A1 (en) 1980-09-24
DE3008257A1 (en) 1980-09-11
BG33292A3 (en) 1983-01-14
MY8500319A (en) 1985-12-31
GB2045755A (en) 1980-11-05
DK159852B (en) 1990-12-17
IN153685B (en) 1984-08-04
DK145690A (en) 1990-06-14
NL180317C (en) 1987-02-02
AU522572B2 (en) 1982-06-17
PT70897A (en) 1980-04-01
IT1130300B (en) 1986-06-11
RO80112A (en) 1982-10-26
YU58580A (en) 1983-02-28
PL125197B1 (en) 1983-04-30
UA6342A1 (en) 1994-12-29
GR67234B (en) 1981-06-25
HK66587A (en) 1987-09-25
IT8020367A0 (en) 1980-03-05
DE3008257C2 (en) 1984-03-01
FR2450836A1 (en) 1980-10-03
AU5610480A (en) 1980-09-11
HU186304B (en) 1985-07-29
IL59515A (en) 1983-02-23
IE800429L (en) 1980-09-05
ES489185A0 (en) 1981-02-16
PL222448A1 (en) 1981-01-02
ATA119080A (en) 1981-09-15
FI70024C (en) 1986-09-12
KE3464A (en) 1984-10-12
SG55884G (en) 1985-03-08
DK145690D0 (en) 1990-06-14
IL59515A0 (en) 1980-06-30
SE8603309L (en) 1986-08-04
DD149367A5 (en) 1981-07-08
IE49535B1 (en) 1985-10-16
SE8000512L (en) 1980-09-06
SE8603309D0 (en) 1986-08-04
MX6032E (en) 1984-10-04
ES8103094A1 (en) 1981-02-16
NL180317B (en) 1986-09-01
YU42328B (en) 1988-08-31
AR225031A1 (en) 1982-02-15
SU1192626A3 (en) 1985-11-15
DK166353B (en) 1993-04-13
FI800661A (en) 1980-09-06
CH644608A5 (en) 1984-08-15
CS215130B2 (en) 1982-07-30
FI70024B (en) 1986-01-31
NO823127L (en) 1980-09-08
SE449103B (en) 1987-04-06
AT366693B (en) 1982-04-26
DK159852C (en) 1991-05-06
EG14437A (en) 1984-09-30

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