IN2012DN01414A - - Google Patents
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- Publication number
- IN2012DN01414A IN2012DN01414A IN1414DEN2012A IN2012DN01414A IN 2012DN01414 A IN2012DN01414 A IN 2012DN01414A IN 1414DEN2012 A IN1414DEN2012 A IN 1414DEN2012A IN 2012DN01414 A IN2012DN01414 A IN 2012DN01414A
- Authority
- IN
- India
- Prior art keywords
- nitroimidazooxazines
- drugs
- alone
- novel
- preparation
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5365—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with heterocyclic ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A61P31/06—Antibacterial agents for tuberculosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Plant Pathology (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Pulmonology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23039609P | 2009-07-31 | 2009-07-31 | |
| PCT/US2010/043906 WO2011014774A1 (en) | 2009-07-31 | 2010-07-30 | Nitroimidazooxazines and their uses in anti-tubercular therapy |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IN2012DN01414A true IN2012DN01414A (ko) | 2015-06-05 |
Family
ID=42937154
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IN1414DEN2012 IN2012DN01414A (ko) | 2009-07-31 | 2010-07-30 |
Country Status (12)
| Country | Link |
|---|---|
| EP (1) | EP2459571B1 (ko) |
| JP (1) | JP5781072B2 (ko) |
| KR (1) | KR101746482B1 (ko) |
| CN (1) | CN102753558B (ko) |
| AU (1) | AU2010278777B2 (ko) |
| BR (1) | BR112012002278A2 (ko) |
| CA (1) | CA2769359C (ko) |
| ES (1) | ES2536997T3 (ko) |
| IN (1) | IN2012DN01414A (ko) |
| NZ (1) | NZ598121A (ko) |
| RU (1) | RU2542988C2 (ko) |
| WO (1) | WO2011014774A1 (ko) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN103596960B (zh) * | 2011-04-15 | 2016-11-16 | 大塚制药株式会社 | 6,7-二氢咪唑并[2,1-b][1,3]噁嗪杀菌剂 |
| CN104059082B (zh) * | 2013-03-21 | 2016-08-03 | 苏州迈泰生物技术有限公司 | 硝基咪唑杂环类化合物及其在制备治疗结核病药物中的应用 |
| KR101682356B1 (ko) | 2014-11-04 | 2016-12-06 | 한국화학연구원 | 이미다조 옥사진 유도체, 이의 약학적으로 허용 가능한 염 또는 이의 광학이성질체 및 이를 유효성분으로 함유하는 약제학적 조성물 |
| CN107207532B (zh) | 2015-01-29 | 2019-07-30 | 南京明德新药研发股份有限公司 | 抗肺结核病的硝基咪唑衍生物 |
| CN108047248A (zh) * | 2018-02-12 | 2018-05-18 | 丹诺医药(苏州）有限公司 | 噁唑烷酮-硝基咪唑类偶联分子的应用 |
| CN113527331B (zh) * | 2020-04-17 | 2024-05-28 | 南京长澳医药科技有限公司 | 硝基咪唑类衍生物及其制备方法和用途 |
| CN113355439A (zh) * | 2021-06-07 | 2021-09-07 | 深圳市普瑞康生物技术有限公司 | 一种结核分枝杆菌潜伏感染及发病的新型组合检测方法 |
| CN114469946B (zh) * | 2022-02-24 | 2023-10-24 | 首都医科大学附属北京胸科医院 | 德拉马尼作为cxcl10抑制剂的用途 |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2184739A1 (en) | 1994-03-08 | 1995-09-14 | Jay E. Wrobel | Thiazolidinedione derivatives as anti-hyperglycemic agents |
| US5668127A (en) * | 1995-06-26 | 1997-09-16 | Pathogenesis Corporation | Nitroimidazole antibacterial compounds and methods of use thereof |
| US6087358A (en) | 1995-06-26 | 2000-07-11 | Pathogenesis Corporation | Nitro-[2,1-b]imidazopyran compounds and antibacterial uses thereof |
| AR041198A1 (es) * | 2002-10-11 | 2005-05-04 | Otsuka Pharma Co Ltd | Compuesto 2,3-dihidro-6-nitroimidazo[2,1-b] oxaxol, y composiciones farmaceuticas que lo contienen |
| CN100497345C (zh) * | 2003-10-31 | 2009-06-10 | 大塚制药株式会社 | 治疗结核病的2,3-二氢-6-硝基咪唑并[2,1-b]唑化合物 |
| DE602005004040T2 (de) | 2004-01-16 | 2008-12-11 | Sumitomo Chemical Co., Ltd. | Malononitrilverbindungen als Pestizide |
| TWI300409B (en) * | 2004-02-18 | 2008-09-01 | Otsuka Pharma Co Ltd | Method for producing 4-nitroimidazole compound |
| WO2006043121A1 (en) * | 2004-10-20 | 2006-04-27 | Ranbaxy Laboratories Limited | Oxazolidinone derivatives as antimicrobials |
| CN101268084A (zh) * | 2005-07-28 | 2008-09-17 | 沃泰克斯药物股份有限公司 | 天冬氨酸特异性半胱氨酸蛋白酶抑制剂前体药物 |
| US20080275035A1 (en) * | 2005-12-23 | 2008-11-06 | Jan Jiricek | Nitroimidazole Compounds |
| WO2009120789A1 (en) * | 2008-03-26 | 2009-10-01 | Global Alliance For Tb Drug Development | Bicyclic nitroimidazoles covalently linked to substituted phenyl oxazolidinones |
-
2010
- 2010-07-30 IN IN1414DEN2012 patent/IN2012DN01414A/en unknown
- 2010-07-30 NZ NZ598121A patent/NZ598121A/xx not_active IP Right Cessation
- 2010-07-30 AU AU2010278777A patent/AU2010278777B2/en not_active Ceased
- 2010-07-30 BR BR112012002278-4A patent/BR112012002278A2/pt not_active IP Right Cessation
- 2010-07-30 JP JP2012523087A patent/JP5781072B2/ja not_active Expired - Fee Related
- 2010-07-30 WO PCT/US2010/043906 patent/WO2011014774A1/en active Application Filing
- 2010-07-30 CN CN201080041453.9A patent/CN102753558B/zh not_active Expired - Fee Related
- 2010-07-30 RU RU2012107176/04A patent/RU2542988C2/ru not_active IP Right Cessation
- 2010-07-30 ES ES10742955.7T patent/ES2536997T3/es active Active
- 2010-07-30 CA CA2769359A patent/CA2769359C/en not_active Expired - Fee Related
- 2010-07-30 KR KR1020127005320A patent/KR101746482B1/ko active IP Right Grant
- 2010-07-30 EP EP10742955.7A patent/EP2459571B1/en not_active Not-in-force
Also Published As
| Publication number | Publication date |
|---|---|
| CA2769359A1 (en) | 2011-02-03 |
| JP2013500996A (ja) | 2013-01-10 |
| CN102753558A (zh) | 2012-10-24 |
| EP2459571A1 (en) | 2012-06-06 |
| KR101746482B1 (ko) | 2017-06-27 |
| AU2010278777B2 (en) | 2015-05-07 |
| BR112012002278A2 (pt) | 2020-09-15 |
| CA2769359C (en) | 2017-03-07 |
| CN102753558B (zh) | 2014-10-15 |
| RU2542988C2 (ru) | 2015-02-27 |
| NZ598121A (en) | 2013-04-26 |
| KR20120084713A (ko) | 2012-07-30 |
| AU2010278777A1 (en) | 2012-03-01 |
| WO2011014774A1 (en) | 2011-02-03 |
| JP5781072B2 (ja) | 2015-09-16 |
| ES2536997T3 (es) | 2015-06-01 |
| RU2012107176A (ru) | 2013-09-10 |
| EP2459571B1 (en) | 2015-03-11 |
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