IN2012DN05125A - - Google Patents

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Publication number
IN2012DN05125A
IN2012DN05125A IN5125DEN2012A IN2012DN05125A IN 2012DN05125 A IN2012DN05125 A IN 2012DN05125A IN 5125DEN2012 A IN5125DEN2012 A IN 5125DEN2012A IN 2012DN05125 A IN2012DN05125 A IN 2012DN05125A
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India
Prior art keywords
sphingosine
modulators
pharmaceuticals
preparing
processes
Prior art date
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English (en)
Inventor
M Heidelbaugh Todd
X Nguyen Phong
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Allergan Inc
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Publication of IN2012DN05125A publication Critical patent/IN2012DN05125A/en

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    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
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JP6294359B2 (ja) * 2013-02-20 2018-03-14 エルジー・ケム・リミテッド スフィンゴシン−１−リン酸受容体アゴニスト、その製造方法及びそれらを活性成分として含有する医薬組成物
US20140256945A1 (en) * 2013-03-07 2014-09-11 Allergan, Inc. Phosphonic acid compounds as sphingosine-1-phosphate receptor modulators
US20150045328A1 (en) * 2013-08-08 2015-02-12 Allergan, Inc. Disubstituted aryl oxy derivatives as sphingosine-1 phosphate receptors modulators
US20150045341A1 (en) * 2013-08-08 2015-02-12 Allergan, Inc. Disubstituted aryl azetidine derivatives as sphingosine-1 phosphate receptors modulators
WO2015073547A1 (en) * 2013-11-13 2015-05-21 Allergan, Inc. Disubstituted phenoxy azetidine derivatives as sphingosine-1-phosphate (s1p) receptor modulators
BR112020015567A2 (pt) 2018-02-02 2021-02-02 Kyoto University medicamento para prevenir ou tratar doença oftálmica associada com neovascularização intraocular e/ou permeabilidade vascular intraocular realçadas
US20240217935A1 (en) * 2021-04-14 2024-07-04 Lg Chem, Ltd. Method for preparing intermediate for synthesis of sphingosine-1-phosphate receptor agonist
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WO2022220611A1 (ko) * 2021-04-14 2022-10-20 주식회사 엘지화학 스핑고신-1-인산 수용체 효능제의 신규한 제조방법

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CA2780908A1 (en) 2011-06-03
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JP2013512244A (ja) 2013-04-11
KR20120098796A (ko) 2012-09-05
US20110212925A1 (en) 2011-09-01
CN102712618B (zh) 2014-11-26
BR112012012259A2 (pt) 2019-09-24
US20110152241A1 (en) 2011-06-23
IL219758A0 (en) 2012-07-31
NZ599966A (en) 2014-09-26
WO2011066179A1 (en) 2011-06-03
AU2010324983A1 (en) 2012-06-07
BR112012012261A2 (pt) 2016-04-26
CN102712607B (zh) 2016-06-22
JP2013512243A (ja) 2013-04-11
RU2012122615A (ru) 2013-12-27
KR20120101686A (ko) 2012-09-14
CA2780987A1 (en) 2011-06-03
AU2010324988B2 (en) 2016-05-26
IN2012DN05171A (zh) 2015-10-23
CA2780987C (en) 2018-03-06
US20140107075A1 (en) 2014-04-17
ZA201203523B (en) 2013-01-31
MX2012006028A (es) 2012-06-19
EP2504323B1 (en) 2017-03-15
JP5939158B2 (ja) 2016-06-22
WO2011066184A1 (en) 2011-06-03
MX2012006022A (es) 2012-08-15
AU2010324988A1 (en) 2012-06-07
IL219759A0 (en) 2012-07-31
CN102712607A (zh) 2012-10-03
CL2012001352A1 (es) 2012-08-31
RU2012125184A (ru) 2013-12-27
ZA201203524B (en) 2013-01-30
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