IN2012DN00369A - - Google Patents

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Publication number
IN2012DN00369A
IN2012DN00369A IN369DEN2012A IN2012DN00369A IN 2012DN00369 A IN2012DN00369 A IN 2012DN00369A IN 369DEN2012 A IN369DEN2012 A IN 369DEN2012A IN 2012DN00369 A IN2012DN00369 A IN 2012DN00369A
Authority
IN
India
Prior art keywords
oxopyrimidinone
carboxamides
fungicides
fluoro
derivatives
Prior art date
Application number
Other languages
English (en)
Inventor
Boebel Timothy
Bryan Kristy
Lorsbach Beth
Martin Timothy
Owen W
Pobanz Mark
Thornburgh Scott
Webster Jeffery
Yao Chenglin
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535294&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2012DN00369(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of IN2012DN00369A publication Critical patent/IN2012DN00369A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IN369DEN2012 2009-08-07 2010-08-05 IN2012DN00369A (enEXAMPLES)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23224509P 2009-08-07 2009-08-07
PCT/US2010/044588 WO2011017545A1 (en) 2009-08-07 2010-08-05 N1-substituted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives

Publications (1)

Publication Number Publication Date
IN2012DN00369A true IN2012DN00369A (enEXAMPLES) 2015-08-21

Family

ID=43535294

Family Applications (1)

Application Number Title Priority Date Filing Date
IN369DEN2012 IN2012DN00369A (enEXAMPLES) 2009-08-07 2010-08-05

Country Status (26)

Country Link
US (2) US8552020B2 (enEXAMPLES)
EP (1) EP2461686B1 (enEXAMPLES)
JP (1) JP5735510B2 (enEXAMPLES)
KR (1) KR101792284B1 (enEXAMPLES)
CN (1) CN102497781B (enEXAMPLES)
BR (1) BR112012002757B1 (enEXAMPLES)
CA (1) CA2769656C (enEXAMPLES)
CL (1) CL2012000312A1 (enEXAMPLES)
CO (1) CO6491115A2 (enEXAMPLES)
CR (1) CR20120032A (enEXAMPLES)
DK (1) DK2461686T3 (enEXAMPLES)
EA (1) EA020910B1 (enEXAMPLES)
EC (1) ECSP12011652A (enEXAMPLES)
ES (1) ES2552097T3 (enEXAMPLES)
HU (1) HUE027390T2 (enEXAMPLES)
IL (1) IL217950A (enEXAMPLES)
IN (1) IN2012DN00369A (enEXAMPLES)
MX (1) MX2012001617A (enEXAMPLES)
NI (1) NI201200021A (enEXAMPLES)
NZ (1) NZ597483A (enEXAMPLES)
PE (1) PE20120692A1 (enEXAMPLES)
PL (1) PL2461686T3 (enEXAMPLES)
PT (1) PT2461686E (enEXAMPLES)
UA (1) UA107671C2 (enEXAMPLES)
WO (1) WO2011017545A1 (enEXAMPLES)
ZA (1) ZA201200813B (enEXAMPLES)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8674109B2 (en) 2009-08-07 2014-03-18 Dow Agrosciences, Llc. Pesticidal compositions
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
UA106764C2 (uk) * 2009-08-07 2014-10-10 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні n1-сульфоніл-5-фторпіримідинону
HUE047711T2 (hu) * 2012-12-28 2020-05-28 Adama Makhteshim Ltd N-(szubsztituált)-5-fluor-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2H)-karboxilát származékok
WO2014105841A1 (en) * 2012-12-28 2014-07-03 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxamides derivatives
EP3689142A1 (en) * 2012-12-28 2020-08-05 Adama Makhteshim Ltd. 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
CN112094262A (zh) 2012-12-31 2020-12-18 阿达玛马克西姆股份有限公司 作为杀真菌剂的化合物
EP3862346A1 (en) 2013-12-31 2021-08-11 Adama Makhteshim Ltd. Processes for the preparation of 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)- 3,4-dihydropyrimidin-2(1h)-one
EA029457B1 (ru) 2013-12-31 2018-03-30 Адама Мактешим Лтд. Синергетические фунгицидные смеси и композиции для борьбы с грибами
JP2020527563A (ja) 2017-07-17 2020-09-10 アダマ・マクテシム・リミテッド 5−フルオロ−4−イミノ−3−メチル−1−トシル−3,4−ジヒドロピリミジン−2−オンの多形体
AU2019374510A1 (en) 2018-11-05 2021-06-17 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
CN114599639A (zh) 2019-09-23 2022-06-07 阿达玛马克西姆有限公司 用于制备5-(氟-4-亚氨基-3-甲基)-1-甲苯磺酰基-3,4-二氢嘧啶-(1h)-酮的方法

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (enEXAMPLES) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
EP0139613A1 (de) 1983-08-29 1985-05-02 Ciba-Geigy Ag N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung
JPS60123486A (ja) 1983-12-09 1985-07-02 Asahi Glass Co Ltd フルオロブラストサイジンsおよびその製法
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
EP0332579B1 (de) 1988-03-09 1994-08-10 Ciba-Geigy Ag Mittel zum Schutz von Pflanzen gegen Krankheiten
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3109012B2 (ja) 1992-06-18 2000-11-13 クミアイ化学工業株式会社 チアゾロ[5,4−d]ピリミジン誘導体及び農園芸用殺菌剤
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
US6066638A (en) * 1995-07-05 2000-05-23 E. I. Du Pont De Nemours And Company Fungicidal pyrimidinones
AU716248B2 (en) 1996-03-11 2000-02-24 Novartis Ag Pyrimidin-4-one derivatives as pesticide
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
WO2003018051A1 (en) * 2001-08-27 2003-03-06 Vic Jira Anti-fungal composition
EP1731523A4 (en) * 2004-04-01 2009-08-12 Takeda Pharmaceutical THIAZOLOPYRIMIDINDERIVAT
EP2044086A2 (en) * 2006-06-30 2009-04-08 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
ES2549046T3 (es) * 2008-01-22 2015-10-22 Dow Agrosciences, Llc Derivados de N-ciano-4-amino-5-fluoro-pirimidina como fungicidas
ES2456272T3 (es) * 2008-08-01 2014-04-21 Dow Agrosciences Llc Uso de 5-fluorocitosina como un fungicida
HUE025349T2 (en) * 2009-01-23 2016-02-29 Euro Celtique Sa Hydroxamic acid derivatives
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
UA106764C2 (uk) * 2009-08-07 2014-10-10 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні n1-сульфоніл-5-фторпіримідинону

Also Published As

Publication number Publication date
JP2013501727A (ja) 2013-01-17
PL2461686T3 (pl) 2016-04-29
CA2769656A1 (en) 2011-02-10
ZA201200813B (en) 2013-05-29
NZ597483A (en) 2014-02-28
CN102497781B (zh) 2014-12-10
JP5735510B2 (ja) 2015-06-17
US20140011824A1 (en) 2014-01-09
IL217950A0 (en) 2012-03-29
EP2461686A1 (en) 2012-06-13
BR112012002757B1 (pt) 2020-10-06
KR101792284B1 (ko) 2017-10-31
US20110034492A1 (en) 2011-02-10
EP2461686A4 (en) 2013-02-13
UA107671C2 (en) 2015-02-10
WO2011017545A1 (en) 2011-02-10
CO6491115A2 (es) 2012-07-31
CA2769656C (en) 2018-05-15
KR20120052281A (ko) 2012-05-23
CR20120032A (es) 2012-03-22
IL217950A (en) 2015-04-30
ECSP12011652A (es) 2012-03-30
CL2012000312A1 (es) 2012-10-05
ES2552097T3 (es) 2015-11-25
EP2461686B1 (en) 2015-10-07
AU2010279409A1 (en) 2012-02-02
EA020910B1 (ru) 2015-02-27
HK1171915A1 (en) 2013-04-12
PT2461686E (pt) 2015-11-18
US8552020B2 (en) 2013-10-08
BR112012002757A2 (pt) 2019-12-17
NI201200021A (es) 2012-05-22
CN102497781A (zh) 2012-06-13
US9000002B2 (en) 2015-04-07
MX2012001617A (es) 2012-04-11
HUE027390T2 (en) 2016-10-28
PE20120692A1 (es) 2012-06-08
EA201270256A1 (ru) 2012-07-30
DK2461686T3 (en) 2016-01-18

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