IN2012DN01661A - - Google Patents

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Publication number
IN2012DN01661A
IN2012DN01661A IN1661DEN2012A IN2012DN01661A IN 2012DN01661 A IN2012DN01661 A IN 2012DN01661A IN 1661DEN2012 A IN1661DEN2012 A IN 1661DEN2012A IN 2012DN01661 A IN2012DN01661 A IN 2012DN01661A
Authority
IN
India
Prior art keywords
disclosed
compounds
intended
kits
abstract
Prior art date
Application number
Other languages
English (en)
Inventor
H Alex Brown
Craig W Lindsley
Alex G Waterson
Sarah A Scott
Original Assignee
Univ Vanderbilt
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Vanderbilt filed Critical Univ Vanderbilt
Publication of IN2012DN01661A publication Critical patent/IN2012DN01661A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10Spiro-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/438The ring being spiro-condensed with carbocyclic or heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
IN1661DEN2012 2009-07-24 2010-07-23 IN2012DN01661A (enExample)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22849209P 2009-07-24 2009-07-24
PCT/US2010/043045 WO2011011680A1 (en) 2009-07-24 2010-07-23 Isoform selective phospholipase d inhibitors

Publications (1)

Publication Number Publication Date
IN2012DN01661A true IN2012DN01661A (enExample) 2015-06-05

Family

ID=43499428

Family Applications (1)

Application Number Title Priority Date Filing Date
IN1661DEN2012 IN2012DN01661A (enExample) 2009-07-24 2010-07-23

Country Status (14)

Country Link
US (1) US9127005B2 (enExample)
EP (1) EP2456307B1 (enExample)
JP (1) JP2013500260A (enExample)
KR (1) KR20120090034A (enExample)
CN (1) CN102573474A (enExample)
AU (1) AU2010275526A1 (enExample)
BR (1) BR112012001586A2 (enExample)
CA (1) CA2768940C (enExample)
IL (1) IL217720A0 (enExample)
IN (1) IN2012DN01661A (enExample)
MX (1) MX2012001064A (enExample)
RU (1) RU2012106657A (enExample)
SG (1) SG178102A1 (enExample)
WO (1) WO2011011680A1 (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9453017B2 (en) 2011-09-30 2016-09-27 Vanderbilt University Antiviral therapies with phospholipase D inhibitors

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN2012DN01661A (enExample) 2009-07-24 2015-06-05 Univ Vanderbilt
WO2014093557A1 (en) * 2012-12-11 2014-06-19 Vanderbilt University Methods and compositions comprising akt inhibitors and/or phospholipase d inhibitors
AU2013359311A1 (en) * 2012-12-11 2015-07-23 Vanderbilt University Methods and compositions of treating HIV infection
CN114778844A (zh) * 2022-03-07 2022-07-22 天津市肿瘤医院(天津医科大学肿瘤医院) Pld1作为评估肿瘤患者对于化疗药物敏感性的分子标志物的用途
AR129618A1 (es) * 2022-06-16 2024-09-11 Japan Tobacco Inc Compuesto de dihidrooxadiazinona y su uso farmacéutico

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1281502B1 (it) 1995-06-13 1998-02-18 Sardinian Antiviral Research C Impiego di un inibitore non nucleosidico della trascrittasi inversa in associazione con inibitori nucleosidici per il trattamento della
US6187559B1 (en) 1997-08-28 2001-02-13 Novartis Ag Phospholipase D gene
WO2001089449A2 (en) 2000-05-25 2001-11-29 Ben Williger Phospholipase d effectors for therapy and screening
US6482829B2 (en) * 2000-06-08 2002-11-19 Hoffmann-La Roche Inc. Substituted heterocyclic siprodecane compound active as an antagonist of neurokinin 1 receptor
US20060172363A1 (en) 2002-09-18 2006-08-03 Postech Foundation Peptide complexes containing phospholipase d
KR20070106690A (ko) * 2004-12-27 2007-11-05 아스트라제네카 아베 피라졸론 화합물 및 대사성 글루타메이트 수용체길항제로서 그들의 용도
WO2006107451A2 (en) 2005-02-23 2006-10-12 Univ Emory Honokiol derivatives for the treatment of proliferative disorders
DE602007009221D1 (de) * 2006-05-18 2010-10-28 Hoffmann La Roche Thiazolopyramidin/pyridinharnstoffderivate als antagonisten am adenosin-a2b-rezeptor
US20100009970A1 (en) 2008-03-19 2010-01-14 Combinatorx (Singapore) Pte. Ltd. Compositions and methods for treatment of viral diseases
WO2010037081A1 (en) 2008-09-29 2010-04-01 Palatin Technologies, Inc. Melanocortin receptor-specific spiro-piperidine compounds
CA2756141A1 (en) 2009-03-31 2010-10-07 Sanofi-Aventis Deutschland Gmbh Drug delivery device body
EP2435563A4 (en) 2009-05-29 2013-10-02 Univ Columbia MODULATION OF PHOSPHOLIPASE D FOR THE TREATMENT OF NEURODEEGENERATIVE DISEASES
IN2012DN01661A (enExample) 2009-07-24 2015-06-05 Univ Vanderbilt
WO2011019498A1 (en) 2009-07-27 2011-02-17 The Trustees Of Princeton University Inhibition of glycerol-3-phosphate acyltransferase (gpat) and associated enzymes for treatment of viral infections
CA2850597A1 (en) 2011-09-30 2013-04-04 Vanderbilt University Antiviral therapies with phospholipase d inhibitors
WO2014093557A1 (en) 2012-12-11 2014-06-19 Vanderbilt University Methods and compositions comprising akt inhibitors and/or phospholipase d inhibitors
AU2013359311A1 (en) 2012-12-11 2015-07-23 Vanderbilt University Methods and compositions of treating HIV infection

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9453017B2 (en) 2011-09-30 2016-09-27 Vanderbilt University Antiviral therapies with phospholipase D inhibitors

Also Published As

Publication number Publication date
CA2768940A1 (en) 2011-01-27
JP2013500260A (ja) 2013-01-07
CA2768940C (en) 2018-03-13
US20120214832A1 (en) 2012-08-23
SG178102A1 (en) 2012-03-29
BR112012001586A2 (pt) 2015-09-01
WO2011011680A1 (en) 2011-01-27
CN102573474A (zh) 2012-07-11
US9127005B2 (en) 2015-09-08
EP2456307B1 (en) 2016-11-02
AU2010275526A1 (en) 2012-03-15
EP2456307A4 (en) 2013-01-16
RU2012106657A (ru) 2013-08-27
MX2012001064A (es) 2012-07-17
KR20120090034A (ko) 2012-08-16
IL217720A0 (en) 2012-03-29
EP2456307A1 (en) 2012-05-30

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