IL97544A - Preparation of penem esters - Google Patents

Preparation of penem esters

Info

Publication number
IL97544A
IL97544A IL9754491A IL9754491A IL97544A IL 97544 A IL97544 A IL 97544A IL 9754491 A IL9754491 A IL 9754491A IL 9754491 A IL9754491 A IL 9754491A IL 97544 A IL97544 A IL 97544A
Authority
IL
Israel
Prior art keywords
formula
compound
process according
group
organic solvent
Prior art date
Application number
IL9754491A
Other languages
English (en)
Other versions
IL97544A0 (en
Inventor
Angelo Bedeschi
Walter Cabri
Marcello Marchi
Ettore Perrone
Original Assignee
Erba Carlo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Carlo Spa filed Critical Erba Carlo Spa
Publication of IL97544A0 publication Critical patent/IL97544A0/xx
Publication of IL97544A publication Critical patent/IL97544A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/09—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00—Preparation of carboxylic acid esters
    • C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
    • C07C67/307—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by introduction of halogen; by substitution of halogen atoms by other halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00—Preparation of carboxylic acid esters
    • C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
    • C07C67/313—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by introduction of doubly bound oxygen containing functional groups, e.g. carboxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
IL9754491A 1990-03-19 1991-03-14 Preparation of penem esters IL97544A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB909006114A GB9006114D0 (en) 1990-03-19 1990-03-19 Process for preparing penem esters

Publications (2)

Publication Number Publication Date
IL97544A0 IL97544A0 (en) 1992-06-21
IL97544A true IL97544A (en) 1995-05-26

Family

ID=10672850

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9754491A IL97544A (en) 1990-03-19 1991-03-14 Preparation of penem esters

Country Status (20)

Country Link
US (1) US5360904A (cs)
EP (1) EP0521018A1 (cs)
JP (1) JPH05505186A (cs)
CN (1) CN1054983A (cs)
AU (1) AU655172B2 (cs)
CA (1) CA2078684C (cs)
CZ (1) CZ279485B6 (cs)
FI (1) FI924154A7 (cs)
GB (1) GB9006114D0 (cs)
HU (1) HU212417B (cs)
IE (1) IE910866A1 (cs)
IL (1) IL97544A (cs)
MY (1) MY105332A (cs)
NO (1) NO923631L (cs)
NZ (1) NZ237433A (cs)
PT (1) PT97064B (cs)
RU (1) RU2086553C1 (cs)
WO (1) WO1991014691A1 (cs)
YU (1) YU45891A (cs)
ZA (1) ZA911984B (cs)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5399679A (en) * 1992-06-16 1995-03-21 Farmitalia Carlo Erba S.R.L. (1'R,3S,4R)4-acylthio azetidinones

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4482565A (en) * 1980-02-22 1984-11-13 Farmitalia Carlo Erba S.P.A. β-Lactam-containing antibacterial agents and β-lactamase inhibitors
DE3688960D1 (de) * 1985-09-11 1993-10-07 Ciba Geigy Synthese von Beta-Lactamverbindungen.
GB8915392D0 (en) * 1989-07-05 1989-08-23 Erba Carlo Spa Process for penems

Also Published As

Publication number Publication date
FI924154L (fi) 1992-09-16
AU655172B2 (en) 1994-12-08
GB9006114D0 (en) 1990-05-16
MY105332A (en) 1994-09-30
FI924154A0 (fi) 1992-09-16
CA2078684A1 (en) 1991-09-20
IE910866A1 (en) 1991-09-25
AU7492691A (en) 1991-10-21
CZ279485B6 (cs) 1995-05-17
NZ237433A (en) 1993-03-26
PT97064A (pt) 1991-10-31
US5360904A (en) 1994-11-01
NO923631D0 (no) 1992-09-18
NO923631L (no) 1992-09-18
WO1991014691A1 (en) 1991-10-03
PT97064B (pt) 1998-07-31
RU2086553C1 (ru) 1997-08-10
JPH05505186A (ja) 1993-08-05
IL97544A0 (en) 1992-06-21
FI924154A7 (fi) 1992-09-16
ZA911984B (en) 1991-12-24
CA2078684C (en) 2001-12-18
EP0521018A1 (en) 1993-01-07
HU9202987D0 (en) 1992-12-28
CN1054983A (zh) 1991-10-02
HU212417B (en) 1996-06-28
YU45891A (sh) 1994-05-10

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Legal Events

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RH Patent void