IL98724A0 - Antiandrogenic(3,2-c)pyrazole and(3,2-d)triazole steroids,processes for the preparation thereof and pharmaceutical compositions containing the same - Google Patents

Antiandrogenic(3,2-c)pyrazole and(3,2-d)triazole steroids,processes for the preparation thereof and pharmaceutical compositions containing the same

Info

Publication number
IL98724A0
IL98724A0 IL98724A IL9872491A IL98724A0 IL 98724 A0 IL98724 A0 IL 98724A0 IL 98724 A IL98724 A IL 98724A IL 9872491 A IL9872491 A IL 9872491A IL 98724 A0 IL98724 A0 IL 98724A0
Authority
IL
Israel
Prior art keywords
antiandrogenic
steroids
pyrazole
triazole
processes
Prior art date
Application number
IL98724A
Other languages
English (en)
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of IL98724A0 publication Critical patent/IL98724A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0036—Nitrogen-containing hetero ring
    • C07J71/0042—Nitrogen only
    • C07J71/0047—Nitrogen only at position 2(3)

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL98724A 1990-07-04 1991-07-04 Antiandrogenic(3,2-c)pyrazole and(3,2-d)triazole steroids,processes for the preparation thereof and pharmaceutical compositions containing the same IL98724A0 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4021433A DE4021433A1 (de) 1990-07-04 1990-07-04 Antiandrogene mit steroid(3,2-c)pyrazol-struktur

Publications (1)

Publication Number Publication Date
IL98724A0 true IL98724A0 (en) 1992-07-15

Family

ID=6409714

Family Applications (1)

Application Number Title Priority Date Filing Date
IL98724A IL98724A0 (en) 1990-07-04 1991-07-04 Antiandrogenic(3,2-c)pyrazole and(3,2-d)triazole steroids,processes for the preparation thereof and pharmaceutical compositions containing the same

Country Status (14)

Country Link
US (2) US5236912A (xx)
EP (1) EP0538312A1 (xx)
JP (1) JPH05508637A (xx)
CN (1) CN1059529A (xx)
AU (1) AU644201B2 (xx)
CA (1) CA2086678A1 (xx)
DE (1) DE4021433A1 (xx)
FI (1) FI925977A0 (xx)
HU (1) HUT64364A (xx)
IE (1) IE912333A1 (xx)
IL (1) IL98724A0 (xx)
PT (1) PT98199A (xx)
WO (1) WO1992000992A1 (xx)
ZA (1) ZA915193B (xx)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5879711A (en) * 1997-11-07 1999-03-09 Sequeira; Joel A. Stable antiandrogenic gel composition
WO1999061055A1 (en) 1998-05-22 1999-12-02 The Board Of Trustees Of The Leland Stanford Junior University Bifunctional molecules and therapies based thereon
WO2006116718A2 (en) 2005-04-28 2006-11-02 Proteus Biomedical, Inc. Pharma-informatics system
WO2007035716A2 (en) 2005-09-16 2007-03-29 Raptor Pharmaceutical Inc. Compositions comprising receptor-associated protein (rap) variants specific for cr-containing proteins and uses thereof
US20080051380A1 (en) 2006-08-25 2008-02-28 Auerbach Alan H Methods and compositions for treating cancer
ES2919563T3 (es) 2009-02-20 2022-07-27 Enhanx Biopharm Inc Sistema de administración de medicamentos a base de glutatión
EA024559B1 (ru) 2009-05-06 2016-09-30 Лаборэтори Скин Кэа, Инк. Композиции для нанесения на кератинизированную поверхность кожи млекопитающего и способ доставки
CN109640991A (zh) 2016-07-29 2019-04-16 詹森药业有限公司 治疗前列腺癌的方法
CN113024513A (zh) * 2021-03-22 2021-06-25 中国药科大学 新型雄激素受体降解剂、制备方法和医药用途

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL100550C (xx) * 1959-02-16
US3290293A (en) * 1961-12-01 1966-12-06 Merck & Co Inc 4-androsteno-[3, 2-c] pyrazoles
US3280112A (en) * 1963-01-28 1966-10-18 Sterling Drug Inc Steroido [2, 3-d] triazoles
US4297350A (en) * 1978-10-10 1981-10-27 The Upjohn Company Male contraceptive steroids and methods of use
US4684636A (en) * 1985-06-24 1987-08-04 Sterling Drug Inc. Antiandrogenic sulfonylsteroidopyrazoles and processes for preparation method of use and compositions thereof

Also Published As

Publication number Publication date
CA2086678A1 (en) 1992-01-05
DE4021433A1 (de) 1992-01-09
US5236912A (en) 1993-08-17
PT98199A (pt) 1992-05-29
IE912333A1 (en) 1992-01-15
CN1059529A (zh) 1992-03-18
HU9204180D0 (en) 1993-09-28
FI925977A (fi) 1992-12-31
EP0538312A1 (de) 1993-04-28
ZA915193B (en) 1992-04-29
AU644201B2 (en) 1993-12-02
HUT64364A (en) 1993-12-28
FI925977A0 (fi) 1992-12-31
US5389624A (en) 1995-02-14
WO1992000992A1 (de) 1992-01-23
AU8188091A (en) 1992-02-04
JPH05508637A (ja) 1993-12-02

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